MA47574A - Inhibiteurs de la sulfoximine glycosidase - Google Patents

Inhibiteurs de la sulfoximine glycosidase

Info

Publication number
MA47574A
MA47574A MA047574A MA47574A MA47574A MA 47574 A MA47574 A MA 47574A MA 047574 A MA047574 A MA 047574A MA 47574 A MA47574 A MA 47574A MA 47574 A MA47574 A MA 47574A
Authority
MA
Morocco
Prior art keywords
sulfoximine
glycosidase inhibitors
glycosidase
inhibitors
sulfoximine glycosidase
Prior art date
Application number
MA047574A
Other languages
English (en)
Inventor
Awadut Gajendra Giri
Santosh S Kulkarni
Anna Quattropani
Original Assignee
Asceneuron Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from PCT/EP2017/054268 external-priority patent/WO2017144633A1/fr
Application filed by Asceneuron Sa filed Critical Asceneuron Sa
Publication of MA47574A publication Critical patent/MA47574A/fr

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
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    • A61K31/4965—Non-condensed pyrazines
    • A61K31/497—Non-condensed pyrazines containing further heterocyclic rings
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KR20180132626A (ko) 2018-12-12
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EP3419972A1 (fr) 2019-01-02
US10995090B2 (en) 2021-05-04
EP3419972B1 (fr) 2023-07-26
KR20230026541A (ko) 2023-02-24
US10556902B2 (en) 2020-02-11
AU2017222964B2 (en) 2020-01-02
IL268501B2 (en) 2026-05-01
US20190388415A1 (en) 2019-12-26
KR102620279B1 (ko) 2024-01-03
CN108884078A (zh) 2018-11-23
AU2017222964A1 (en) 2018-08-02
US20190055239A1 (en) 2019-02-21
MA47573A (fr) 2021-04-28
WO2017144639A1 (fr) 2017-08-31
CA3012624A1 (fr) 2017-08-31
KR20190118184A (ko) 2019-10-17
MA43680A (fr) 2018-11-28
IL268501A (en) 2019-09-26
CA3053200A1 (fr) 2018-08-30
IL268501B1 (en) 2026-01-01
BR112019017514A2 (pt) 2020-03-31
MX2018010191A (es) 2019-05-20

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