ID24714A - Turunan tiazolidindion tersubstitusi, proses pembuatannya dan penggunaan bahan farmasinya - Google Patents

Turunan tiazolidindion tersubstitusi, proses pembuatannya dan penggunaan bahan farmasinya

Info

Publication number: ID24714A
Authority: ID; Indonesia
Prior art keywords: tiazolidindion; derivates; substitution; production; pharmaceutical materials
Prior art date: 1997-12-16

Application number

IDW20001128A

Other languages

English (en)

Inventor

Ian Robert Lynch

Michael John Sasse

Bernadette Marie Choudary

Original Assignee

Smithkline Beecham Plc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1997-12-16

Filing date

1998-12-14

Publication date

2000-08-03

1998-12-14 Application filed by Smithkline Beecham Plc filed Critical Smithkline Beecham Plc

2000-08-03 Publication of ID24714A publication Critical patent/ID24714A/id

Links

238000000034 method Methods 0.000 title 1
238000006467 substitution reaction Methods 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/48—Drugs for disorders of the endocrine system of the pancreatic hormones
- A61P5/50—Drugs for disorders of the endocrine system of the pancreatic hormones for increasing or potentiating the activity of insulin

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Diabetes (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Veterinary Medicine (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Public Health (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Obesity (AREA)
Hematology (AREA)
Endocrinology (AREA)
Emergency Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Thiazole And Isothizaole Compounds (AREA)
Medicines Containing Material From Animals Or Micro-Organisms (AREA)

IDW20001128A 1997-12-16 1998-12-14 Turunan tiazolidindion tersubstitusi, proses pembuatannya dan penggunaan bahan farmasinya ID24714A (id)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
GBGB9726563.1A GB9726563D0 (en)	1997-12-16	1997-12-16	Novel pharmaceutical

Publications (1)

Publication Number	Publication Date
ID24714A true ID24714A (id)	2000-08-03

Family

ID=10823691

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
IDW20001128A ID24714A (id)	1997-12-16	1998-12-14	Turunan tiazolidindion tersubstitusi, proses pembuatannya dan penggunaan bahan farmasinya

Country Status (37)

Country	Link
US (4)	US20020133016A1 (id)
EP (1)	EP1042321A1 (id)
JP (1)	JP2002508371A (id)
KR (1)	KR100549141B1 (id)
CN (3)	CN1285831A (id)
AP (1)	AP1363A (id)
AR (2)	AR017211A1 (id)
AU (2)	AU2272299A (id)
BG (1)	BG64850B1 (id)
BR (1)	BR9813598A (id)
CA (1)	CA2314967A1 (id)
CO (1)	CO4990943A1 (id)
CZ (1)	CZ300081B6 (id)
DZ (1)	DZ2679A1 (id)
EA (1)	EA002833B1 (id)
EG (1)	EG22250A (id)
GB (1)	GB9726563D0 (id)
HR (1)	HRP20000404A2 (id)
HU (1)	HUP0102292A3 (id)
ID (1)	ID24714A (id)
IL (2)	IL136425A (id)
MA (1)	MA26581A1 (id)
MY (1)	MY128573A (id)
NO (1)	NO317255B1 (id)
NZ (1)	NZ504703A (id)
OA (1)	OA11900A (id)
PE (1)	PE20000125A1 (id)
PL (1)	PL341213A1 (id)
RS (1)	RS50080B (id)
SA (1)	SA99200200B1 (id)
SK (1)	SK286422B6 (id)
TR (2)	TR200001793T2 (id)
TW (1)	TW487709B (id)
UA (1)	UA66821C2 (id)
UY (2)	UY25309A1 (id)
WO (1)	WO1999031093A1 (id)
ZA (1)	ZA9811504B (id)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
USRE39384E1 (en)	1993-09-01	2006-11-07	Smithkline Beecham P.L.C.	Substituted thiazolidinedione derivatives
US20020137940A1 (en)	1997-12-16	2002-09-26	Smithkline Beecham P.L.C.	5-[4-[2-(N-methyl-N-(2-pyridyl)amino)ethoxy]benzyl]thiazolidine-2, 4-dione, maleic acid salt, hydrate as pharmaceutical
GB9726568D0 (en)	1997-12-16	1998-02-11	Smithkline Beecham Plc	Novel pharmaceutical
US6664278B2 (en)	1997-12-16	2003-12-16	Smithkline Beecham P.L.C.	Hydrate of 5-[4-[2-(N-methyl-N-(2-pyridil)amino)ethoxy]benzyl]thiazolidine-2,4-dione maleic acid salt
GB9909041D0 (en) *	1999-04-20	1999-06-16	Smithkline Beecham Plc	Novel pharmaceutical
US20040248945A1 (en)	1999-04-23	2004-12-09	Smithkline Beecham P.L.C.	Thiazolidinedione derivative and its use as antidiabetic
HK1045152A1 (zh) *	1999-04-23	2002-11-15	Smithkline Beecham Plc	噻唑烷二酮衍生物及其用作抗糖尿病藥的應用
PL351684A1 (en) *	1999-04-23	2003-06-02	Smithkline Beecham Plc	Polymorph of 5−[4−[2− (n−methyl−n−( 2−pyridyl)amino) ethoxy]benzyl] thiazolidine−2,4−dione, maleic acid salt
AU765498B2 (en) *	1999-04-23	2003-09-18	Smithkline Beecham Plc	Novel pharmaceutical
GB0014005D0 (en) *	2000-06-08	2000-08-02	Smithkline Beecham Plc	Novel pharmaceutical
GB0021784D0 (en) *	2000-09-05	2000-10-18	Smithkline Beecham Plc	Novel pharmaceutical
GB0021978D0 (en) *	2000-09-07	2000-10-25	Smithkline Beecham Plc	Novel pharmaceutical
AU2002350965A1 (en) *	2001-12-13	2003-06-23	Smithkline Beecham Plc	Toluenesulfonate hydrates of a thiazolidinedione derivative
GB0129876D0 (en) *	2001-12-13	2002-02-06	Smithkline Beecham Plc	Novel pharmaceutical
KR100450700B1 (ko) *	2002-03-22	2004-10-01	주식회사종근당	티아졸리딘디온 유도체 화합물 및 이를 함유하는 약제학적조성물
EP1468997A3 (en) *	2003-04-18	2004-11-03	CHEMI S.p.A.	Polymorphous forms of rosiglitazone maleate
GB2405403A (en) *	2003-08-29	2005-03-02	Cipla Ltd	Rosiglitazone maleate of particular polymorphic forms and methods of preparing rosiglitazone free base
EP1841414A1 (en) *	2003-12-31	2007-10-10	Alpharma, Inc.	Rosiglitazone and metformin formulations
WO2005065654A2 (en) *	2003-12-31	2005-07-21	Alpharma, Inc.	Rosiglitazone formulations
ITMI20041537A1 (it) *	2004-07-28	2004-10-28	Chemi Spa	Nuova forma polimorfa del rosiglitazone maleato
CZ298424B6 (cs) *	2005-05-24	2007-09-26	Zentiva, A. S.	Zpusob krystalizace rosiglitazonu a jeho derivátuze smesných rozpouštedel
US7435741B2 (en) *	2006-05-09	2008-10-14	Teva Pharmaceutical Industries, Ltd.	2-N{5-[[4-[2-(methyl-2-pyridinylamino) ethoxy] phenyl]methyl]-2,4-thiazolidinedione} butanedioic acid, methods of preparation and compositions with rosiglitazone maleate
EP2184055A1 (en)	2008-11-07	2010-05-12	LEK Pharmaceuticals d.d.	Process for preparing solid dosage forms of rosiglitazone maleate

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US6288095B1 (en) *	1987-09-04	2001-09-11	Beecham Group P.L.C.	Compounds
ATE186724T1 (de) *	1987-09-04	1999-12-15	Beecham Group Plc	Substituierte thiazolidindionderivate
GB8820389D0 (en) *	1988-08-26	1988-09-28	Beecham Group Plc	Novel compounds
GB9124513D0 (en) *	1991-11-19	1992-01-08	Smithkline Beecham Plc	Novel process
GB9218830D0 (en) *	1992-09-05	1992-10-21	Smithkline Beecham Plc	Novel compounds
US5741803A (en) *	1992-09-05	1998-04-21	Smithkline Beecham Plc	Substituted thiazolidinedionle derivatives
JPH09512249A (ja) *	1994-02-10	1997-12-09	スミスクライン・ビーチャム・パブリック・リミテッド・カンパニー	腎臓疾患を治療するためのインスリンセンシタイザーの使用
DE4404198A1 (de)	1994-02-10	1995-08-17	Henkel Kgaa	2-Fluor-6-nitroaniline
US20020137940A1 (en)	1997-12-16	2002-09-26	Smithkline Beecham P.L.C.	5-[4-[2-(N-methyl-N-(2-pyridyl)amino)ethoxy]benzyl]thiazolidine-2, 4-dione, maleic acid salt, hydrate as pharmaceutical
US6664278B2 (en)	1997-12-16	2003-12-16	Smithkline Beecham P.L.C.	Hydrate of 5-[4-[2-(N-methyl-N-(2-pyridil)amino)ethoxy]benzyl]thiazolidine-2,4-dione maleic acid salt
MXPA03002580A (es)	2000-09-26	2003-10-15	Cord Janet I	Nuevas formas polimorficas de maleato de 5-(4-(2-(n-metil-n-(2-piridil) amino)etoxi)bencil) tiazolidin-2, 4-diona y proceso para su preparacion.

1997
- 1997-12-16 GB GBGB9726563.1A patent/GB9726563D0/en not_active Ceased
1998
- 1998-12-14 SK SK918-2000A patent/SK286422B6/sk not_active IP Right Cessation
- 1998-12-14 OA OA00000177A patent/OA11900A/en unknown
- 1998-12-14 RS YUP-364/00A patent/RS50080B/sr unknown
- 1998-12-14 BR BR9813598-8A patent/BR9813598A/pt not_active Application Discontinuation
- 1998-12-14 EA EA200000656A patent/EA002833B1/ru not_active IP Right Cessation
- 1998-12-14 CN CN98812091A patent/CN1285831A/zh active Pending
- 1998-12-14 CZ CZ20002206A patent/CZ300081B6/cs not_active IP Right Cessation
- 1998-12-14 UA UA2000063483A patent/UA66821C2/uk unknown
- 1998-12-14 IL IL13642598A patent/IL136425A/en unknown
- 1998-12-14 PL PL98341213A patent/PL341213A1/xx not_active Application Discontinuation
- 1998-12-14 AP APAP/P/2000/001829A patent/AP1363A/en active
- 1998-12-14 ID IDW20001128A patent/ID24714A/id unknown
- 1998-12-14 WO PCT/EP1998/008153 patent/WO1999031093A1/en not_active Ceased
- 1998-12-14 HR HR20000404A patent/HRP20000404A2/hr not_active Application Discontinuation
- 1998-12-14 CN CNA2008100919932A patent/CN101318957A/zh active Pending
- 1998-12-14 MA MA25391A patent/MA26581A1/fr unknown
- 1998-12-14 TR TR2000/01793T patent/TR200001793T2/xx unknown
- 1998-12-14 IL IL16084798A patent/IL160847A0/xx unknown
- 1998-12-14 NZ NZ504703A patent/NZ504703A/xx unknown
- 1998-12-14 JP JP2000539017A patent/JP2002508371A/ja not_active Withdrawn
- 1998-12-14 HU HU0102292A patent/HUP0102292A3/hu unknown
- 1998-12-14 AU AU22722/99A patent/AU2272299A/en not_active Abandoned
- 1998-12-14 KR KR1020007006514A patent/KR100549141B1/ko not_active Expired - Fee Related
- 1998-12-14 CA CA002314967A patent/CA2314967A1/en not_active Abandoned
- 1998-12-14 CN CNA2008100919928A patent/CN101318956A/zh active Pending
- 1998-12-14 EP EP98966320A patent/EP1042321A1/en not_active Withdrawn
- 1998-12-15 AR ARP980106364A patent/AR017211A1/es unknown
- 1998-12-15 UY UY25309A patent/UY25309A1/es not_active IP Right Cessation
- 1998-12-15 UY UY25306A patent/UY25306A1/es unknown
- 1998-12-15 MY MYPI98005673A patent/MY128573A/en unknown
- 1998-12-15 DZ DZ980289A patent/DZ2679A1/xx active
- 1998-12-15 AR ARP980106368A patent/AR016161A1/es not_active Application Discontinuation
- 1998-12-15 EG EG155398A patent/EG22250A/xx active
- 1998-12-15 ZA ZA9811504A patent/ZA9811504B/xx unknown
- 1998-12-16 TW TW087121120A patent/TW487709B/zh not_active IP Right Cessation
- 1998-12-16 CO CO98074832A patent/CO4990943A1/es unknown
- 1998-12-16 PE PE1998001231A patent/PE20000125A1/es not_active Application Discontinuation
- 1998-12-16 TR TR1998/02624A patent/TR199802624A2/xx unknown
1999
- 1999-05-31 SA SA99200200A patent/SA99200200B1/ar unknown
2000
- 2000-06-15 NO NO20003070A patent/NO317255B1/no not_active IP Right Cessation
- 2000-07-13 BG BG104606A patent/BG64850B1/bg unknown
2002
- 2002-02-08 US US10/071,339 patent/US20020133016A1/en not_active Abandoned
- 2002-03-20 AU AU27538/02A patent/AU770818B2/en not_active Ceased
2003
- 2003-01-30 US US10/354,365 patent/US20030139604A1/en not_active Abandoned
2005
- 2005-08-17 US US11/205,426 patent/US20050288513A1/en not_active Abandoned
2006
- 2006-09-28 US US11/536,313 patent/US7368574B2/en not_active Expired - Fee Related

Also Published As

Publication number	Publication date
NZ504703A (en)	2002-12-20
UY25306A1 (es)	2000-12-29
UY25309A1 (es)	1999-07-19
BG64850B1 (bg)	2006-06-30
YU36400A (sh)	2003-12-31
JP2002508371A (ja)	2002-03-19
BR9813598A (pt)	2000-10-10
AP1363A (en)	2005-01-21
AU2753802A (en)	2002-05-16
AU770818B2 (en)	2004-03-04
NO317255B1 (no)	2004-09-27
HRP20000404A2 (en)	2000-12-31
WO1999031093A1 (en)	1999-06-24
GB9726563D0 (en)	1998-02-11
SK9182000A3 (en)	2000-12-11
CN101318956A (zh)	2008-12-10
AP2000001829A0 (en)	2000-06-30
KR100549141B1 (ko)	2006-02-03
SK286422B6 (sk)	2008-09-05
CZ20002206A3 (cs)	2000-12-13
PE20000125A1 (es)	2000-03-03
CN101318957A (zh)	2008-12-10
CA2314967A1 (en)	1999-06-24
US20070037859A1 (en)	2007-02-15
OA11900A (en)	2006-04-10
EA002833B1 (ru)	2002-10-31
CN1285831A (zh)	2001-02-28
AR017211A1 (es)	2001-08-22
TW487709B (en)	2002-05-21
CZ300081B6 (cs)	2009-01-28
BG104606A (en)	2001-02-28
ZA9811504B (en)	2000-06-15
US20050288513A1 (en)	2005-12-29
HUP0102292A2 (hu)	2002-05-29
US20020133016A1 (en)	2002-09-19
SA99200200B1 (ar)	2006-11-11
HUP0102292A3 (en)	2003-12-29
RS50080B (sr)	2009-01-22
TR200001793T2 (tr)	2000-10-23
UA66821C2 (uk)	2004-06-15
US20030139604A1 (en)	2003-07-24
EA200000656A1 (ru)	2000-12-25
AU2272299A (en)	1999-07-05
PL341213A1 (en)	2001-03-26
EP1042321A1 (en)	2000-10-11
IL136425A0 (en)	2001-06-14
TR199802624A3 (tr)	1999-10-21
IL136425A (en)	2004-08-31
US7368574B2 (en)	2008-05-06
MA26581A1 (fr)	2004-12-20
EG22250A (en)	2002-11-30
NO20003070L (no)	2000-06-15
AR016161A1 (es)	2001-06-20
CO4990943A1 (es)	2000-12-26
NO20003070D0 (no)	2000-06-15
TR199802624A2 (xx)	1999-10-21
IL160847A0 (en)	2004-08-31
KR20010033140A (ko)	2001-04-25
DZ2679A1 (fr)	2003-03-29
MY128573A (en)	2007-02-28

Publication	Publication Date	Title
ID22821A (id)	1999-12-09	Turunan sulfonamida, proses pembuatannya dan penggunaannya sebagai obat
ID26207A (id)	2000-12-07	ESTRATRIENA TERSUBSTITUSI 11β-HALOGEN-7 αTERSUBSTITUTASI, PROSES UNTUK MEMPRODUKSI SEDIAAN FARMASI YANG MENGANDUNG ESTRATRIENA 11β-HALOGEN-7 αINI DAN JUGA PENGGUNAANNYA UNTUK PRODUKSI ZAT-ZAT FARMASI
ID27408A (id)	2001-04-05	Benda penyerap dan proses pembuatannya
ID21459A (id)	1999-06-17	Produk pembersih dan proses produksinya
ID26172A (id)	2000-11-30	Proses pembuatan surfaktan-surfaktan alkilbenzenasulfonat dan produk-produknya
ID27757A (id)	2001-04-26	Indolinona-indolinona tersubstitusi baru, preparasi dan penggunaannya sebagai obat
AU742593C (en)	2004-04-29	Disubstituted bicyclic heterocycles, their production and use as medicaments
NO20021714L (no)	2000-05-11	2-fenyl-substituerte imidazotriazinoner, fremgangsmåte for fremstilling derav samt anvendelse av forbindelsene
ID25528A (id)	2000-10-12	Karboksamidotiazol tersubstitusi, pembuatannya dan komposisi farmasi yang mengandungnya
HUP0001153A3 (en)	2000-12-28	Chemically modified polypeptides, process for producing thereof, pharmaceutical compositions comprising these polypeptides and their use
ID17307A (id)	1997-12-18	Komposisi oral dan proses pembuatannya.
ID23600A (id)	1995-11-30	Turunan tiazolidin dan oksazolidin, pembuatan dan penggunaannya untuk pengobatan (pecahan dari p-950453)
ID30299A (id)	2001-11-22	Turunan oksazolidinon, proses pembuatannya dan komposisi farmasi yang mengandungnya
ID22528A (id)	1999-10-28	Komposisi farmasi fenofibrat yang memiliki biovabilitas tinggi dan metoda pembuatannya
ID26351A (id)	2000-12-14	Isosianat-isosianat oligomerik tersumbat, pembuatan dan penggunaannya
ID17810A (id)	1998-01-29	Turunan-turunan 2,4-tiazolidindion tersubstitusi baru, proses untuk pembuatannya dan komposisi farmasi yang mengandungnya
ID20137A (id)	1998-10-08	Turunan propanolamina, proses pembuatannya, sediaan farmasi yang mengandung senyawa ini, dan penggunannya
ID22911A (id)	1999-12-16	Turunan-turunan triazol baru, proses pembuatan dan komposisi-komposisi farmasi yang mengandungnya
IS5331A (is)	1999-12-30	Ný lyfjablanda
ID24173A (id)	2000-07-13	1,2,3,4,5,6 heksahidro-2-6-metano-3-benzazosin-10-ol, proses pembuatan dan penggunannya untuk obat-obatan
ID26985A (id)	2001-02-22	Amina-amina polisiklik tiazolidin-2-ilidena, proses pembuatannya, dan penggunaannya a sebagai bahas farmasi
ID26344A (id)	2000-12-14	Pakaian atas sekali pakai dan proses pembuatannya
ID20967A (id)	1999-04-01	Kroman tersubstitusi sulfonamida, proses pembuatannya, penggunaannya sebagai obat, dan sediaan farmasi yang mengandung bahan tersebut
NO993912L (no)	1999-08-13	FremgangsmÕte for fremstilling av eprosartan
NO993913D0 (no)	1999-08-13	Fremgangsmåte for fremstilling av eprosartan