ID26208A - Turunan-turunan asam amino amidino terhalogenasi yang berguna sebagai penghambat sintase nitrat oksida - Google Patents
Turunan-turunan asam amino amidino terhalogenasi yang berguna sebagai penghambat sintase nitrat oksidaInfo
- Publication number
- ID26208A ID26208A IDW20001739A ID20001739A ID26208A ID 26208 A ID26208 A ID 26208A ID W20001739 A IDW20001739 A ID W20001739A ID 20001739 A ID20001739 A ID 20001739A ID 26208 A ID26208 A ID 26208A
- Authority
- ID
- Indonesia
- Prior art keywords
- acid
- synthase
- resident
- halogenation
- drugs
- Prior art date
Links
- 239000002253 acid Substances 0.000 title 2
- -1 AMINO AMIDINO Chemical class 0.000 title 1
- 229910002651 NO3 Inorganic materials 0.000 title 1
- NHNBFGGVMKEFGY-UHFFFAOYSA-N Nitrate Chemical compound [O-][N+]([O-])=O NHNBFGGVMKEFGY-UHFFFAOYSA-N 0.000 title 1
- 239000003814 drug Substances 0.000 title 1
- 229940079593 drug Drugs 0.000 title 1
- 230000026030 halogenation Effects 0.000 title 1
- 238000005658 halogenation reaction Methods 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
- C07D333/24—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C257/00—Compounds containing carboxyl groups, the doubly-bound oxygen atom of a carboxyl group being replaced by a doubly-bound nitrogen atom, this nitrogen atom not being further bound to an oxygen atom, e.g. imino-ethers, amidines
- C07C257/10—Compounds containing carboxyl groups, the doubly-bound oxygen atom of a carboxyl group being replaced by a doubly-bound nitrogen atom, this nitrogen atom not being further bound to an oxygen atom, e.g. imino-ethers, amidines with replacement of the other oxygen atom of the carboxyl group by nitrogen atoms, e.g. amidines
- C07C257/14—Compounds containing carboxyl groups, the doubly-bound oxygen atom of a carboxyl group being replaced by a doubly-bound nitrogen atom, this nitrogen atom not being further bound to an oxygen atom, e.g. imino-ethers, amidines with replacement of the other oxygen atom of the carboxyl group by nitrogen atoms, e.g. amidines having carbon atoms of amidino groups bound to acyclic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
- C07C323/50—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton
- C07C323/51—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton
- C07C323/57—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being further substituted by nitrogen atoms, not being part of nitro or nitroso groups
- C07C323/58—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being further substituted by nitrogen atoms, not being part of nitro or nitroso groups with amino groups bound to the carbon skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2601/00—Systems containing only non-condensed rings
- C07C2601/02—Systems containing only non-condensed rings with a three-membered ring
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Physical Education & Sports Medicine (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Heterocyclic Compounds Containing Sulfur Atoms (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US3828498A | 1998-03-11 | 1998-03-11 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ID26208A true ID26208A (id) | 2000-11-07 |
Family
ID=21899068
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IDW20001739A ID26208A (id) | 1998-03-11 | 1999-03-04 | Turunan-turunan asam amino amidino terhalogenasi yang berguna sebagai penghambat sintase nitrat oksida |
Country Status (35)
| Country | Link |
|---|---|
| US (1) | US6344483B1 (id) |
| EP (2) | EP1062201B1 (id) |
| JP (1) | JP2002506056A (id) |
| KR (1) | KR20010034598A (id) |
| CN (1) | CN1171861C (id) |
| AP (1) | AP2000001900A0 (id) |
| AR (1) | AR018159A1 (id) |
| AT (1) | ATE277894T1 (id) |
| AU (1) | AU746235B2 (id) |
| BG (1) | BG104766A (id) |
| BR (1) | BR9908702A (id) |
| CA (1) | CA2322873A1 (id) |
| CU (1) | CU23047A3 (id) |
| DE (1) | DE69920670T2 (id) |
| EA (1) | EA200000826A1 (id) |
| EE (1) | EE200000519A (id) |
| ES (1) | ES2239839T3 (id) |
| GE (1) | GEP20043179B (id) |
| HR (1) | HRP20000595A2 (id) |
| HU (1) | HUP0101467A3 (id) |
| ID (1) | ID26208A (id) |
| IL (1) | IL137654A0 (id) |
| IS (1) | IS5583A (id) |
| NO (1) | NO20004531L (id) |
| NZ (1) | NZ506721A (id) |
| OA (1) | OA11901A (id) |
| PL (1) | PL343380A1 (id) |
| PT (1) | PT1062201E (id) |
| SI (1) | SI1062201T1 (id) |
| SK (1) | SK13012000A3 (id) |
| TR (1) | TR200002605T2 (id) |
| UA (1) | UA67767C2 (id) |
| WO (1) | WO1999046240A2 (id) |
| YU (1) | YU52200A (id) |
| ZA (1) | ZA991894B (id) |
Families Citing this family (23)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DK1265859T3 (da) | 2000-03-24 | 2006-05-01 | Pharmacia Corp | Amidinoforbindelser der er nyttige som nitrogenoxidsyntaseinhibitorer |
| US6787668B2 (en) | 2000-04-13 | 2004-09-07 | Pharmacia Corporation | 2-amino-4,5 heptenoic acid derivatives useful as nitric oxide synthase inhibitors |
| AR030416A1 (es) | 2000-04-13 | 2003-08-20 | Pharmacia Corp | COMPUESTO DERIVADO HALOGENADO DEL ACIDO 2-AMINO-3,4 HEPTENOICO, COMPOSICION FARMACEUTICA QUE LO COMPRENDE Y SU USO EN LA FABRICACION DE UN MEDICAMENTO uTIL COMO INHIBIDOR DE LA OXIDO NITRICO SINTETASA |
| US6956131B2 (en) * | 2000-04-13 | 2005-10-18 | Pharmacia Corporation | 2-amino-3, 4 heptenoic compounds useful as nitric oxide synthase inhibitors |
| US6545170B2 (en) | 2000-04-13 | 2003-04-08 | Pharmacia Corporation | 2-amino-5, 6 heptenoic acid derivatives useful as nitric oxide synthase inhibitors |
| AR032318A1 (es) * | 2000-04-13 | 2003-11-05 | Pharmacia Corp | Compuesto derivado halogenado del acido 2-amino-5,6 heptenoico; composicion farmaceutica que lo comprende y su uso en la fabricacion de un medicamento util como inhibidor de la oxido nitrico sintetasa |
| AR034120A1 (es) * | 2000-04-13 | 2004-02-04 | Pharmacia Corp | Compuesto derivado halogenado del acido 2-amino-4,5 heptenoico, composicion farmaceutica que lo comprende y el uso de dicho compuesto y dicha composicion en la fabricacion de un medicamento para inhibir o modular la sintesis de acido nitrico |
| AR031129A1 (es) | 2000-09-15 | 2003-09-10 | Pharmacia Corp | Derivados de los acidos 2-amino-2-alquil-4-hexenoico y -hexinoico utiles como inhibidores de oxido nitrico sintetasa |
| AR035585A1 (es) * | 2000-09-15 | 2004-06-16 | Pharmacia Corp | Derivados del acido 2-amino-2-alquil-4-heptenoico, composicion farmaceutica y su uso en la fabricacion de medicamentos |
| AR031608A1 (es) * | 2000-09-15 | 2003-09-24 | Pharmacia Corp | Derivados de los acidos 2-amino-2-alquil-3-hexenoico y -hexinoico utiles como inhibidores de oxido nitrico sintetasa |
| AR031609A1 (es) * | 2000-09-15 | 2003-09-24 | Pharmacia Corp | Derivados de acido 2-amino-2-alquil-3 heptenoico y heptinoico utiles como inhibidores de oxido nitrico sintetasa |
| GB0031179D0 (en) | 2000-12-21 | 2001-01-31 | Glaxo Group Ltd | Nitric oxide synthase inhibitors |
| US6613280B2 (en) * | 2001-03-20 | 2003-09-02 | Therox, Inc. | Disposable cartridge for producing gas-enriched fluids |
| US6582387B2 (en) * | 2001-03-20 | 2003-06-24 | Therox, Inc. | System for enriching a bodily fluid with a gas |
| US7012098B2 (en) | 2001-03-23 | 2006-03-14 | Pharmacia Corporation | Inhibitors of inducible nitric oxide synthase for chemoprevention and treatment of cancers |
| US20040087653A1 (en) * | 2002-05-16 | 2004-05-06 | Manning Pamela T. | Methods for the treatment of respiratory diseases and conditions with a selective iNOS inhibitor and a PDE inhibitor and compositions therefor |
| MX2007007590A (es) | 2004-12-22 | 2007-12-10 | Ambrx Inc | Composiciones que contienen, metodos que involucran y usos de aminoacidos no naturales y polipeptidos. |
| MX2007011409A (es) * | 2005-03-14 | 2008-02-22 | Johnson & Johnson | Procedimiento de preparacion de moduladores opioides. |
| HRP20110404T1 (hr) * | 2005-11-08 | 2011-08-31 | Ambrx | Ubrzivači za modifikaciju ne-prirodnih aminokiselina i polipeptida ne-prirodnih aminokiselina |
| ES2529065T3 (es) * | 2005-12-14 | 2015-02-16 | Ambrx, Inc. | Composiciones que contienen, procedimientos que implican y usos de aminoácidos no naturales y polipéptidos |
| KR101103720B1 (ko) * | 2011-06-02 | 2012-01-11 | 한국건설기술연구원 | 자연환기에 의한 중공층의 온도제어가 가능한 일체형 다중유리 복합창짝 |
| CN105744944B (zh) | 2013-09-09 | 2020-07-07 | 卡尼姆盖德治疗学公司 | 免疫系统调节器 |
| WO2016144650A1 (en) | 2015-03-06 | 2016-09-15 | Canimguide Therapeutics Ab | Immune system modulators and compositions |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB9127376D0 (en) * | 1991-12-24 | 1992-02-19 | Wellcome Found | Amidino derivatives |
| GB9312761D0 (en) * | 1993-06-21 | 1993-08-04 | Wellcome Found | Amino acid derivatives |
| SI0765308T1 (sl) | 1994-06-15 | 2000-08-31 | The Wellcome Foundation Limited | Encimski inhibitorji |
| GB9425701D0 (en) * | 1994-12-20 | 1995-02-22 | Wellcome Found | Enzyme inhibitors |
| US5945408A (en) * | 1996-03-06 | 1999-08-31 | G.D. Searle & Co. | Hydroxyanidino derivatives useful as nitric oxide synthase inhibitors |
| US5981511A (en) * | 1996-03-06 | 1999-11-09 | G.D. Searle & Co. | Hydroxyamidino derivatives useful as nitric oxide synthase inhibitors |
-
1999
- 1999-03-04 PL PL99343380A patent/PL343380A1/xx unknown
- 1999-03-04 DE DE69920670T patent/DE69920670T2/de not_active Expired - Fee Related
- 1999-03-04 CU CU20000199A patent/CU23047A3/es unknown
- 1999-03-04 CA CA002322873A patent/CA2322873A1/en not_active Abandoned
- 1999-03-04 AP APAP/P/2000/001900A patent/AP2000001900A0/en unknown
- 1999-03-04 GE GEAP19995542A patent/GEP20043179B/en unknown
- 1999-03-04 OA OA1200000239A patent/OA11901A/en unknown
- 1999-03-04 EP EP99908324A patent/EP1062201B1/en not_active Expired - Lifetime
- 1999-03-04 HU HU0101467A patent/HUP0101467A3/hu unknown
- 1999-03-04 AU AU27786/99A patent/AU746235B2/en not_active Ceased
- 1999-03-04 PT PT99908324T patent/PT1062201E/pt unknown
- 1999-03-04 JP JP2000535621A patent/JP2002506056A/ja active Pending
- 1999-03-04 WO PCT/US1999/003728 patent/WO1999046240A2/en not_active Ceased
- 1999-03-04 ID IDW20001739A patent/ID26208A/id unknown
- 1999-03-04 TR TR2000/02605T patent/TR200002605T2/xx unknown
- 1999-03-04 ES ES99908324T patent/ES2239839T3/es not_active Expired - Lifetime
- 1999-03-04 EE EEP200000519A patent/EE200000519A/xx unknown
- 1999-03-04 NZ NZ506721A patent/NZ506721A/en unknown
- 1999-03-04 SK SK1301-2000A patent/SK13012000A3/sk unknown
- 1999-03-04 CN CNB998037907A patent/CN1171861C/zh not_active Expired - Fee Related
- 1999-03-04 IL IL13765499A patent/IL137654A0/xx unknown
- 1999-03-04 KR KR1020007010096A patent/KR20010034598A/ko not_active Ceased
- 1999-03-04 AT AT99908324T patent/ATE277894T1/de not_active IP Right Cessation
- 1999-03-04 EA EA200000826A patent/EA200000826A1/ru unknown
- 1999-03-04 BR BR9908702-2A patent/BR9908702A/pt not_active Application Discontinuation
- 1999-03-04 HR HR20000595A patent/HRP20000595A2/hr not_active Application Discontinuation
- 1999-03-04 YU YU52200A patent/YU52200A/sh unknown
- 1999-03-04 SI SI9930718T patent/SI1062201T1/xx unknown
- 1999-03-04 US US09/402,953 patent/US6344483B1/en not_active Expired - Fee Related
- 1999-03-04 EP EP20040001236 patent/EP1415982A1/en not_active Withdrawn
- 1999-03-09 ZA ZA9901894A patent/ZA991894B/xx unknown
- 1999-03-11 AR ARP990101062A patent/AR018159A1/es unknown
- 1999-04-03 UA UA2000095233A patent/UA67767C2/uk unknown
-
2000
- 2000-08-04 IS IS5583A patent/IS5583A/is unknown
- 2000-09-11 NO NO20004531A patent/NO20004531L/no not_active Application Discontinuation
- 2000-09-14 BG BG104766A patent/BG104766A/bg unknown
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