IL88629A - Macrolides, their production and pharmaceutical compositions containing them - Google Patents

Macrolides, their production and pharmaceutical compositions containing them

Info

Publication number
IL88629A
IL88629A IL8862988A IL8862988A IL88629A IL 88629 A IL88629 A IL 88629A IL 8862988 A IL8862988 A IL 8862988A IL 8862988 A IL8862988 A IL 8862988A IL 88629 A IL88629 A IL 88629A
Authority
IL
Israel
Prior art keywords
compound
hydroxy
dioxa
formula
dimethoxy
Prior art date
Application number
IL8862988A
Other languages
English (en)
Original Assignee
Fisons Plc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB878728821A external-priority patent/GB8728821D0/en
Priority claimed from GB878728820A external-priority patent/GB8728820D0/en
Priority claimed from GB888803372A external-priority patent/GB8803372D0/en
Priority claimed from GB888803374A external-priority patent/GB8803374D0/en
Priority claimed from GB888803371A external-priority patent/GB8803371D0/en
Priority claimed from GB888803373A external-priority patent/GB8803373D0/en
Priority claimed from GB888803375A external-priority patent/GB8803375D0/en
Priority claimed from GB888803377A external-priority patent/GB8803377D0/en
Priority claimed from GB888803370A external-priority patent/GB8803370D0/en
Priority claimed from GB888809174A external-priority patent/GB8809174D0/en
Priority claimed from GB888817624A external-priority patent/GB8817624D0/en
Priority claimed from GB888818426A external-priority patent/GB8818426D0/en
Application filed by Fisons Plc filed Critical Fisons Plc
Publication of IL88629A publication Critical patent/IL88629A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D498/18—Bridged systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/22—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains four or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Immunology (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Transplantation (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Saccharide Compounds (AREA)
  • Solid-Sorbent Or Filter-Aiding Compositions (AREA)
  • Steroid Compounds (AREA)
  • Heterocyclic Compounds That Contain Two Or More Ring Oxygen Atoms (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
IL8862988A 1987-12-09 1988-12-08 Macrolides, their production and pharmaceutical compositions containing them IL88629A (en)

Applications Claiming Priority (12)

Application Number Priority Date Filing Date Title
GB878728821A GB8728821D0 (en) 1987-12-09 1987-12-09 Compounds
GB878728820A GB8728820D0 (en) 1987-12-09 1987-12-09 Compounds
GB888803374A GB8803374D0 (en) 1988-02-13 1988-02-13 Compound
GB888803371A GB8803371D0 (en) 1988-02-13 1988-02-13 Compound
GB888803372A GB8803372D0 (en) 1988-02-13 1988-02-13 Compound
GB888803373A GB8803373D0 (en) 1988-02-13 1988-02-13 Compound
GB888803375A GB8803375D0 (en) 1988-02-13 1988-02-13 Compound
GB888803377A GB8803377D0 (en) 1988-02-13 1988-02-13 Compound
GB888803370A GB8803370D0 (en) 1988-02-13 1988-02-13 Compound
GB888809174A GB8809174D0 (en) 1988-04-19 1988-04-19 Compounds
GB888817624A GB8817624D0 (en) 1988-07-23 1988-07-23 Compounds
GB888818426A GB8818426D0 (en) 1988-08-03 1988-08-03 Compounds

Publications (1)

Publication Number Publication Date
IL88629A true IL88629A (en) 1994-04-12

Family

ID=27583057

Family Applications (1)

Application Number Title Priority Date Filing Date
IL8862988A IL88629A (en) 1987-12-09 1988-12-08 Macrolides, their production and pharmaceutical compositions containing them

Country Status (16)

Country Link
EP (2) EP0323042A1 (fr)
JP (1) JP2799208B2 (fr)
KR (1) KR900700494A (fr)
CN (1) CN1033458A (fr)
AT (1) ATE120466T1 (fr)
AU (1) AU630866B2 (fr)
CA (1) CA1339128C (fr)
DE (1) DE3853477T2 (fr)
DK (1) DK387889A (fr)
ES (1) ES2071681T3 (fr)
FI (1) FI90550C (fr)
IE (1) IE66163B1 (fr)
IL (1) IL88629A (fr)
NO (1) NO893166D0 (fr)
NZ (1) NZ227251A (fr)
WO (1) WO1989005304A1 (fr)

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EP0358508A3 (fr) * 1988-09-08 1991-03-20 Merck & Co. Inc. Composé immunosuppreseur
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US5268370A (en) * 1989-01-13 1993-12-07 Merck & Co., Inc. Microbial transformation product of L-679,934
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US4975372A (en) * 1989-01-13 1990-12-04 Merck & Co., Inc. Microbial transformation product of L-683,590
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EP0356399A3 (fr) * 1988-08-26 1991-03-20 Sandoz Ag Dérivés substitués du 4-azatricyclo (22.3.1.04.9) octacos-18-ène, leur préparation et les compositions pharmaceutiques les contenant

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DK387889D0 (da) 1989-08-08
EP0346427B1 (fr) 1995-03-29
CN1033458A (zh) 1989-06-21
EP0346427A1 (fr) 1989-12-20
ES2071681T3 (es) 1995-07-01
WO1989005304A1 (fr) 1989-06-15
IE66163B1 (en) 1995-12-13
AU630866B2 (en) 1992-11-12
FI90550C (fi) 1994-02-25
EP0323042A1 (fr) 1989-07-05
KR900700494A (ko) 1990-08-13
FI90550B (fi) 1993-11-15
IE883662L (en) 1989-06-09
DE3853477D1 (de) 1995-05-04
DE3853477T2 (de) 1995-11-09
AU2822889A (en) 1989-07-05
NO893166L (no) 1989-08-04
NZ227251A (en) 1990-02-26
JP2799208B2 (ja) 1998-09-17
FI893750A0 (fi) 1989-08-09
ATE120466T1 (de) 1995-04-15
JPH02502463A (ja) 1990-08-09
DK387889A (da) 1989-08-08
CA1339128C (fr) 1997-07-29
NO893166D0 (no) 1989-08-04

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