IL87468A - Polymorphic modification of buspirone and pharmaceutical compositions containing it - Google Patents

Polymorphic modification of buspirone and pharmaceutical compositions containing it

Info

Publication number
IL87468A
IL87468A IL87468A IL8746888A IL87468A IL 87468 A IL87468 A IL 87468A IL 87468 A IL87468 A IL 87468A IL 8746888 A IL8746888 A IL 8746888A IL 87468 A IL87468 A IL 87468A
Authority
IL
Israel
Prior art keywords
buspirone
pharmaceutical compositions
compositions containing
polymorphic modification
polymorphic
Prior art date
Application number
IL87468A
Other languages
English (en)
Other versions
IL87468A0 (en
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=22225222&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=IL87468(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Publication of IL87468A0 publication Critical patent/IL87468A0/xx
Publication of IL87468A publication Critical patent/IL87468A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Epidemiology (AREA)
  • Anesthesiology (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Addition Polymer Or Copolymer, Post-Treatments, Or Chemical Modifications (AREA)
  • Body Structure For Vehicles (AREA)
IL87468A 1987-08-28 1988-08-16 Polymorphic modification of buspirone and pharmaceutical compositions containing it IL87468A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US07/090,984 US5015646A (en) 1987-08-28 1987-08-28 Pharmaceutically useful polymorphic modification of buspirone

Publications (2)

Publication Number Publication Date
IL87468A0 IL87468A0 (en) 1989-01-31
IL87468A true IL87468A (en) 1992-12-01

Family

ID=22225222

Family Applications (1)

Application Number Title Priority Date Filing Date
IL87468A IL87468A (en) 1987-08-28 1988-08-16 Polymorphic modification of buspirone and pharmaceutical compositions containing it

Country Status (22)

Country Link
US (1) US5015646A (de)
EP (1) EP0304941B1 (de)
JP (1) JP2716740B2 (de)
KR (1) KR970011297B1 (de)
AT (1) ATE101147T1 (de)
AU (1) AU618549B2 (de)
CY (1) CY1785A (de)
DE (1) DE3887598T2 (de)
DK (1) DK170821B1 (de)
ES (1) ES2061576T3 (de)
FI (1) FI883961L (de)
HK (1) HK74494A (de)
HU (1) HU201322B (de)
IE (1) IE63071B1 (de)
IL (1) IL87468A (de)
MY (1) MY104061A (de)
NO (1) NO883805D0 (de)
NZ (1) NZ225896A (de)
OA (1) OA08908A (de)
PT (1) PT88356B (de)
YU (1) YU46962B (de)
ZA (1) ZA886082B (de)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4810789A (en) * 1987-08-28 1989-03-07 Bristol-Myers Company Process for buspirone hydrochloride polymorphic crystalline form conversion
US5631017A (en) * 1993-03-26 1997-05-20 Beth Israel Deaconess Medical Center, Inc. Topical application of buspirone for treatment of pathological conditions associated with immune responses
US5484788A (en) * 1993-03-26 1996-01-16 Beth Israel Hospital Association Buspirone as a systemic immunosuppressant
HU217129B (hu) * 1993-07-16 1999-11-29 EGIS Gyógyszergyár Rt. Eljárás nagy tisztaságú buspiron gyógyászati hatóanyag előállítására
US5637314A (en) * 1995-06-07 1997-06-10 Beth Israel Deaconess Medical Center, Inc. Topical and systemic application of buspirone or derivatives thereof for treating atopic dermatitis
CA2566652C (en) 1998-06-19 2008-10-21 Teijin Limited Polymorphic modifications of 2-(3-cyano-4-isobutyloxyphenyl)-4-methyl-5-thiazole-carboxylic acid and processes for the preparation thereof
US6465255B1 (en) * 1999-01-29 2002-10-15 The Regents Of The University Of California Method for identifying and probing phase transitions in materials
KR100433165B1 (ko) * 2000-10-10 2004-05-27 엔앤비텍 주식회사 가공란의 제조 방법, 상기 방법에 의하여 제조된 가공란,및 가공란을 제조하기 위한 장치
CL2004001034A1 (es) 2003-05-14 2005-03-28 Teijin Pharma Ltd Formas cristalinas de acido 4-(1-((,etilbenzotiofen-3-il)me til)benzimidazol-2-iltio)butanoico; procedimiento de preparacion de las formas cristalinas; composicion farmaceutica; y su uso para el tratamiento de enfermedades inflamatorias, alergicas, r
EP1750766B1 (de) 2004-05-11 2013-07-03 Emotional Brain B.V. Pharmazeutische Formulierungen und ihre Verwendungen bei der Behandlung von weiblicher sexueller Dysfunktion
JPWO2006052026A1 (ja) * 2004-11-12 2008-05-29 帝人ファーマ株式会社 ベンズイミダゾール誘導体の酸性塩及びその結晶
EP1790343A1 (de) 2005-11-11 2007-05-30 Emotional Brain B.V. Pharmazeutische Zusammensetzungen und deren Verwendung zur Behandlung sexueller Störungen der Frau
EP1925307A1 (de) * 2006-11-03 2008-05-28 Emotional Brain B.V. Verwendung von 3-alpha-androstanediol zur Behandlung sexueller Dysfunktion
CN118702676B (zh) * 2024-07-09 2026-01-27 济南大学 一种盐酸丁螺环酮晶型ii的制备方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE759371A (fr) * 1969-11-24 1971-05-24 Bristol Myers Co Azaspirodecanediones heterocycliques et procedes pour leur preparation
US3976776A (en) * 1972-12-06 1976-08-24 Mead Johnson & Company Tranquilizer process employing N-(heteroarcyclic)piperazinylalkylazaspiroalkanediones
US4351939A (en) * 1980-10-16 1982-09-28 Mead Johnson & Company Spiro-quaternary ammonium halides and N-(2-pyrimidinyl)piperazinylalkylazaspiroalkanedione process
US4476248A (en) * 1983-02-28 1984-10-09 The Upjohn Company Crystallization of ibuprofen

Also Published As

Publication number Publication date
NO883805D0 (no) 1988-08-25
OA08908A (en) 1989-10-31
ZA886082B (en) 1989-04-26
IL87468A0 (en) 1989-01-31
MY104061A (en) 1993-11-30
AU618549B2 (en) 1992-01-02
FI883961A7 (fi) 1989-03-01
DK478788D0 (da) 1988-08-26
NZ225896A (en) 1991-04-26
ES2061576T3 (es) 1994-12-16
HK74494A (en) 1994-08-05
FI883961A0 (fi) 1988-08-26
DE3887598D1 (de) 1994-03-17
PT88356A (pt) 1989-06-30
KR970011297B1 (ko) 1997-07-09
IE882528L (en) 1989-02-28
YU46962B (sh) 1994-09-09
DE3887598T2 (de) 1994-05-19
DK478788A (da) 1989-03-01
JPS6471816A (en) 1989-03-16
DK170821B1 (da) 1996-01-29
IE63071B1 (en) 1995-03-22
JP2716740B2 (ja) 1998-02-18
HUT47564A (en) 1989-03-28
AU2107688A (en) 1989-03-02
ATE101147T1 (de) 1994-02-15
FI883961L (fi) 1989-03-01
EP0304941A1 (de) 1989-03-01
YU161688A (en) 1990-10-31
CY1785A (en) 1995-10-20
EP0304941B1 (de) 1994-02-02
HU201322B (en) 1990-10-28
KR890003740A (ko) 1989-04-17
PT88356B (pt) 1995-03-31
US5015646A (en) 1991-05-14

Similar Documents

Publication Publication Date Title
IL87468A0 (en) Polymorphic modification of buspirone and pharmaceutical compositions containing it
EP0363415A4 (en) Compounds for the treatment of alzheimer's disease
EP0397697A4 (en) Quinoline derivatives as antagonists of leukotriene d 4?
LTIP919A (en) Drugs and process for preparing thereof
EP0328251A3 (en) 2-(2-hydroxy-3-phenoxypropylamino)ethylphenoxyacetamides and processes and intermediates for their preparation
IL86423A0 (en) Pharmaceutical compositions for the treatment of alzheimer's disease
PT87294A (pt) Process for the preparation of 17beta-(cyclopropylamino)-androst-5-en-3beta-ol and related compounds useful as c17-20 lyase inhibitors and of pharmaceutical compositions containing the same
HU904201D0 (en) Process for producing peptides with haemoregulating effect and pharmaceutical preparatives containing these compounds
EP0328634A4 (en) Pharmaceutical compositions for the treatment of psoriasis
HUT47263A (en) Process for production of 5-/3-alkyl-5-terc-butil/-4-hydroxi-phenil/-2-amino-6h-1,3,4-tiadiasines and medical compositions containing them
YU130089A (en) Process for obtaining nedocromyl calcium compounds
IL74351A (en) 4-(cyclic amino)carbonyl isoxazole derivatives,process for their preparation and medicaments containing these compounds
ES2009689A6 (es) Procedimiento para preparar derivados de 3-piperidina-carbaldehido-oxima.
HUT57209A (en) Process for producing hydroxymethyl-indolizidine and kinolizidine derivatives and pharmaceutical compositions containing them
ZA88639B (en) Substituted 3-phenyl-7h-thiazolo(3,2-b)(1,2,4)triazin-7-ones,a process for the preparation thereof,medicaments containing same and the use thereof,and also some intermediates formed in the preparation of the compounds mentioned
IL70452A0 (en) 6alpha-methylprednisolone derivatives,process for the manufacture thereof and pharmaceutical compositions containing the same
IL86151A (en) Antiasthmatic compositions comprising 2-(2-phenyl-2-(2-pyridyl)) ethyl-2-imidazoline

Legal Events

Date Code Title Description
KB Patent renewed
KB Patent renewed
MM9K Patent not in force due to non-payment of renewal fees