ID29514A - 2-ARIL-3-(HETEROARIL)-IMIDAZO [1,2-a]PIRIMIDIN TERSUBSTITUSI, DAN METODE-METODE DAN KOMPOSISI-KOMPOSISI FARMASI YANG TERKAIT - Google Patents

2-ARIL-3-(HETEROARIL)-IMIDAZO [1,2-a]PIRIMIDIN TERSUBSTITUSI, DAN METODE-METODE DAN KOMPOSISI-KOMPOSISI FARMASI YANG TERKAIT

Info

Publication number: ID29514A
Authority: ID; Indonesia
Prior art keywords: heteroaril; aril; imidazo; compositions; substituted pyrimidine
Prior art date: 1999-11-10

Application number

IDW00200101720A

Other languages

English (en)

Inventor

John H Dodd

James R Henry

Kenneth C Rupert

Original Assignee

Ortho Mcneil Pharmacetical Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1999-11-10

Filing date

2000-10-27

Publication date

2001-09-06

2000-10-27 Application filed by Ortho Mcneil Pharmacetical Inc filed Critical Ortho Mcneil Pharmacetical Inc

2001-09-06 Publication of ID29514A publication Critical patent/ID29514A/id

Links

CZPWVGJYEJSRLH-UHFFFAOYSA-N Pyrimidine Chemical class C1=CN=CN=C1 CZPWVGJYEJSRLH-UHFFFAOYSA-N 0.000 title 1
239000000203 mixture Substances 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/02—Stomatological preparations, e.g. drugs for caries, aphtae, periodontitis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/18—Drugs for disorders of the alimentary tract or the digestive system for pancreatic disorders, e.g. pancreatic enzymes
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/06—Antipsoriatics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/14—Drugs for dermatological disorders for baldness or alopecia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmacology & Pharmacy (AREA)
General Chemical & Material Sciences (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Immunology (AREA)
Rheumatology (AREA)
Physical Education & Sports Medicine (AREA)
Oncology (AREA)
Diabetes (AREA)
Orthopedic Medicine & Surgery (AREA)
Virology (AREA)
Neurosurgery (AREA)
Neurology (AREA)
Biomedical Technology (AREA)
Communicable Diseases (AREA)
Pain & Pain Management (AREA)
Heart & Thoracic Surgery (AREA)
Dermatology (AREA)
Pulmonology (AREA)
Cardiology (AREA)
Obesity (AREA)
Hospice & Palliative Care (AREA)
Urology & Nephrology (AREA)
Molecular Biology (AREA)
Tropical Medicine & Parasitology (AREA)
Hematology (AREA)
Endocrinology (AREA)
Vascular Medicine (AREA)
Psychiatry (AREA)

IDW00200101720A 1999-11-10 2000-10-27 2-ARIL-3-(HETEROARIL)-IMIDAZO [1,2-a]PIRIMIDIN TERSUBSTITUSI, DAN METODE-METODE DAN KOMPOSISI-KOMPOSISI FARMASI YANG TERKAIT ID29514A (id)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US16470099P	1999-11-10	1999-11-10

Publications (1)

Publication Number	Publication Date
ID29514A true ID29514A (id)	2001-09-06

Family

ID=22595694

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
IDW00200101720A ID29514A (id)	1999-11-10	2000-10-27	2-ARIL-3-(HETEROARIL)-IMIDAZO [1,2-a]PIRIMIDIN TERSUBSTITUSI, DAN METODE-METODE DAN KOMPOSISI-KOMPOSISI FARMASI YANG TERKAIT

Country Status (27)

Country	Link
US (1)	US6610697B1 (id)
EP (1)	EP1140939B1 (id)
JP (1)	JP2003513977A (id)
KR (1)	KR20010089805A (id)
CN (1)	CN1255406C (id)
AR (1)	AR026410A1 (id)
AT (1)	ATE288915T1 (id)
AU (1)	AU784484B2 (id)
BG (1)	BG65106B1 (id)
BR (1)	BR0007447A (id)
CA (1)	CA2361139A1 (id)
CZ (1)	CZ20012494A3 (id)
DE (1)	DE60018037T2 (id)
ES (1)	ES2237470T3 (id)
HK (1)	HK1043591B (id)
HU (1)	HUP0200207A3 (id)
ID (1)	ID29514A (id)
IL (1)	IL144238A (id)
MX (1)	MXPA01007019A (id)
NO (1)	NO320422B1 (id)
NZ (1)	NZ512957A (id)
PL (1)	PL348924A1 (id)
PT (1)	PT1140939E (id)
RU (1)	RU2264403C2 (id)
SK (1)	SK9892001A3 (id)
UA (1)	UA70350C2 (id)
WO (1)	WO2001034605A1 (id)

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GB0124933D0 (en)	2001-10-17	2001-12-05	Glaxo Group Ltd	Chemical compounds
GB0124934D0 (en)	2001-10-17	2001-12-05	Glaxo Group Ltd	Chemical compounds
GB0124938D0 (en)	2001-10-17	2001-12-05	Glaxo Group Ltd	Chemical compounds
US6921762B2 (en) *	2001-11-16	2005-07-26	Amgen Inc.	Substituted indolizine-like compounds and methods of use
WO2003051886A1 (en)	2001-12-17	2003-06-26	Smithkline Beecham Corporation	Pyrazolopyridazine derivatives
ATE375980T1 (de)	2002-02-12	2007-11-15	Smithkline Beecham Corp	Nicotinamide und deren verwendung als p38 inhibitoren
US7388009B2 (en)	2002-04-23	2008-06-17	Bristol-Myers Squibb Company	Heteroaryl-substituted pyrrolo-triazine compounds useful as kinase inhibitors
TW200306841A (en)	2002-04-23	2003-12-01	Bristol Myers Squibb Co	Aryl ketone pyrrolo-triazine compounds useful as kinase inhibitors
PT1497019E (pt)	2002-04-23	2015-09-10	Bristol Myers Squibb Co	Compostos de pirrolotriazina anilina úteis como inibidores de quinase
TW200400034A (en)	2002-05-20	2004-01-01	Bristol Myers Squibb Co	Pyrazolo-pyrimidine aniline compounds useful as kinase inhibitors
ES2278170T3 (es)	2002-07-09	2007-08-01	BOEHRINGER INGELHEIM PHARMA GMBH & CO.KG	Composiciones farmaceuticas de anticolinergicos e inhibidores de la quinasa p38 en el tratamiento de enfermedades respiratorias.
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US7652044B2 (en)	2003-06-03	2010-01-26	Novartis A.G.	P-38 inhibitors
PL2298743T3 (pl)	2003-06-26	2013-02-28	Novartis Ag	Inhibitory kinaz P38 na bazie 5-członowych heterocykli
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GB0318814D0 (en)	2003-08-11	2003-09-10	Smithkline Beecham Corp	Novel compounds
US7419978B2 (en)	2003-10-22	2008-09-02	Bristol-Myers Squibb Company	Phenyl-aniline substituted bicyclic compounds useful as kinase inhibitors
CN100584844C (zh) *	2004-01-31	2010-01-27	艾克提麦斯医药品有限公司	咪唑[1,2-c]嘧啶基乙酸衍生物
AU2005260031B2 (en) *	2004-06-25	2008-10-09	Amgen Inc.	Condensed triazoles and indazoles useful in treating citokines mediated diseases and other diseases
US7504521B2 (en)	2004-08-05	2009-03-17	Bristol-Myers Squibb Co.	Methods for the preparation of pyrrolotriazine compounds
US20060035893A1 (en)	2004-08-07	2006-02-16	Boehringer Ingelheim International Gmbh	Pharmaceutical compositions for treatment of respiratory and gastrointestinal disorders
TW200618803A (en)	2004-08-12	2006-06-16	Bristol Myers Squibb Co	Process for preparing pyrrolotriazine aniline compounds useful as kinase inhibitors
AU2005278292B2 (en)	2004-08-31	2011-09-08	Msd K.K.	Novel substituted imidazole derivatives
PE20060777A1 (es)	2004-12-24	2006-10-06	Boehringer Ingelheim Int	Derivados de indolinona para el tratamiento o la prevencion de enfermedades fibroticas
WO2006070943A1 (ja) *	2004-12-28	2006-07-06	Takeda Pharmaceutical Company Limited	縮合イミダゾール化合物およびその用途
US20060178388A1 (en)	2005-02-04	2006-08-10	Wrobleski Stephen T	Phenyl-substituted pyrimidine compounds useful as kinase inhibitors
US7473784B2 (en)	2005-08-01	2009-01-06	Bristol-Myers Squibb Company	Benzothiazole and azabenzothiazole compounds useful as kinase inhibitors
JP2009507032A (ja)	2005-09-02	2009-02-19	アボット・ラボラトリーズ	新規なイミダゾ系複素環
KR20080107408A (ko)	2006-03-07	2008-12-10	브리스톨-마이어스 스큅 컴퍼니	키나제 억제제로서 유용한 피롤로트리아진 아닐린 전구약물화합물
EP2057164A1 (en)	2006-08-07	2009-05-13	Incyte Corporation	Triazolotriazines as kinase inhibitors
EP2083816A2 (en)	2006-10-27	2009-08-05	Brystol-Myers Squibb Company	Heterocyclic amide compounds useful as kinase inhibitors
RS54510B1 (sr)	2006-11-22	2016-06-30	Incyte Holdings Corporation	Imidazotriazini i imidazopirimidini kao inhibitori kinaze
US7943617B2 (en)	2006-11-27	2011-05-17	Bristol-Myers Squibb Company	Heterobicyclic compounds useful as kinase inhibitors
US7977336B2 (en) *	2006-12-28	2011-07-12	Banyu Pharmaceutical Co. Ltd	Aminopyrimidine derivatives as PLK1 inhibitors
WO2008133192A1 (ja) *	2007-04-19	2008-11-06	Takeda Pharmaceutical Company Limited	縮合イミダゾール化合物およびその用途
EP1992344A1 (en)	2007-05-18	2008-11-19	Institut Curie	P38 alpha as a therapeutic target in pathologies linked to FGFR3 mutation
KR101002490B1 (ko) *	2007-06-09	2010-12-17	동아제약주식회사	유데나필을 유효성분으로 함유하는 만성 심부전증 치료용약학적 조성물
TWI472529B (zh)	2008-05-21	2015-02-11	Incyte Corp	２－氟－Ｎ－甲基－４－〔７－（喹啉－６－基－甲基）－咪唑并〔１，２－ｂ〕〔１，２，４〕三－２－基〕苯甲醯胺之鹽類及其相關製備方法
CN102131805A (zh)	2008-06-20	2011-07-20	百时美施贵宝公司	用作激酶抑制剂的咪唑并吡啶和咪唑并吡嗪化合物
WO2009155389A1 (en)	2008-06-20	2009-12-23	Bristol-Myers Squibb Company	Triazolopyridine compounds useful as kinase inhibitors
PE20121438A1 (es) *	2009-09-24	2012-10-26	Hoffmann La Roche	Derivados de imidazopiridina o imidazopirimidina como inhibidores de fosfodiesterasa 10a
MX2012008898A (es)	2010-02-03	2012-11-06	Incyte Corp	Imidazo - [1, 2 - b] [1, 2, 4] triazinas como inhibidores de c - met.
US8410117B2 (en) *	2010-03-26	2013-04-02	Hoffmann-La Roche Inc.	Imidazopyrimidine derivatives
WO2012031057A1 (en)	2010-09-01	2012-03-08	Bristol-Myers Squibb Company	Bms- 582949 for the treatment of resistant rheumatic disease
CN105229009B (zh) *	2013-05-23	2017-09-29	豪夫迈·罗氏有限公司	作为成像剂的2‑苯基咪唑并[1,2‑a]嘧啶
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EP3221318B1 (en) *	2014-11-21	2021-08-25	Rigel Pharmaceuticals, Inc.	Fused imidazole derivatives as tgf-beta inhibitors
US20190060286A1 (en)	2016-02-29	2019-02-28	University Of Florida Research Foundation, Incorpo	Chemotherapeutic Methods
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2000
- 2000-10-27 ES ES00976710T patent/ES2237470T3/es not_active Expired - Lifetime
- 2000-10-27 HK HK02105224.5A patent/HK1043591B/zh not_active IP Right Cessation
- 2000-10-27 NZ NZ512957A patent/NZ512957A/en unknown
- 2000-10-27 CZ CZ20012494A patent/CZ20012494A3/cs unknown
- 2000-10-27 PL PL00348924A patent/PL348924A1/xx not_active IP Right Cessation
- 2000-10-27 JP JP2001536552A patent/JP2003513977A/ja active Pending
- 2000-10-27 KR KR1020017008715A patent/KR20010089805A/ko not_active Ceased
- 2000-10-27 AT AT00976710T patent/ATE288915T1/de not_active IP Right Cessation
- 2000-10-27 WO PCT/US2000/029875 patent/WO2001034605A1/en not_active Ceased
- 2000-10-27 SK SK989-2001A patent/SK9892001A3/sk unknown
- 2000-10-27 US US09/698,448 patent/US6610697B1/en not_active Expired - Lifetime
- 2000-10-27 AU AU14445/01A patent/AU784484B2/en not_active Ceased
- 2000-10-27 ID IDW00200101720A patent/ID29514A/id unknown
- 2000-10-27 EP EP00976710A patent/EP1140939B1/en not_active Expired - Lifetime
- 2000-10-27 MX MXPA01007019A patent/MXPA01007019A/es active IP Right Grant
- 2000-10-27 UA UA2001075135A patent/UA70350C2/uk unknown
- 2000-10-27 RU RU2001122339/04A patent/RU2264403C2/ru not_active IP Right Cessation
- 2000-10-27 PT PT00976710T patent/PT1140939E/pt unknown
- 2000-10-27 DE DE60018037T patent/DE60018037T2/de not_active Expired - Fee Related
- 2000-10-27 CN CNB008045682A patent/CN1255406C/zh not_active Expired - Fee Related
- 2000-10-27 BR BR0007447-0A patent/BR0007447A/pt not_active IP Right Cessation
- 2000-10-27 CA CA002361139A patent/CA2361139A1/en not_active Abandoned
- 2000-10-27 HU HU0200207A patent/HUP0200207A3/hu unknown
- 2000-11-09 AR ARP000105910A patent/AR026410A1/es not_active Application Discontinuation
2001
- 2001-07-10 NO NO20013419A patent/NO320422B1/no not_active Application Discontinuation
- 2001-07-10 IL IL144238A patent/IL144238A/en not_active IP Right Cessation
- 2001-07-17 BG BG105712A patent/BG65106B1/bg unknown

Also Published As

Publication number	Publication date
AU1444501A (en)	2001-06-06
CN1342162A (zh)	2002-03-27
IL144238A (en)	2007-03-08
SK9892001A3 (en)	2002-04-04
RU2264403C2 (ru)	2005-11-20
BG105712A (en)	2002-06-28
HUP0200207A2 (hu)	2002-05-29
CN1255406C (zh)	2006-05-10
BR0007447A (pt)	2002-04-09
US6610697B1 (en)	2003-08-26
NO20013419D0 (no)	2001-07-10
ES2237470T3 (es)	2005-08-01
AU784484B2 (en)	2006-04-13
KR20010089805A (ko)	2001-10-08
ATE288915T1 (de)	2005-02-15
UA70350C2 (en)	2004-10-15
EP1140939A1 (en)	2001-10-10
CA2361139A1 (en)	2001-05-17
DE60018037D1 (de)	2005-03-17
DE60018037T2 (de)	2006-01-12
JP2003513977A (ja)	2003-04-15
NO20013419L (no)	2001-08-27
MXPA01007019A (es)	2002-09-18
HUP0200207A3 (en)	2004-07-28
NO320422B1 (no)	2005-12-05
AR026410A1 (es)	2003-02-12
CZ20012494A3 (cs)	2001-10-17
PL348924A1 (en)	2002-06-17
BG65106B1 (bg)	2007-02-28
HK1043591B (zh)	2006-12-29
NZ512957A (en)	2005-01-28
EP1140939B1 (en)	2005-02-09
PT1140939E (pt)	2005-05-31
HK1043591A1 (en)	2002-09-20
WO2001034605A1 (en)	2001-05-17

Publication	Publication Date	Title
ID29514A (id)	2001-09-06	2-ARIL-3-(HETEROARIL)-IMIDAZO [1,2-a]PIRIMIDIN TERSUBSTITUSI, DAN METODE-METODE DAN KOMPOSISI-KOMPOSISI FARMASI YANG TERKAIT
IL191960A (en)	2015-11-30	History of imidazo [5,1– a] pyridine and pharmaceutical preparations containing them
DK1214318T3 (da)	2004-02-09	Imidazo [1,2-a] pyridin- og pyrazolo [2,3-a] pyridin-derivater
NO20021694D0 (no)	2002-04-10	Pyrazolo[4,3-d]pyrimidinderivater
HUP0303350A3 (en)	2006-02-28	Use of substituted imidazo[1,2-a]pyridine-, imidazo[1,2-a]pyrimidine and imidazo[1,2-a]pyrazine-3-yl-amine derivatives for producing nos-inhibiting pharmaceutical compositions
HUP0400692A3 (en)	2007-09-28	Substituted 7h-pyrrolo[2,3-d]pyrimidine derivatives, their use and pharmaceutical compositions containing them
HUP0402018A3 (en)	2008-06-30	5-amino-7h-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidine derivatives, their use and pharmaceutical compositions containing them
HUP0203503A3 (en)	2004-12-28	Pyrrolo[2,3-d]pirimidine compounds, pharmaceutical compositions containing them and their use
HUP0301114A3 (en)	2004-11-29	Pyrrolo[2,3-d]pyrimidine compounds as immunosuppressive agents and pharmaceutical compositions containing them
IL128869A (en)	2003-09-17	ARYSULFONYL-SUBSTITUTED-PYRAZOLO [1,5-a]-PYRIMIDINE AND PYRAZOLO [1,5-a] [1, 3, 5]-TRIAZINE DERIVATIVES, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
HUP0401047A3 (en)	2007-12-28	Triazolo[4,5-d]pyrimidine derivatives, their use as purinergic receptor antagonist and pharmaceutical compositions containing same
ID24506A (id)	2000-07-20	Turunan-turunan 1,2,4-triazolo [4,3-b] pirido [3,2-d]-piridazina dan komposisi-komposisi farmasi yang mengandung senyawa tersebut
DE69804273D1 (de)	2002-04-25	5h-Thiazolo[3,2-a]pyrimidinderivate
HUP0500332A3 (en)	2009-12-28	Substituted 2-pyrimidinyl-6,7,8,9-tetrahydropyrimido[1,2-a]pyrimidin-4-one and 7-pyrimidinyl-2,3-dihydroimidazo[1,2-a]pyrimidin-5(1h)-one derivatives, their use and pharmaceutical compositions containing them
HUP0500328A3 (en)	2009-12-28	Substituted 2-pyridinyl-6,7,8,9-tetrahydropyrimido[1,2-a]pyrimidin-4-one and 7-pyridinyl-2,3-dihydroimidazo[1,2-a]pyrimidin-5(1h)-one derivatives, their use and pharmaceutical compositions containing them
IL156536A0 (en)	2004-01-04	Pyrazolo [3,4-d] pyrimidin-4-one derivatives and pharmaceutical compositions containing the same
DE60103909D1 (de)	2004-07-22	2-pyridinyl-6,7,8,9-tetrahydropyrimido[1,2-a]pyrimidin-4-on- und 7-pyridinyl-2,3-dihydroimidazo[1,2-a]pyrimidin-5 1honderivate
DE50001191D1 (de)	2003-03-06	Pyrazolo[4, 3-d]pyrimidine
EE200100377A (et)	2002-10-15	Imidaso[1,5-a]-pürido[3,2-e]-pürasinoonide kasutamine arstimitena
NO20000605D0 (no)	2000-02-07	3-Substituerte 3,4,5,7-tetrahydro-pyrrolo[3',4':4,5]tieno[2,3- D]pyrimidinderivater, deres fremstilling og anvendelse som 5HT- antagonister
PT1326866E (pt)	2005-08-31	3,4-di-hidropirido[1,2-a]pirimidinas substituidas
PT1325010E (pt)	2005-08-31	3, 4-di-hidropirimido [1,2-a] pirimidinas e 3, 4-di-hidropirazino [1,2-a] pirimidinas substituidas
HUP0400443A3 (en)	2005-09-28	Pyrazolo[1,2-a][1,2,4]triazole compounds useful as anti-inflammatory agents and pharmaceutical compositions containing them
IL144238A0 (en)	2002-05-23	SUBSTITUTED 2-ARYL-3-(HETEROARYL) - IMIDAZO [1,2α] PYRIMIDINES, AND RELATED PHARMACEUTICAL COMPOSITIONS AND METHODS
AU1309301A (en)	2001-06-12	Pyrazolopyrazines and their use as adenosine antagonists