PT82254B - Processo para a preparacao de novos derivados de 1,2-benzisoxazol-3-ilo e 1,2-benzisotiazol-3-ilo - Google Patents

Processo para a preparacao de novos derivados de 1,2-benzisoxazol-3-ilo e 1,2-benzisotiazol-3-ilo

Info

Publication number
PT82254B
PT82254B PT82254A PT8225486A PT82254B PT 82254 B PT82254 B PT 82254B PT 82254 A PT82254 A PT 82254A PT 8225486 A PT8225486 A PT 8225486A PT 82254 B PT82254 B PT 82254B
Authority
PT
Portugal
Prior art keywords
halo
alkyl
ilo
new
benzisozyazole
Prior art date
Application number
PT82254A
Other languages
English (en)
Portuguese (pt)
Other versions
PT82254A (en
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=24880589&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PT82254(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of PT82254A publication Critical patent/PT82254A/pt
Publication of PT82254B publication Critical patent/PT82254B/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
PT82254A 1985-03-27 1986-03-24 Processo para a preparacao de novos derivados de 1,2-benzisoxazol-3-ilo e 1,2-benzisotiazol-3-ilo PT82254B (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US71706785A 1985-03-27 1985-03-27

Publications (2)

Publication Number Publication Date
PT82254A PT82254A (en) 1986-04-01
PT82254B true PT82254B (pt) 1988-04-21

Family

ID=24880589

Family Applications (1)

Application Number Title Priority Date Filing Date
PT82254A PT82254B (pt) 1985-03-27 1986-03-24 Processo para a preparacao de novos derivados de 1,2-benzisoxazol-3-ilo e 1,2-benzisotiazol-3-ilo

Country Status (13)

Country Link
KR (1) KR910000165B1 (de)
AT (1) ATE79379T1 (de)
DE (1) DE3686341T2 (de)
ES (1) ES8705881A1 (de)
FI (1) FI81800C (de)
GR (1) GR860800B (de)
HU (1) HU195793B (de)
IL (1) IL78250A (de)
NO (2) NO162765C (de)
NZ (1) NZ215462A (de)
PH (1) PH24016A (de)
PT (1) PT82254B (de)
ZA (1) ZA862279B (de)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2050069B1 (es) * 1992-07-10 1994-12-16 Vita Invest Sa Procedimiento para la obtencion de 3-(2-(4-(6-fluoro-1,2-benzisoxazol-3-il)piperidino)etil)-2-metil-6,7,8,9-tetrahidro-4h-pirido(1,2-a) pirimidin-4-ona.
ES2085234B1 (es) * 1994-02-24 1997-01-16 Vita Invest Sa Agente activo sobre el sistema nervioso central, procedimiento para su preparacion y composiciones farmaceuticas que lo contienen.
HUP0402163A2 (en) * 2004-10-25 2006-05-29 Richter Gedeon Vegyeszet Process for the preparation of risperidone

Also Published As

Publication number Publication date
DE3686341D1 (de) 1992-09-17
FI81800C (fi) 1990-12-10
FI81800B (fi) 1990-08-31
ES8705881A1 (es) 1987-05-16
PH24016A (en) 1990-02-09
FI861328A7 (fi) 1986-09-28
GR860800B (en) 1986-07-21
ATE79379T1 (de) 1992-08-15
PT82254A (en) 1986-04-01
DE3686341T2 (de) 1993-01-14
KR860007247A (ko) 1986-10-10
IL78250A0 (en) 1986-07-31
HUT42461A (en) 1987-07-28
NO861230L (no) 1986-09-29
IL78250A (en) 1991-05-12
NZ215462A (en) 1988-09-29
FI861328A0 (fi) 1986-03-26
KR910000165B1 (ko) 1991-01-21
ZA862279B (en) 1987-11-25
HU195793B (en) 1988-07-28
NO162765B (no) 1989-11-06
ES553419A0 (es) 1987-05-16
NO162765C (no) 1990-02-14
NO1994021I1 (no) 1994-11-03

Similar Documents

Publication Publication Date Title
NO177424C (no) Analogifremgangsmåte for fremstilling av terapeutisk aktive N-(4-piperidinyl)(dihydrobenzofuran- eller dihydro-2H-benzopyran)karboksamidderivater samt mellomprodukter
NO2007017I2 (no) 3-[2-[4-(6-fluor-1,2-benzoksazol-3-yl)-1-piperidinyl]etyl]-6,7,8,9-tetrahydro-9-hydroksy-2-metyl-4H-pyridol]1,2-a]pyrimidin-4-on(palperidone)
ES2085259T3 (es) Uso de ciertos antagonistas del receptor 5-ht3 en el tratamiento del dolor visceral.
MXPA04003474A (es) Imidazo (4,3-e)-1,2,4-triazolo(1,5-c) pirimidinas como antagonistas del receptor de adenosina a2a.
ZA885788B (en) 2-((4-piperidyl)methyl)-1,2,3,4-tetrahydro-9h-pyrido(3,4-b)indole derivatives,their preparation and their application in therapy
PT96255A (pt) Processo para a preparacao de novos derivados da 1-naftil-piperazina
AR036864A1 (es) Uso de compuestos de acido benzacepin-n-acetico, y procedimiento para la preparacion de dichos compuestos
PT82254B (pt) Processo para a preparacao de novos derivados de 1,2-benzisoxazol-3-ilo e 1,2-benzisotiazol-3-ilo
ATE127466T1 (de) Antivirale purin-derivate und verfahren zu ihrer herstellung.
DE3368414D1 (en) 1,4-dihydropyridines, processes for their preparation and their use in medicines
RU2003106191A (ru) Способ лечения аллергии с использованием замещенных пиразолов
CO5200845A1 (es) Derivados del acido monociclico 4-fenilbutanoico como antagonista del receptor vitronectina
NO20052360L (no) Forbedrede formuleringer inneholdende substituerte imidazolderivater
HUP0104873A2 (hu) Javított eljárás 3-{2-[4-(6-fluor-1,2-benzizoxazol-3-il)-1-piperidinil]-etil}-6,7,8,9-tetrahidro-2-metil-4H-pirido[1,2-a]pirimidin-4-on előállítására
DE60122350D1 (de) Benzoesaüre derivate und deren verwendung
RU2003106190A (ru) Способ лечения аллергии с использованием замещенных пиразолов
DE3474958D1 (en) 1-(aminoalkylphenyl and aminoalkylbenzyl)-indoles and indolines, a process for their preparation and their use as medicaments
PT84247A (en) Process for the preparation of purine derivatives and pharmaceutical compositions
HUT60742A (en) Method for producing imidqzo-benzodiazepine-2-(1h)-one derivatives and pharmaceutical preparatives containing them
PT78465A (en) 1-(aminoalkylphenyl and aminoalkylbenzyl) - indoles and indolines a process for their preparation and their use as medicaments
PT91204A (pt) Processo para a preparacao de derivados de 3-piranona e de seus analogos
MX9703074A (es) Inhibidores de sintesis de apoliproteina-b.