IL75533A - Preparation of heteroaryloxyacetamides - Google Patents
Preparation of heteroaryloxyacetamidesInfo
- Publication number
- IL75533A IL75533A IL75533A IL7553385A IL75533A IL 75533 A IL75533 A IL 75533A IL 75533 A IL75533 A IL 75533A IL 7553385 A IL7553385 A IL 7553385A IL 75533 A IL75533 A IL 75533A
- Authority
- IL
- Israel
- Prior art keywords
- heteroaryloxyacetamides
- preparation
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/52—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings condensed with carbocyclic rings or ring systems
- C07D263/54—Benzoxazoles; Hydrogenated benzoxazoles
- C07D263/58—Benzoxazoles; Hydrogenated benzoxazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D271/00—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms
- C07D271/02—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms not condensed with other rings
- C07D271/06—1,2,4-Oxadiazoles; Hydrogenated 1,2,4-oxadiazoles
- C07D271/07—1,2,4-Oxadiazoles; Hydrogenated 1,2,4-oxadiazoles with oxygen, sulfur or nitrogen atoms, directly attached to ring carbon atoms, the nitrogen atoms not forming part of a nitro radical
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/34—Oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
- C07D277/62—Benzothiazoles
- C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
- C07D285/01—Five-membered rings
- C07D285/02—Thiadiazoles; Hydrogenated thiadiazoles
- C07D285/04—Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
- C07D285/08—1,2,4-Thiadiazoles; Hydrogenated 1,2,4-thiadiazoles
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
- C07D285/01—Five-membered rings
- C07D285/02—Thiadiazoles; Hydrogenated thiadiazoles
- C07D285/04—Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
- C07D285/12—1,3,4-Thiadiazoles; Hydrogenated 1,3,4-thiadiazoles
- C07D285/125—1,3,4-Thiadiazoles; Hydrogenated 1,3,4-thiadiazoles with oxygen, sulfur or nitrogen atoms, directly attached to ring carbon atoms, the nitrogen atoms not forming part of a nitro radical
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
- C07D285/01—Five-membered rings
- C07D285/02—Thiadiazoles; Hydrogenated thiadiazoles
- C07D285/04—Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
- C07D285/12—1,3,4-Thiadiazoles; Hydrogenated 1,3,4-thiadiazoles
- C07D285/125—1,3,4-Thiadiazoles; Hydrogenated 1,3,4-thiadiazoles with oxygen, sulfur or nitrogen atoms, directly attached to ring carbon atoms, the nitrogen atoms not forming part of a nitro radical
- C07D285/13—Oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE19843422861 DE3422861A1 (de) | 1984-06-20 | 1984-06-20 | Verfahren zur herstellung von heteroaryloxyacetamiden |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| IL75533A0 IL75533A0 (en) | 1985-10-31 |
| IL75533A true IL75533A (en) | 1990-01-18 |
Family
ID=6238800
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL75533A IL75533A (en) | 1984-06-20 | 1985-06-17 | Preparation of heteroaryloxyacetamides |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US5101034A (fr) |
| EP (1) | EP0165537B1 (fr) |
| JP (1) | JPH0714925B2 (fr) |
| KR (1) | KR920010393B1 (fr) |
| DE (2) | DE3422861A1 (fr) |
| ES (1) | ES8604542A1 (fr) |
| IL (1) | IL75533A (fr) |
Families Citing this family (27)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3505902A1 (de) * | 1985-02-21 | 1986-08-21 | Bayer Ag, 5090 Leverkusen | 4,5-disubstituierte 1,3-thiazol-2-yloxyacetamide |
| DE3724467A1 (de) * | 1987-07-24 | 1989-02-02 | Bayer Ag | 6-chlorbenzoxazolyl-oxyacetanilide |
| NZ225999A (en) * | 1987-09-10 | 1992-04-28 | Merck Sharp & Dohme | Azacyclic- or azabicyclic-substituted thiadiazole derivatives and pharmaceutical compositions |
| DE3821600A1 (de) | 1988-06-27 | 1989-12-28 | Bayer Ag | Heteroaryloxyessigsaeure-n-isopropylanilide |
| DE4003436A1 (de) * | 1990-02-06 | 1991-08-08 | Bayer Ag | Verfahren zur herstellung von 2-alkylthio-1,3,4-thiadiazolen |
| DE4133673A1 (de) * | 1991-10-11 | 1993-04-15 | Bayer Ag | Neue 2- (2-benzoxazolyl-oxy)-acetamide |
| DE4225024A1 (de) | 1992-07-29 | 1994-02-03 | Bayer Ag | Chlorthiazolderivate |
| US5547967A (en) * | 1993-12-08 | 1996-08-20 | Kali-Chemie Pharma Gmbh | (Phenylalkylaminoalkyloxy)-heteroaryl-compounds, processes and intermediates for their production and pharmaceutical compositions containing them |
| DE19530767A1 (de) * | 1995-08-22 | 1997-02-27 | Bayer Ag | N-(1-Isopropyl-2-methyl-1-propenyl) -heteroaryloxyacetamide |
| KR20010032160A (ko) * | 1997-11-18 | 2001-04-16 | 윌리암 에이취 캘넌, 에곤 이 버그 | 제초성 엔-알케닐 헤테로아릴일옥시아세트아미드 |
| CA2254579C (fr) * | 1997-12-12 | 2007-10-30 | Bayer Corporation | Synthese du 2-(methylsulfonyl)-5-(trifluoromethyle)-1,3,4-thiadiazole par l'oxydation de 2-(methylthio)-5-(trifluoromethyle)-1,3,4-thiadiazole avec un catalysateur de molybdene oude tungstene |
| US5808153A (en) * | 1997-12-12 | 1998-09-15 | Prasad; Vidyanatha A. | Conversion of N-(4-fluorophenyl)-2-hydroxy-N-(1-methylethyl) acetamide acetate to N-4-fluorophenyl)-2-hydroxy-N-(1-methylethyl) acetamide |
| US6005114A (en) * | 1997-12-12 | 1999-12-21 | Bayer Corporation | Process for making 2-(methylthio)-5(trifluoromethyl)-1,3,4,-thiadiazole using methyldithiocarbazinate with trifluoroacetic acid with selective removal of 2,5-bis(methylthio)-1,3,4-thiadiazole |
| US5792872A (en) * | 1997-12-12 | 1998-08-11 | Bayer Corporation | Process for producing N-(4-fluorophenyl)-N-(1-methylethyl)-2- (5-trifluoromethyl-1,3,4-thiadiazol-2-yl)oxy!acetamide |
| US5895818A (en) * | 1997-12-12 | 1999-04-20 | Bayer Corporation | Process for making N-(4-fluorophenyl)-N-(1-methylethyl)-2- (5-trifuloromethyl)-1,3,4-thiadiazol-2-yl)oxy!acetamide using an aprotic, aromatic solvent |
| US5905157A (en) * | 1997-12-12 | 1999-05-18 | Bayer Corporation | Process for producing 2-(methylthio)-5-(trifluoromethyl)-1,3,4-thiadiazole using methyldithiocarbazinate and trifluoroacetic acid |
| US5852202A (en) * | 1997-12-12 | 1998-12-22 | Bayer Corporation | Process for isolating N-(4-fluorophenyl)-N-(1-methylethyl)-2- (5-trifluoromethyl)-1,3,4-thiadiazol-2-yl)oxy!acetamide |
| US5898074A (en) * | 1997-12-12 | 1999-04-27 | Bayer Corporation | Process for preparing 2-(methylthio)-5-(trifluoromethyl) -1,3,4-thiadiazole using methyldithiocarbazinate and a molar excess of trifluoroacetic acid with recovery of trifluoroacetic acid |
| US6031108A (en) * | 1998-09-16 | 2000-02-29 | Bayer Corporation | Process for the preparation of 2-(methylsulfonyl)-5-(trifluoromethyl)-1,3,4-thiadiazole (TDA sulfone) |
| DE19935964A1 (de) | 1999-07-30 | 2001-02-01 | Bayer Ag | 5-Chlordifluormethyl-1,3,4-thiadiazol-2-yl-oxyacetanilide |
| US6339042B1 (en) | 1999-11-29 | 2002-01-15 | American Cyanamid Co. | Herbicidal N-cyclohexadienyl heteroaryloxyacetamides |
| JP4513251B2 (ja) * | 2002-10-11 | 2010-07-28 | 住友化学株式会社 | チアジアゾール化合物およびその用途 |
| US8916550B2 (en) * | 2005-05-09 | 2014-12-23 | Hydra Biosciences, Inc. | Compounds for modulating TRPV3 function |
| EP2392328A1 (fr) * | 2005-05-09 | 2011-12-07 | Hydra Biosciences, Inc. | Composés pour moduler la fonction TRPV3 |
| US7998980B2 (en) | 2006-09-15 | 2011-08-16 | Hydra Biosciences, Inc. | Compounds for modulating TRPV3 function |
| CN106478547B (zh) * | 2016-08-30 | 2019-02-01 | 京博农化科技股份有限公司 | 一种2-甲砜基-5-三氟甲基-1,3,4-噻二唑的合成方法 |
| WO2021154966A1 (fr) | 2020-01-29 | 2021-08-05 | Kamari Pharma Ltd. | Composés et compositions pour leur utilisation dans le traitement de troubles cutanés |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0005501B1 (fr) * | 1978-05-20 | 1981-11-25 | Bayer Ag | Heteroaryloxy-acetamides, procédé pour leur préparation et leur utilisation comme herbicides |
| DE3060330D1 (en) * | 1979-04-06 | 1982-06-09 | Bayer Ag | Azolyloxy-acetamides, process for their preparation and their use as herbicides |
| EP0022750B1 (fr) * | 1979-07-13 | 1983-05-18 | Ciba-Geigy Ag | 1,3,4-Thiadiazolyloxy-phényl urées, leur préparation et herbicides les contenant |
| DE2946524A1 (de) * | 1979-11-17 | 1981-06-11 | Bayer Ag, 5090 Leverkusen | Azolyloxy-carbonsaeure-n-oxy-amide, verfahren zu ihrer herstellung und ihre verwendung als herbizide |
| DE3027483A1 (de) * | 1980-07-19 | 1982-02-25 | Hoechst Ag, 6000 Frankfurt | Verfahren zur herstellung heterocyclisch substituierter 4-oxiphenoxialkancarbonsaeurederivate |
| DE3038636A1 (de) * | 1980-10-13 | 1982-05-27 | Bayer Ag, 5090 Leverkusen | Verfahren zur herstellung von substituierten oxyessigsaeureamiden |
| DE3148839A1 (de) * | 1981-12-10 | 1983-06-23 | Bayer Ag, 5090 Leverkusen | Verfahren zur herstellung von hetaryloxyacetamiden |
| DE3400168A1 (de) * | 1984-01-04 | 1985-07-11 | Bayer Ag, 5090 Leverkusen | 5-halogenalkyl-1,3,4-thiadiazol-2-yloxyacetamide |
| DE3418168A1 (de) * | 1984-05-16 | 1985-11-21 | Bayer Ag, 5090 Leverkusen | 6-chlorbenzazolyloxyacetamide |
-
1984
- 1984-06-20 DE DE19843422861 patent/DE3422861A1/de not_active Withdrawn
-
1985
- 1985-06-10 EP EP85107108A patent/EP0165537B1/fr not_active Expired - Lifetime
- 1985-06-10 DE DE8585107108T patent/DE3575423D1/de not_active Expired - Lifetime
- 1985-06-17 IL IL75533A patent/IL75533A/xx not_active IP Right Cessation
- 1985-06-17 JP JP60130072A patent/JPH0714925B2/ja not_active Expired - Fee Related
- 1985-06-19 ES ES544341A patent/ES8604542A1/es not_active Expired
- 1985-06-20 KR KR1019850004370A patent/KR920010393B1/ko not_active Expired
-
1991
- 1991-03-07 US US07/668,796 patent/US5101034A/en not_active Expired - Lifetime
Also Published As
| Publication number | Publication date |
|---|---|
| JPS6117575A (ja) | 1986-01-25 |
| ES8604542A1 (es) | 1986-02-01 |
| US5101034A (en) | 1992-03-31 |
| EP0165537A2 (fr) | 1985-12-27 |
| IL75533A0 (en) | 1985-10-31 |
| EP0165537B1 (fr) | 1990-01-17 |
| DE3422861A1 (de) | 1986-01-02 |
| KR920010393B1 (ko) | 1992-11-27 |
| KR860000272A (ko) | 1986-01-27 |
| EP0165537A3 (en) | 1987-03-04 |
| JPH0714925B2 (ja) | 1995-02-22 |
| ES544341A0 (es) | 1986-02-01 |
| DE3575423D1 (de) | 1990-02-22 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| NZ213844A (en) | Preparation of 1-hydroxyvitamin d compounds | |
| IL76753A0 (en) | Preparation of 1alpha-hydroxy-vitamin d compounds | |
| DE3571613D1 (en) | Preparation of (threo)-1-aryl-2-acylamido-3-fluoro-1-propanols | |
| IL75533A0 (en) | Preparation of heteroaryloxyacetamides | |
| GB8509322D0 (en) | Determination of microconstituent | |
| IL74661A0 (en) | Preparation of proteins | |
| GB2167739B (en) | Preparation of materials | |
| IL74751A (en) | Preparation of cephalosporins | |
| DE3573772D1 (en) | Preparation process of 2-chloropropionaldehyde | |
| IL80305A0 (en) | Preparation of epsilon-butyrolactams | |
| GB8507789D0 (en) | Preparation of 2-amino-s-triazines | |
| IL76249A0 (en) | Preparation of fluoroformates | |
| GB8529729D0 (en) | Preparation of fish-noodles | |
| GB8530319D0 (en) | Preparation of alcohols | |
| DE3566540D1 (en) | Preparation of fluoropyridines | |
| IL75811A0 (en) | Preparation of quinoline-and naphthyridone-carboxylic acids | |
| IL80657A0 (en) | Preparation of monochloropinacolone | |
| IL78379A0 (en) | Preparation of 2- ercaptobenzoxazoles | |
| AU566580B2 (en) | Preparation of 1-azidoaldoses | |
| GB8422162D0 (en) | Preparation of alkyfurans | |
| IL76216A0 (en) | Preparation of sulphonylisoureas and-thioureas | |
| GB8520403D0 (en) | Preparation of aminolactone | |
| IL78977A (en) | Preparation of alkyloxiranes | |
| GB8426101D0 (en) | Preparation of barbiturates | |
| DE3566532D1 (en) | Preparation of 4-fluorophenols |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| KB | Patent renewed | ||
| KB | Patent renewed | ||
| EXP | Patent expired |