IE43917L - 4-(9, 10-DIHYDRO-4H-BENZO [4,5] CYCLOHEPTA [1,2-b]¹THIOPHEN-4-YLIDENE) PIPERIDINES - Google Patents
4-(9, 10-DIHYDRO-4H-BENZO [4,5] CYCLOHEPTA [1,2-b]¹THIOPHEN-4-YLIDENE) PIPERIDINESInfo
- Publication number
- IE43917L IE43917L IE761353A IE135376A IE43917L IE 43917 L IE43917 L IE 43917L IE 761353 A IE761353 A IE 761353A IE 135376 A IE135376 A IE 135376A IE 43917 L IE43917 L IE 43917L
- Authority
- IE
- Ireland
- Prior art keywords
- ylidene
- dihydro
- benzo
- 1thiophen
- cyclohepta
- Prior art date
Links
- 150000003053 piperidines Chemical class 0.000 title abstract 3
- 125000000217 alkyl group Chemical group 0.000 abstract 4
- 229940035676 analgesics Drugs 0.000 abstract 2
- 239000000730 antalgic agent Substances 0.000 abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 2
- 229910052739 hydrogen Inorganic materials 0.000 abstract 2
- 239000001257 hydrogen Substances 0.000 abstract 2
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 2
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
- C07D333/24—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pain & Pain Management (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
Case 100-4362 n4-(9,10-Dihydro-4H-Benzo4,5!Cyclcohepta1,2-b!Thiophen- 4-Ylidene)Piperidine Compounds This invention provides new compounds of formula I, (I) wherein R1 is hydrogen or alkyl, and R2 is alkyl, useful as analgesics.
Case 100-4362 n4-(9,10-Dihydro-4H-Benzo¢4,5!Cyclcohepta¢1,2-b!Thiophen- 4-Ylidene)Piperidine Compounds This invention provides new compounds of formula I, (I) wherein R1 is hydrogen or alkyl, and R2 is alkyl, useful as analgesics.
[CA1085403A]
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CH817375A CH615927A5 (en) | 1975-06-24 | 1975-06-24 | Process for the preparation of novel benzocycloheptathiophene derivatives |
| CH817475A CH613204A5 (en) | 1975-06-24 | 1975-06-24 | Process for the preparation of novel benzocycloheptathiophene derivatives |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| IE43917L true IE43917L (en) | 1976-12-24 |
| IE43917B1 IE43917B1 (en) | 1981-07-01 |
Family
ID=25702907
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IE1353/76A IE43917B1 (en) | 1975-06-24 | 1976-06-22 | 4-(9,10-dihydro-4h-benzo/4,5/cyclohepta/1,2-b/thiophen-4-ylidine piperidines |
Country Status (17)
| Country | Link |
|---|---|
| JP (1) | JPS523075A (en) |
| AU (1) | AU508585B2 (en) |
| CA (1) | CA1085403A (en) |
| DE (1) | DE2626583A1 (en) |
| DK (1) | DK267976A (en) |
| ES (1) | ES449099A1 (en) |
| FI (1) | FI761721A7 (en) |
| FR (1) | FR2316949A1 (en) |
| GB (1) | GB1554427A (en) |
| IE (1) | IE43917B1 (en) |
| IL (1) | IL49862A (en) |
| NL (1) | NL7606700A (en) |
| NO (1) | NO762085L (en) |
| NZ (1) | NZ181236A (en) |
| PH (1) | PH14805A (en) |
| PT (1) | PT65264B (en) |
| SE (1) | SE7606877L (en) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS597963B2 (en) * | 1977-06-28 | 1984-02-22 | 沖電気工業株式会社 | Circular interpolation circuit in numerical control |
| DE3170504D1 (en) * | 1980-09-02 | 1985-06-20 | Sandoz Ag | Piperidylidene derivatives, their production and pharmaceutical compositions containing them |
| JPS63205706A (en) * | 1987-02-23 | 1988-08-25 | Yaskawa Electric Mfg Co Ltd | Arc machining control method |
| ID24487A (en) * | 1997-04-03 | 2000-07-20 | Bridge Pharma Inc | COMPOUND, BENZOSIKLOHEPTATIOFEN COMPOUNDS |
| CN101932575B (en) | 2008-01-30 | 2013-06-12 | 日本脏器制药株式会社 | Piperidine derivative |
| JP5083989B2 (en) * | 2008-11-20 | 2012-11-28 | 日本臓器製薬株式会社 | Medicaments containing piperidine derivatives |
| CN113227037A (en) * | 2018-09-30 | 2021-08-06 | 北京生命科学研究所 | Monohalogen or methyl substituted 5-HT2B antagonists with increased activity |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR1437412A (en) * | 1963-12-19 | 1966-05-06 | Sandoz Sa | New benzo-cyclohepta-thiophenes and their preparation |
-
1976
- 1976-06-14 DE DE19762626583 patent/DE2626583A1/en not_active Withdrawn
- 1976-06-15 FI FI761721A patent/FI761721A7/fi not_active Application Discontinuation
- 1976-06-15 DK DK267976A patent/DK267976A/en not_active Application Discontinuation
- 1976-06-16 SE SE7606877A patent/SE7606877L/en unknown
- 1976-06-16 NO NO762085A patent/NO762085L/no unknown
- 1976-06-21 CA CA255,311A patent/CA1085403A/en not_active Expired
- 1976-06-21 NL NL7606700A patent/NL7606700A/en not_active Application Discontinuation
- 1976-06-22 IE IE1353/76A patent/IE43917B1/en unknown
- 1976-06-22 ES ES449099A patent/ES449099A1/en not_active Expired
- 1976-06-22 IL IL49862A patent/IL49862A/en unknown
- 1976-06-22 GB GB25887/76A patent/GB1554427A/en not_active Expired
- 1976-06-22 NZ NZ181236A patent/NZ181236A/en unknown
- 1976-06-23 PH PH18600A patent/PH14805A/en unknown
- 1976-06-23 FR FR7619092A patent/FR2316949A1/en active Granted
- 1976-06-23 PT PT65264A patent/PT65264B/en unknown
- 1976-06-23 JP JP51073391A patent/JPS523075A/en active Pending
- 1976-06-23 AU AU15203/76A patent/AU508585B2/en not_active Expired
Also Published As
| Publication number | Publication date |
|---|---|
| JPS523075A (en) | 1977-01-11 |
| NZ181236A (en) | 1978-06-20 |
| IL49862A (en) | 1980-11-30 |
| PH14805A (en) | 1981-12-14 |
| AU1520376A (en) | 1978-01-05 |
| DE2626583A1 (en) | 1977-01-13 |
| SE7606877L (en) | 1976-12-25 |
| DK267976A (en) | 1976-12-25 |
| IL49862A0 (en) | 1976-08-31 |
| FR2316949A1 (en) | 1977-02-04 |
| FR2316949B1 (en) | 1979-10-12 |
| AU508585B2 (en) | 1980-03-27 |
| NO762085L (en) | 1976-12-28 |
| NL7606700A (en) | 1976-12-28 |
| PT65264A (en) | 1976-07-01 |
| ES449099A1 (en) | 1978-03-01 |
| GB1554427A (en) | 1979-10-24 |
| IE43917B1 (en) | 1981-07-01 |
| CA1085403A (en) | 1980-09-09 |
| FI761721A7 (en) | 1976-12-25 |
| PT65264B (en) | 1978-03-24 |
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