IL268501B1 - Sulfoxyamine glycosidase inhibitors - Google Patents

Sulfoxyamine glycosidase inhibitors

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Publication number
IL268501B1
IL268501B1 IL268501A IL26850119A IL268501B1 IL 268501 B1 IL268501 B1 IL 268501B1 IL 268501 A IL268501 A IL 268501A IL 26850119 A IL26850119 A IL 26850119A IL 268501 B1 IL268501 B1 IL 268501B1
Authority
IL
Israel
Prior art keywords
mmol
formula
compounds
group
pct
Prior art date
Application number
IL268501A
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English (en)
Hebrew (he)
Other versions
IL268501A (en
Original Assignee
Asceneuron S A
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from PCT/EP2017/054268 external-priority patent/WO2017144633A1/en
Priority claimed from PCT/EP2017/071385 external-priority patent/WO2018153508A2/en
Application filed by Asceneuron S A filed Critical Asceneuron S A
Publication of IL268501A publication Critical patent/IL268501A/en
Publication of IL268501B1 publication Critical patent/IL268501B1/en

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    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
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