IL78250A - 1,2-benzisoxazol-3-yl and 1,2-benzisothiazol-3-yl derivatives,their preparation and pharmaceutical compositions containing them - Google Patents

1,2-benzisoxazol-3-yl and 1,2-benzisothiazol-3-yl derivatives,their preparation and pharmaceutical compositions containing them

Info

Publication number: IL78250A
Authority: IL; Israel
Prior art keywords: halo; alkyl; benzisothiazol; benzisoxazol; derivatives
Prior art date: 1985-03-27

Application number

IL78250A

Other languages

English (en)

Other versions

IL78250A0 (en

Original Assignee

Janssen Pharmaceutica Nv

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1985-03-27

Filing date

1986-03-25

Publication date

1991-05-12

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=24880589&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=IL78250(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

1986-03-25 Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv

1986-07-31 Publication of IL78250A0 publication Critical patent/IL78250A0/xx

1991-05-12 Publication of IL78250A publication Critical patent/IL78250A/xx

Links

-1 1,2-benzisoxazol-3-yl Chemical class 0.000 title 2
239000008194 pharmaceutical composition Substances 0.000 title 1
125000000217 alkyl group Chemical group 0.000 abstract 7
125000005843 halogen group Chemical group 0.000 abstract 7
125000003545 alkoxy group Chemical group 0.000 abstract 3
NQRYJNQNLNOLGT-UHFFFAOYSA-N Piperidine Chemical compound C1CCNCC1 NQRYJNQNLNOLGT-UHFFFAOYSA-N 0.000 abstract 2
239000002253 acid Substances 0.000 abstract 1
125000005236 alkanoylamino group Chemical group 0.000 abstract 1
125000000852 azido group Chemical group *N=[N+]=[N-] 0.000 abstract 1
125000000051 benzyloxy group Chemical group [H]C1=C([H])C([H])=C(C([H])=C1[H])C([H])([H])O* 0.000 abstract 1
125000000816 ethylene group Chemical group [H]C([H])([*:1])C([H])([H])[*:2] 0.000 abstract 1
125000002924 primary amino group Chemical group [H]N([H])* 0.000 abstract 1
150000003839 salts Chemical class 0.000 abstract 1
125000003258 trimethylene group Chemical group [H]C([H])([*:2])C([H])([H])C([H])([H])[*:1] 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Thiazole And Isothizaole Compounds (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Plural Heterocyclic Compounds (AREA)
Other In-Based Heterocyclic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)

IL78250A 1985-03-27 1986-03-25 1,2-benzisoxazol-3-yl and 1,2-benzisothiazol-3-yl derivatives,their preparation and pharmaceutical compositions containing them IL78250A (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US71706785A	1985-03-27	1985-03-27

Publications (2)

Publication Number	Publication Date
IL78250A0 IL78250A0 (en)	1986-07-31
IL78250A true IL78250A (en)	1991-05-12

Family

ID=24880589

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
IL78250A IL78250A (en)	1985-03-27	1986-03-25	1,2-benzisoxazol-3-yl and 1,2-benzisothiazol-3-yl derivatives,their preparation and pharmaceutical compositions containing them

Country Status (13)

Country	Link
KR (1)	KR910000165B1 (de)
AT (1)	ATE79379T1 (de)
DE (1)	DE3686341T2 (de)
ES (1)	ES8705881A1 (de)
FI (1)	FI81800C (de)
GR (1)	GR860800B (de)
HU (1)	HU195793B (de)
IL (1)	IL78250A (de)
NO (2)	NO162765C (de)
NZ (1)	NZ215462A (de)
PH (1)	PH24016A (de)
PT (1)	PT82254B (de)
ZA (1)	ZA862279B (de)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
ES2050069B1 (es) *	1992-07-10	1994-12-16	Vita Invest Sa	Procedimiento para la obtencion de 3-(2-(4-(6-fluoro-1,2-benzisoxazol-3-il)piperidino)etil)-2-metil-6,7,8,9-tetrahidro-4h-pirido(1,2-a) pirimidin-4-ona.
ES2085234B1 (es) *	1994-02-24	1997-01-16	Vita Invest Sa	Agente activo sobre el sistema nervioso central, procedimiento para su preparacion y composiciones farmaceuticas que lo contienen.
HUP0402163A2 (en) *	2004-10-25	2006-05-29	Richter Gedeon Vegyeszet	Process for the preparation of risperidone

1986
- 1986-02-10 KR KR1019860000902A patent/KR910000165B1/ko not_active Expired
- 1986-03-12 NZ NZ215462A patent/NZ215462A/xx unknown
- 1986-03-13 AT AT86200400T patent/ATE79379T1/de active
- 1986-03-13 DE DE8686200400T patent/DE3686341T2/de not_active Expired - Lifetime
- 1986-03-24 PT PT82254A patent/PT82254B/pt unknown
- 1986-03-25 IL IL78250A patent/IL78250A/xx unknown
- 1986-03-25 ES ES553419A patent/ES8705881A1/es not_active Expired
- 1986-03-26 HU HU861278A patent/HU195793B/hu unknown
- 1986-03-26 GR GR860800A patent/GR860800B/el unknown
- 1986-03-26 ZA ZA862279A patent/ZA862279B/xx unknown
- 1986-03-26 PH PH33589A patent/PH24016A/en unknown
- 1986-03-26 NO NO861230A patent/NO162765C/no unknown
- 1986-03-26 FI FI861328A patent/FI81800C/fi not_active IP Right Cessation
1994
- 1994-11-03 NO NO1994021C patent/NO1994021I1/no unknown

Also Published As

Publication number	Publication date
DE3686341D1 (de)	1992-09-17
FI81800C (fi)	1990-12-10
FI81800B (fi)	1990-08-31
ES8705881A1 (es)	1987-05-16
PH24016A (en)	1990-02-09
FI861328A7 (fi)	1986-09-28
GR860800B (en)	1986-07-21
ATE79379T1 (de)	1992-08-15
PT82254A (en)	1986-04-01
DE3686341T2 (de)	1993-01-14
KR860007247A (ko)	1986-10-10
PT82254B (pt)	1988-04-21
IL78250A0 (en)	1986-07-31
HUT42461A (en)	1987-07-28
NO861230L (no)	1986-09-29
NZ215462A (en)	1988-09-29
FI861328A0 (fi)	1986-03-26
KR910000165B1 (ko)	1991-01-21
ZA862279B (en)	1987-11-25
HU195793B (en)	1988-07-28
NO162765B (no)	1989-11-06
ES553419A0 (es)	1987-05-16
NO162765C (no)	1990-02-14
NO1994021I1 (no)	1994-11-03

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Legal Events

Date	Code	Title
1996-06-18	KB	Patent renewed
2000-08-13	KB	Patent renewed
2004-06-01	KB	Patent renewed