IE33174L - Antibiotic 66-40 - Google Patents

Antibiotic 66-40

Info

Publication number
IE33174L
IE33174L IE690865A IE86569A IE33174L IE 33174 L IE33174 L IE 33174L IE 690865 A IE690865 A IE 690865A IE 86569 A IE86569 A IE 86569A IE 33174 L IE33174 L IE 33174L
Authority
IE
Ireland
Prior art keywords
antibiotic
mull
condensation products
aldehydes
ketones
Prior art date
Application number
IE690865A
Other versions
IE33174B1 (en
Original Assignee
Scherico Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Scherico Ltd filed Critical Scherico Ltd
Publication of IE33174L publication Critical patent/IE33174L/en
Publication of IE33174B1 publication Critical patent/IE33174B1/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20Carbocyclic rings
    • C07H15/22Cyclohexane rings, substituted by nitrogen atoms
    • C07H15/222Cyclohexane rings substituted by at least two nitrogen atoms
    • C07H15/226Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings
    • C07H15/234Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings attached to non-adjacent ring carbon atoms of the cyclohexane rings, e.g. kanamycins, tobramycin, nebramycin, gentamicin A2
    • C07H15/236Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings attached to non-adjacent ring carbon atoms of the cyclohexane rings, e.g. kanamycins, tobramycin, nebramycin, gentamicin A2 a saccharide radical being substituted by an alkylamino radical in position 3 and by two substituents different from hydrogen in position 4, e.g. gentamicin complex, sisomicin, verdamycin

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Micro-Organisms Or Cultivation Processes Thereof (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Saccharide Compounds (AREA)

Abstract

1,274,518. Antibiotic 66-40. SCHERICO Ltd. 24 June, 1969 [27 June, 1968; 16 Dec., 1968], No. 31887/69. Heading C2A. Novel Antibiotic 66-40 having the formula and characterized as being a basic pseudooligosaccharide having the following properties: elemental analysis, C = 49À80, H = 8À20, N = 14À95 and 0=27À05; molecular weight 447À26; empirical formula C 19 H 37 N 5 O 7 .H 2 O; melting point 185-190‹ C.; equivalent weight 92; pKa 8À0; [α]<SP>26‹</SP> D + 188À9‹ (C = 0À3% in H 2 O); U.V. absorption: transparent between 220 and 440 mÁ; I.R. absorption peaks at 2À98, 3À05, 3À16, 3À35- 3À50 (mull), 5À93, 6À25, 6À82 (mull), 7À25 (mull), 8À77, 9À00, 9À47, 9À72-10À07, 10À46, 11À97, 12À75 and 13À45-13À90 Á; and forming hydrates and other solvates, condensation products with aldehydes and ketones and salts with acids, is prepared by aerobically cultivating Micromonospora inyoensis (NRRL 3292). The condensation products, which are probably Schiff bases, are formed by reacting 66-40 with aldehydes and/or ketones such as acetaldehyde, acetone, methyl - ethyl - ketone, crotonaldehyde, furfural, cyclopentylacetaldehyde, vanillin, veratraldehyde, benzophenone, benzaldehyde, acetophenone, salicylaldehyde and pyridoxal. Antibiotic 66-40 has bacteriostatic activity on Gram-positive and Gram-negative bacteria and Rickettsia. Pharmaceutical compositions comprise the antibiotic 66-40 or its acid addition salts or aldehyde or ketone condensation products together with a pharmaceutically acceptable carrier or diluent, and may be in forms for topical, oral or parenteral administration. [GB1274518A]
IE865/69A 1968-06-27 1969-06-24 Antibiotic 66-40 and methods for its production IE33174B1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US74074268A 1968-06-27 1968-06-27
US79730468A 1968-12-16 1968-12-16

Publications (2)

Publication Number Publication Date
IE33174L true IE33174L (en) 1969-12-27
IE33174B1 IE33174B1 (en) 1974-04-03

Family

ID=27113740

Family Applications (1)

Application Number Title Priority Date Filing Date
IE865/69A IE33174B1 (en) 1968-06-27 1969-06-24 Antibiotic 66-40 and methods for its production

Country Status (26)

Country Link
AT (2) AT299448B (en)
BE (1) BE735145A (en)
BG (1) BG15881A3 (en)
BR (1) BR6910078D0 (en)
CA (1) CA931515A (en)
CH (2) CH529833A (en)
CS (1) CS149666B2 (en)
CY (1) CY817A (en)
DE (1) DE1932309C3 (en)
DK (1) DK126510B (en)
ES (1) ES368762A1 (en)
FI (1) FI46177C (en)
FR (1) FR2011732B1 (en)
GB (1) GB1274518A (en)
IE (1) IE33174B1 (en)
IL (1) IL32476A (en)
IT (1) IT1033250B (en)
KE (1) KE2540A (en)
LU (1) LU58942A1 (en)
MY (1) MY7500184A (en)
NL (1) NL155886B (en)
NO (1) NO129960B (en)
OA (1) OA04043A (en)
RO (1) RO57462A (en)
SE (2) SE366560B (en)
YU (1) YU34906B (en)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4297486A (en) * 1979-04-04 1981-10-27 Toyo Jozo Kabushiki Kaisha Aminoglycoside antibiotic G-367-1 and method for the production thereof
JPS5629598A (en) * 1979-08-18 1981-03-24 Toyo Jozo Co Ltd Novel amino sugar antibiotic g-367-2 and its preparation

Also Published As

Publication number Publication date
AT299448B (en) 1972-06-26
ES368762A1 (en) 1971-04-01
NL6909642A (en) 1969-12-30
CH529743A (en) 1972-10-31
OA04043A (en) 1979-10-15
BE735145A (en) 1969-12-29
KE2540A (en) 1975-07-18
NL155886B (en) 1978-02-15
SE366560B (en) 1974-04-29
AT297929B (en) 1972-04-10
CA931515A (en) 1973-08-07
RO57462A (en) 1974-12-15
CH529833A (en) 1972-10-31
FR2011732B1 (en) 1973-01-12
GB1274518A (en) 1972-05-17
IT1033250B (en) 1979-07-10
CY817A (en) 1976-12-01
MY7500184A (en) 1975-12-31
BG15881A3 (en) 1972-04-12
NO129960B (en) 1974-06-17
DE1932309B2 (en) 1974-06-20
IL32476A (en) 1972-09-28
FI46177C (en) 1973-01-10
IE33174B1 (en) 1974-04-03
YU161669A (en) 1979-10-31
DK126510B (en) 1973-07-23
IL32476A0 (en) 1969-08-27
DE1932309A1 (en) 1970-01-29
YU34906B (en) 1980-04-30
FR2011732A1 (en) 1970-03-06
CS149666B2 (en) 1973-07-25
DE1932309C3 (en) 1975-02-20
BR6910078D0 (en) 1973-02-08
SE376425B (en) 1975-05-26
FI46177B (en) 1972-10-02
LU58942A1 (en) 1969-11-11

Similar Documents

Publication Publication Date Title
RU93050124A (en) NEW DERIVATIVES OF ERYTHROMYCIN, THE METHOD OF THEIR PRODUCTION AND PHARMACEUTICAL COMPOSITION ON THEIR BASIS
IE832652L (en) Derivatives of epimeric azahomoerythromycin.
RU93050129A (en) NEW ERYTHROMYCIN DERIVATIVES, THE METHOD FOR THEIR PRODUCTION AND THE PHARMACEUTICAL COMPOSITION ON THE BASIS AND INTERMEDIATE SYNTHESIS COMPOUNDS
IE38012B1 (en) Benzothiadiazoles
GB1393521A (en) Berberine derivatives and their use in pharmaceutical compositions
GB1360420A (en) Substituted aminomethyl-dihalophenols
EP0136830A3 (en) Azahomoerythromycin d derivative and intermediates therefor
IE36607L (en) 2 - amino -2&#39;, 6&#39; - propionoxylidide
IE33174L (en) Antibiotic 66-40
JPS5270083A (en) Manufacture of an antibiotics, trans-pseudomonic acid
Gomez-Lus et al. AAC(3) and AAC(6') Enzymes Produced by R Plasmids Isolated in General Hospital.
CA938619A (en) Procede de preparation de phenols par oxydation d&#39;aldehydes aromatiques
IE36781B1 (en) Antibiotic a477 and process for preparation thereof
IE37892L (en) Antibiotic a.2315.
CA2027650A1 (en) Hair treatment composition
IE42285L (en) Butirosin-a derivatives
IE40748L (en) Antibiotic 20,798 r.p.
IE43106L (en) Mocimycin derivatives
IE38819B1 (en) Crystalline pivaloyloxymethyl d(-)- a - aminobenzylpenicillinate
ES8300773A1 (en) 7- alpha -methoxycephalosporin derivatives, and antibacterial drugs onctaining the same
JPS55151597A (en) New material 2-hydroxysagamicin and its preparation
IE38063L (en) Antibiotic g-52
JPS5629598A (en) Novel amino sugar antibiotic g-367-2 and its preparation
JPS54117478A (en) New antibiotics fortimicin kg1, kg2, and kg3, and their preparation
Joly et al. In vitro activity of co-trimazole(SMZ-TMP) on bacteria involved in upper respiratory tract infections, comparison with other antibiotics.