IL103151A0 - Beta-carboline derivatives,processes for the preparation thereof and pharmaceutical compositions containing the same - Google Patents
Beta-carboline derivatives,processes for the preparation thereof and pharmaceutical compositions containing the sameInfo
- Publication number
- IL103151A0 IL103151A0 IL103151A IL10315192A IL103151A0 IL 103151 A0 IL103151 A0 IL 103151A0 IL 103151 A IL103151 A IL 103151A IL 10315192 A IL10315192 A IL 10315192A IL 103151 A0 IL103151 A0 IL 103151A0
- Authority
- IL
- Israel
- Prior art keywords
- beta
- processes
- preparation
- same
- pharmaceutical compositions
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Psychiatry (AREA)
- Hospice & Palliative Care (AREA)
- Pain & Pain Management (AREA)
- Anesthesiology (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE4130933A DE4130933A1 (de) | 1991-09-13 | 1991-09-13 | Neue (beta)-carbolinderivate, deren herstellung und verwendung in arzneimitteln |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| IL103151A0 true IL103151A0 (en) | 1993-02-21 |
Family
ID=6440817
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL103151A IL103151A0 (en) | 1991-09-13 | 1992-09-13 | Beta-carboline derivatives,processes for the preparation thereof and pharmaceutical compositions containing the same |
Country Status (17)
| Country | Link |
|---|---|
| US (1) | US5506234A (fr) |
| EP (1) | EP0557497A1 (fr) |
| JP (1) | JPH06502871A (fr) |
| KR (1) | KR930703313A (fr) |
| CN (1) | CN1033391C (fr) |
| AU (1) | AU655503B2 (fr) |
| CA (1) | CA2096138A1 (fr) |
| CZ (1) | CZ72593A3 (fr) |
| DE (1) | DE4130933A1 (fr) |
| FI (1) | FI932145A0 (fr) |
| HU (1) | HUT64343A (fr) |
| IL (1) | IL103151A0 (fr) |
| MX (1) | MX9205164A (fr) |
| NZ (1) | NZ244328A (fr) |
| PT (1) | PT100860A (fr) |
| WO (1) | WO1993006100A1 (fr) |
| ZA (1) | ZA926969B (fr) |
Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE4330175A1 (de) * | 1993-08-31 | 1995-03-02 | Schering Ag | Alkoxy-substituierte beta-Carboline |
| DE19502753A1 (de) * | 1995-01-23 | 1996-07-25 | Schering Ag | Neue 9H-Pyrido[3,4-b]indol-Derivate |
| DE19514524A1 (de) * | 1995-04-12 | 1996-10-17 | Schering Ag | Anellierte beta-Carboline |
| PL220850B1 (pl) * | 2002-05-03 | 2016-01-29 | Janssen Pharmaceutica Nv | Kopolimer dwublokowy, kompozycja zawierająca składnik aktywny i jej zastosowanie oraz sposób jej wytwarzania |
| US7504401B2 (en) | 2003-08-29 | 2009-03-17 | Locus Pharmaceuticals, Inc. | Anti-cancer agents and uses thereof |
| BRPI0907122B8 (pt) | 2008-01-11 | 2021-05-25 | Albany Molecular Res Inc | compostos de piridoindóis (1-azinona) substituídos, composição farmacêutica compreendendo os referidos compostos, e usos dos mesmos |
| WO2011003012A1 (fr) * | 2009-07-01 | 2011-01-06 | Albany Molecular Research, Inc. | Antagonistes de mch-1 azapolycycles substitués par azinone, leurs procédés de fabrication et leur utilisation |
| US8637501B2 (en) * | 2009-07-01 | 2014-01-28 | Albany Molecular Research, Inc. | Azinone-substituted azepino[b]indole and pyrido-pyrrolo-azepine MCH-1 antagonists, methods of making, and use thereof |
| US9073925B2 (en) * | 2009-07-01 | 2015-07-07 | Albany Molecular Research, Inc. | Azinone-substituted azabicycloalkane-indole and azabicycloalkane-pyrrolo-pyridine MCH-1 antagonists, methods of making, and use thereof |
| WO2011003007A1 (fr) * | 2009-07-01 | 2011-01-06 | Albany Molecular Research, Inc. | Antagonistes de mch-1 dazabicycloalcane-indole et dazabicycloalcane-pyrrolo-pyridine, procédés de préparation, et utilisation de ceux-ci |
| EP2582666B1 (fr) | 2010-06-16 | 2014-08-13 | Purdue Pharma L.P. | Indoles à substitution aryle et leur utilisation en tant que bloqueur des canaux sodium |
| EP2455378A1 (fr) | 2010-11-03 | 2012-05-23 | Philip Morris Products S.A. | Dérivés de carbazole et de carboline, et préparation et applications thérapeutiques associées |
| WO2012088038A2 (fr) | 2010-12-21 | 2012-06-28 | Albany Molecular Research, Inc. | Antagonistes de mch-1 consistant en tétrahydro-carbolines substituées par pipérazinone, leurs procédés de fabrication et utilisations |
| WO2012088124A2 (fr) | 2010-12-21 | 2012-06-28 | Albany Molecular Research, Inc. | Antagonistes de la mch-1 à base de tétrahydro-azacarboline, leurs procédés de fabrication et leurs utilisations |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS57123180A (en) * | 1980-12-17 | 1982-07-31 | Schering Ag | 3-substituted beta-carboline, manufacture and psychotropic drug containing same |
| DE3335323A1 (de) * | 1983-09-27 | 1985-04-04 | Schering AG, 1000 Berlin und 4709 Bergkamen | Substituierte ss-carboline, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel |
| DK240084D0 (da) * | 1984-05-15 | 1984-05-15 | Ferrosan As | New beta-carboline-3-oxadiazolyl derivatives |
| DE3504045A1 (de) * | 1985-02-04 | 1986-08-07 | Schering AG, 1000 Berlin und 4709 Bergkamen | Verfahren zur herstellung von ss-carbolinen durch dehydrierung |
| DE3545776A1 (de) * | 1985-12-20 | 1987-06-25 | Schering Ag | 5-aminoalkyl-ss-carbolinderivate, ihre herstellung und ihre verwendung als arzneimittel |
| DE3608089A1 (de) * | 1986-03-08 | 1987-09-10 | Schering Ag | Heteroaryl-oxy-ss-carbolinderivate, ihre herstellung und ihre verwendung als arzneimittel |
| IL87563A (en) * | 1987-08-28 | 1993-08-18 | Schering Ag | Isoxazole-b-carboline derivatives, processes for the preparation thereof and pharmaceutical compositions containing the same |
| DE3925507A1 (de) * | 1989-07-28 | 1991-01-31 | Schering Ag | 14,17(alpha)-etheno- und ethanoestratriene, verfahren zur herstellung dieser verbindungen, sowie ihre verwendung zur herstellung von arzneimitteln |
| DE3943225A1 (de) * | 1989-12-23 | 1991-06-27 | Schering Ag | Neue ss-carboline, verfahren zu deren herstellung und deren verwendung in arzneimitteln |
-
1991
- 1991-09-13 DE DE4130933A patent/DE4130933A1/de not_active Withdrawn
-
1992
- 1992-09-10 MX MX9205164A patent/MX9205164A/es not_active Application Discontinuation
- 1992-09-11 CA CA002096138A patent/CA2096138A1/fr not_active Abandoned
- 1992-09-11 AU AU25578/92A patent/AU655503B2/en not_active Ceased
- 1992-09-11 KR KR1019930701425A patent/KR930703313A/ko not_active Withdrawn
- 1992-09-11 FI FI932145A patent/FI932145A0/fi not_active Application Discontinuation
- 1992-09-11 EP EP92919414A patent/EP0557497A1/fr not_active Withdrawn
- 1992-09-11 CZ CS93725A patent/CZ72593A3/cs unknown
- 1992-09-11 HU HU9301379A patent/HUT64343A/hu unknown
- 1992-09-11 PT PT100860A patent/PT100860A/pt not_active Application Discontinuation
- 1992-09-11 ZA ZA926969A patent/ZA926969B/xx unknown
- 1992-09-11 JP JP5505694A patent/JPH06502871A/ja active Pending
- 1992-09-11 WO PCT/DE1992/000786 patent/WO1993006100A1/fr not_active Ceased
- 1992-09-12 CN CN92110560A patent/CN1033391C/zh not_active Expired - Fee Related
- 1992-09-13 IL IL103151A patent/IL103151A0/xx unknown
- 1992-09-14 US US07/943,177 patent/US5506234A/en not_active Expired - Fee Related
- 1992-09-14 NZ NZ244328A patent/NZ244328A/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| EP0557497A1 (fr) | 1993-09-01 |
| AU2557892A (en) | 1993-04-27 |
| HUT64343A (en) | 1993-12-28 |
| CA2096138A1 (fr) | 1993-03-14 |
| WO1993006100A1 (fr) | 1993-04-01 |
| FI932145L (fi) | 1993-05-12 |
| JPH06502871A (ja) | 1994-03-31 |
| DE4130933A1 (de) | 1993-03-18 |
| PT100860A (pt) | 1993-11-30 |
| CZ72593A3 (en) | 1994-01-19 |
| NZ244328A (en) | 1995-02-24 |
| AU655503B2 (en) | 1994-12-22 |
| ZA926969B (en) | 1993-03-17 |
| FI932145A7 (fi) | 1993-05-12 |
| MX9205164A (es) | 1993-03-01 |
| CN1033391C (zh) | 1996-11-27 |
| CN1070403A (zh) | 1993-03-31 |
| HU9301379D0 (en) | 1993-09-28 |
| FI932145A0 (fi) | 1993-05-12 |
| US5506234A (en) | 1996-04-09 |
| KR930703313A (ko) | 1993-11-29 |
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