IL117631A - Polysubstituted condensed di (and tri) cyclic heterocyclic compounds their production and pharmaceutical compositions containing them - Google Patents

Polysubstituted condensed di (and tri) cyclic heterocyclic compounds their production and pharmaceutical compositions containing them

Info

Publication number
IL117631A
IL117631A IL11763196A IL11763196A IL117631A IL 117631 A IL117631 A IL 117631A IL 11763196 A IL11763196 A IL 11763196A IL 11763196 A IL11763196 A IL 11763196A IL 117631 A IL117631 A IL 117631A
Authority
IL
Israel
Prior art keywords
tri
production
pharmaceutical compositions
compositions containing
heterocyclic compounds
Prior art date
Application number
IL11763196A
Other languages
English (en)
Other versions
IL117631A0 (en
Original Assignee
Takeda Chemical Industries Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Takeda Chemical Industries Ltd filed Critical Takeda Chemical Industries Ltd
Publication of IL117631A0 publication Critical patent/IL117631A0/xx
Publication of IL117631A publication Critical patent/IL117631A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/02Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/14Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pulmonology (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Pain & Pain Management (AREA)
  • Urology & Nephrology (AREA)
  • Immunology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
IL11763196A 1995-03-24 1996-03-24 Polysubstituted condensed di (and tri) cyclic heterocyclic compounds their production and pharmaceutical compositions containing them IL117631A (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
JP9143695 1995-03-24
JP20755395 1995-07-20
JP26472795 1995-09-18
JP3003396 1996-01-23

Publications (2)

Publication Number Publication Date
IL117631A0 IL117631A0 (en) 1996-07-23
IL117631A true IL117631A (en) 2000-11-21

Family

ID=27459171

Family Applications (1)

Application Number Title Priority Date Filing Date
IL11763196A IL117631A (en) 1995-03-24 1996-03-24 Polysubstituted condensed di (and tri) cyclic heterocyclic compounds their production and pharmaceutical compositions containing them

Country Status (17)

Country Link
US (3) US5786352A (de)
EP (1) EP0733632B1 (de)
KR (1) KR960034203A (de)
CN (1) CN1140172A (de)
AR (1) AR003937A1 (de)
AT (1) ATE242243T1 (de)
AU (1) AU699611B2 (de)
BR (1) BR9601125A (de)
CA (1) CA2172421A1 (de)
DE (1) DE69628484T2 (de)
ES (1) ES2194937T3 (de)
HU (1) HUP9600732A3 (de)
IL (1) IL117631A (de)
MX (1) MX9601072A (de)
NO (1) NO309272B1 (de)
NZ (1) NZ286256A (de)
TW (1) TW394773B (de)

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PT1035115E (pt) * 1999-02-24 2005-01-31 Hoffmann La Roche Derivados de 4-fenilpiridina e a sua utilizacao como antagonistas do receptor nk-1
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US7163949B1 (en) 1999-11-03 2007-01-16 Amr Technology, Inc. 4-phenyl substituted tetrahydroisoquinolines and use thereof
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KR100821410B1 (ko) 2000-07-11 2008-04-10 에이엠알 테크놀로지, 인크. 4-페닐 치환된 테트라하이드로이소퀴놀린 및 이의치료학적 용도
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EP3525785B1 (de) 2016-10-12 2025-08-27 Merck Sharp & Dohme LLC Kdm5-inhibitoren
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EP3706747B1 (de) 2017-11-08 2025-09-03 Merck Sharp & Dohme LLC Prmt5-inhibitoren
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DE2357253A1 (de) * 1973-11-16 1975-05-22 Thomae Gmbh Dr K Neue chinolinderivate
ES431307A1 (es) * 1973-11-16 1976-09-01 Thomae Gmbh Dr K Procedimiento para la preparacion de nuevos derivados de quinoleina.
DE2617101A1 (de) * 1976-04-17 1977-11-17 Thomae Gmbh Dr K Neue naphthyridine
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TW241258B (de) * 1992-04-15 1995-02-21 Takeda Pharm Industry Co Ltd
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TW263498B (de) * 1993-11-10 1995-11-21 Takeda Pharm Industry Co Ltd

Also Published As

Publication number Publication date
ATE242243T1 (de) 2003-06-15
US5786352A (en) 1998-07-28
CA2172421A1 (en) 1996-09-25
EP0733632B1 (de) 2003-06-04
CN1140172A (zh) 1997-01-15
MX9601072A (es) 1997-03-29
US6489315B1 (en) 2002-12-03
AU4826196A (en) 1996-10-03
NO961160D0 (no) 1996-03-21
US6147071A (en) 2000-11-14
HU9600732D0 (en) 1996-05-28
NZ286256A (en) 1999-05-28
AR003937A1 (es) 1998-09-30
NO309272B1 (no) 2001-01-08
EP0733632A1 (de) 1996-09-25
HUP9600732A2 (en) 1997-03-28
DE69628484D1 (de) 2003-07-10
BR9601125A (pt) 1998-01-06
ES2194937T3 (es) 2003-12-01
NO961160L (no) 1996-09-25
KR960034203A (ko) 1996-10-22
IL117631A0 (en) 1996-07-23
DE69628484T2 (de) 2004-05-19
TW394773B (en) 2000-06-21
AU699611B2 (en) 1998-12-10
HUP9600732A3 (en) 2000-03-28

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