IL64502A0 - Novel benzo(b)thiophenes,benzo(b)furans,thiochromans and chromans,processes for their preparation and antimicrobial compositions containing them - Google Patents

Novel benzo(b)thiophenes,benzo(b)furans,thiochromans and chromans,processes for their preparation and antimicrobial compositions containing them

Info

Publication number
IL64502A0
IL64502A0 IL64502A IL6450281A IL64502A0 IL 64502 A0 IL64502 A0 IL 64502A0 IL 64502 A IL64502 A IL 64502A IL 6450281 A IL6450281 A IL 6450281A IL 64502 A0 IL64502 A0 IL 64502A0
Authority
IL
Israel
Prior art keywords
group
groups
lower alkyl
alkyl
aryl
Prior art date
Application number
IL64502A
Other languages
English (en)
Original Assignee
Schering Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Corp filed Critical Schering Corp
Publication of IL64502A0 publication Critical patent/IL64502A0/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
    • C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
    • C07D295/182—Radicals derived from carboxylic acids
    • C07D295/185—Radicals derived from carboxylic acids from aliphatic carboxylic acids
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/50—1,3-Diazoles; Hydrogenated 1,3-diazoles
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/64—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with three nitrogen atoms as the only ring hetero atoms
    • A01N43/647—Triazoles; Hydrogenated triazoles
    • A01N43/653—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D335/00—Heterocyclic compounds containing six-membered rings having one sulfur atom as the only ring hetero atom
    • C07D335/04—Heterocyclic compounds containing six-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D335/06—Benzothiopyrans; Hydrogenated benzothiopyrans

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Dentistry (AREA)
  • Engineering & Computer Science (AREA)
  • Plant Pathology (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cosmetics (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
IL64502A 1980-12-12 1981-12-10 Novel benzo(b)thiophenes,benzo(b)furans,thiochromans and chromans,processes for their preparation and antimicrobial compositions containing them IL64502A0 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/215,948 US4352808A (en) 1980-12-12 1980-12-12 3-Aralkyloxy-2,3-dihydro-2-(imidazolylmethyl)benzo(b)thiophenes and related derivatives, their use as antimicrobials and pharmaceutical formulations useful therefore

Publications (1)

Publication Number Publication Date
IL64502A0 true IL64502A0 (en) 1982-03-31

Family

ID=22805054

Family Applications (1)

Application Number Title Priority Date Filing Date
IL64502A IL64502A0 (en) 1980-12-12 1981-12-10 Novel benzo(b)thiophenes,benzo(b)furans,thiochromans and chromans,processes for their preparation and antimicrobial compositions containing them

Country Status (13)

Country Link
US (1) US4352808A (fr)
EP (1) EP0054233B1 (fr)
JP (1) JPS57131787A (fr)
AT (1) ATE22444T1 (fr)
AU (1) AU546360B2 (fr)
DE (1) DE3175392D1 (fr)
IE (1) IE52220B1 (fr)
IL (1) IL64502A0 (fr)
MY (1) MY8700623A (fr)
NZ (1) NZ199232A (fr)
OA (1) OA07075A (fr)
PH (1) PH18750A (fr)
ZA (1) ZA818593B (fr)

Families Citing this family (64)

* Cited by examiner, † Cited by third party
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JPS5845426B2 (ja) * 1978-09-29 1983-10-08 杏林製薬株式会社 置換キノリンカルボン酸誘導体
US4468404A (en) * 1980-12-12 1984-08-28 Schering Corporation 3-Aralkyloxy-2,3-dihydro-2-(triazolymethyl)benzo(b)thiophenes
JPS59225183A (ja) * 1983-02-01 1984-12-18 Yoshitomi Pharmaceut Ind Ltd ジヒドロベンゾフラン誘導体
IT1161927B (it) * 1983-03-31 1987-03-18 Montedison Spa Furano-derivati ad attivita' fungicida
US4659730A (en) * 1984-06-18 1987-04-21 Eli Lilly And Company Aromatase inhibiting imidazole derivatives
US4695579A (en) * 1984-12-21 1987-09-22 Schering Corporation Antifungal 2-azolylmethyl-3-difluorobenzyloxy-2,3-dihydrofluoro-benzo(B) thiophens
US4731364A (en) * 1985-08-12 1988-03-15 Schering Corporation Dihydrobenzo(B)thiophenes and pharmaceutical compositions thereof useful as antifungals
US4820724A (en) * 1986-03-31 1989-04-11 University Of Southern California Dual phase solvent carrier system
US4765978A (en) * 1986-12-16 1988-08-23 Schering Corporation Novel vaginal suppository
GB8726505D0 (en) * 1987-11-12 1987-12-16 Ici Plc Naphtho(2 1-b)furan derivatives
US4943311A (en) * 1988-05-09 1990-07-24 Uniroyal Chemical Company, Inc. Azole derivatives of spiroheterocycles
DE4010797A1 (de) * 1990-04-04 1991-10-10 Hoechst Ag Substituierte azole, verfahren zu deren herstellung, diese enthaltende mittel und deren verwendung
EP0457716A1 (fr) * 1990-04-20 1991-11-21 Ciba-Geigy Ag Dérivés de naphtaline
DE4024206A1 (de) * 1990-07-31 1992-02-06 Basf Ag 2,2'-thienyl-benzothiophene, ihre herstellung und ihre verwendung zur bekaempfung von schaedlingen
TW224461B (fr) * 1990-09-18 1994-06-01 Ciba Geigy Ag
DE4128690A1 (de) * 1991-08-29 1993-03-04 Boehringer Mannheim Gmbh Bicyclische sulfone, verfahren zu ihrer herstellung und diese enthaltende arzneimittel
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US6147077A (en) * 1999-04-29 2000-11-14 Sepracor Inc. 2R,4S-hydroxyitraconazole isomers
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US8900554B2 (en) 2002-10-25 2014-12-02 Foamix Pharmaceuticals Ltd. Foamable composition and uses thereof
US9668972B2 (en) 2002-10-25 2017-06-06 Foamix Pharmaceuticals Ltd. Nonsteroidal immunomodulating kit and composition and uses thereof
ES2532906T5 (es) 2002-10-25 2022-03-23 Foamix Pharmaceuticals Ltd Espuma cosmética y farmacéutica
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DE10328049A1 (de) * 2003-06-20 2005-01-13 Ernst-Moritz-Arndt-Universität Neue antimikrobielle Chroman-4-one
US8795693B2 (en) 2003-08-04 2014-08-05 Foamix Ltd. Compositions with modulating agents
US8486374B2 (en) 2003-08-04 2013-07-16 Foamix Ltd. Hydrophilic, non-aqueous pharmaceutical carriers and compositions and uses
US20080260655A1 (en) 2006-11-14 2008-10-23 Dov Tamarkin Substantially non-aqueous foamable petrolatum based pharmaceutical and cosmetic compositions and their uses
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US9439857B2 (en) 2007-11-30 2016-09-13 Foamix Pharmaceuticals Ltd. Foam containing benzoyl peroxide
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JP2019529670A (ja) 2016-10-04 2019-10-17 ダウ シリコーンズ コーポレーション シリコーン樹脂−直鎖状コポリマー及び関連する方法
WO2018067691A1 (fr) 2016-10-04 2018-04-12 Dow Silicones Corporation Copolymère linéaire-résine de silicone et procédés associés
WO2019232151A1 (fr) 2018-05-30 2019-12-05 Dow Silicones Corporation Émulsion et procédé pour la préparer
WO2020142282A2 (fr) 2018-12-31 2020-07-09 Dow Silicones Corporation Composition de soins personnels, procédé de préparation de la composition et procédé de traitement impliquant la composition
KR20210110338A (ko) 2018-12-31 2021-09-07 다우 실리콘즈 코포레이션 분지형 유기규소 화합물, 이의 제조 방법, 및 관련 조성물
JP7561738B2 (ja) 2018-12-31 2024-10-04 ダウ シリコーンズ コーポレーション 組成物、コポリマーの調製方法、並びにその方法及び最終用途
EP3906274A1 (fr) 2018-12-31 2021-11-10 Dow Silicones Corporation Composé d'organosilicium ramifié à fonction acrylate, son procédé de préparation et copolymère formé avec celui-ci
KR20210110843A (ko) 2018-12-31 2021-09-09 다우 실리콘즈 코포레이션 분지형 유기규소 화합물, 이의 제조 방법, 및 이로 형성된 공중합체
WO2020142444A1 (fr) 2018-12-31 2020-07-09 Dow Silicones Corporation Composé d'organosilicium ramifié, procédé de préparation dudit composé et compositions comportant ledit composé
EP3906275A1 (fr) 2018-12-31 2021-11-10 Dow Silicones Corporation Composé d'organosilicium ramifié, son procédé de préparation et compositions le comprenant
KR20210114430A (ko) 2018-12-31 2021-09-23 다우 실리콘즈 코포레이션 분지형 유기규소 화합물, 그의 제조 방법, 및 그로 형성된 공중합체
KR20240016356A (ko) 2021-06-04 2024-02-06 액세스 비지니스 그룹 인터내셔날 엘엘씨 피부 적용분야를 위한 오리스 뿌리 추출물, 조성물 및 방법

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Also Published As

Publication number Publication date
AU7845881A (en) 1982-06-17
PH18750A (en) 1985-09-19
US4352808A (en) 1982-10-05
NZ199232A (en) 1985-04-30
AU546360B2 (en) 1985-08-29
ATE22444T1 (de) 1986-10-15
DE3175392D1 (en) 1986-10-30
EP0054233B1 (fr) 1986-09-24
IE52220B1 (en) 1987-08-05
IE812910L (en) 1982-06-12
OA07075A (fr) 1984-01-31
JPS57131787A (en) 1982-08-14
EP0054233A1 (fr) 1982-06-23
ZA818593B (en) 1982-09-29
MY8700623A (en) 1987-12-31

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