IL98231A - Pyrido (3,4-b) pyrrolo (1,2-e) (1,4,5) oxadiazepines and related analogs, a process for their preparation and their use as medicaments - Google Patents

Pyrido (3,4-b) pyrrolo (1,2-e) (1,4,5) oxadiazepines and related analogs, a process for their preparation and their use as medicaments

Info

Publication number
IL98231A
IL98231A IL9823191A IL9823191A IL98231A IL 98231 A IL98231 A IL 98231A IL 9823191 A IL9823191 A IL 9823191A IL 9823191 A IL9823191 A IL 9823191A IL 98231 A IL98231 A IL 98231A
Authority
IL
Israel
Prior art keywords
compound
loweralkyl
hydrogen
methyl
pyrido
Prior art date
Application number
IL9823191A
Other languages
English (en)
Other versions
IL98231A0 (en
Original Assignee
Hoechst Roussel Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Roussel Pharma filed Critical Hoechst Roussel Pharma
Publication of IL98231A0 publication Critical patent/IL98231A0/xx
Publication of IL98231A publication Critical patent/IL98231A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D498/14—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pain & Pain Management (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
IL9823191A 1990-05-25 1991-05-23 Pyrido (3,4-b) pyrrolo (1,2-e) (1,4,5) oxadiazepines and related analogs, a process for their preparation and their use as medicaments IL98231A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US07/529,082 US5015637A (en) 1990-05-25 1990-05-25 Pyrido[3,4-b]pyrrolo[1,2-e][1,4,5]oxadiazepines

Publications (2)

Publication Number Publication Date
IL98231A0 IL98231A0 (en) 1992-06-21
IL98231A true IL98231A (en) 1994-11-28

Family

ID=24108456

Family Applications (1)

Application Number Title Priority Date Filing Date
IL9823191A IL98231A (en) 1990-05-25 1991-05-23 Pyrido (3,4-b) pyrrolo (1,2-e) (1,4,5) oxadiazepines and related analogs, a process for their preparation and their use as medicaments

Country Status (22)

Country Link
US (1) US5015637A (cs)
EP (1) EP0458331B1 (cs)
JP (1) JP3090500B2 (cs)
KR (1) KR100286405B1 (cs)
AT (1) ATE183746T1 (cs)
AU (1) AU638572B2 (cs)
CA (1) CA2043229C (cs)
CS (1) CS157191A3 (cs)
DE (1) DE69131546T2 (cs)
DK (1) DK0458331T3 (cs)
ES (1) ES2135383T3 (cs)
FI (1) FI912499L (cs)
GR (1) GR3031538T3 (cs)
HU (1) HU207520B (cs)
IE (1) IE911788A1 (cs)
IL (1) IL98231A (cs)
MX (1) MX25922A (cs)
NO (1) NO911998L (cs)
NZ (1) NZ238238A (cs)
PL (1) PL290405A1 (cs)
PT (1) PT97762B (cs)
ZA (1) ZA913951B (cs)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE199569T1 (de) * 1993-05-27 2001-03-15 Univ Washington Cyclisch gmp bindende cyclisch gmp spezifische phosphodiesterase materialien und verfahren.
AR037853A1 (es) * 2001-12-18 2004-12-09 Syngenta Participations Ag Proceso para la preparacion de derivados de [1,4,5]-oxadiazepinas, y empleo de esos derivados en la preparacion de un herbicida del tipo de la tetrahidropirazolodiona
US8347435B2 (en) 2010-04-18 2013-01-08 Chang Jun Yu Pillow with positionable inserts

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4045448A (en) * 1976-02-26 1977-08-30 American Hoechst Corporation Pyrrolo[2,1-c][1,4]benzoxazepine and benzoxazocine derivatives
US4029672A (en) * 1976-02-26 1977-06-14 American Hoechst Corporation Aminoalkylpyrrolobenzoxazalkanes
EP0031115A1 (en) * 1979-12-21 1981-07-01 Sandoz Ag New pyrrolobenzotriazepines, their production and pharmaceutical compositions containing them
US4608374A (en) * 1983-11-07 1986-08-26 Hoechst-Roussel Pharmaceuticals Inc. 11-substituted 5H,11H-pyrrolo[2,1-c][1,4]benzoxazepines as antipsychotic and analgesic agents
US4794110A (en) * 1987-07-20 1988-12-27 Hoechst-Roussel Pharmaceuticals, Inc. 5-Aryl-11-substituted-5H,11H-pyrrolo[2,1-c][1,4]benzoxazepined as analgesic and hypotensive agents
US4879382A (en) * 1988-07-25 1989-11-07 Hoechst-Roussel Pharmaceuticals, Inc. Pyrido(3,4-f)pyrrolo(1,2-b)(1,2,5)triazepines

Also Published As

Publication number Publication date
PL290405A1 (en) 1992-08-24
EP0458331A1 (en) 1991-11-27
AU7621391A (en) 1991-11-28
PT97762A (pt) 1992-02-28
DE69131546D1 (de) 1999-09-30
FI912499A7 (fi) 1991-11-26
JPH04235186A (ja) 1992-08-24
NO911998L (no) 1991-11-26
ATE183746T1 (de) 1999-09-15
EP0458331B1 (en) 1999-08-25
HU207520B (en) 1993-04-28
CS157191A3 (en) 1992-01-15
GR3031538T3 (en) 2000-01-31
IE911788A1 (en) 1991-12-04
MX25922A (es) 1993-10-01
NZ238238A (en) 1993-06-25
CA2043229C (en) 2003-02-11
CA2043229A1 (en) 1991-11-26
ES2135383T3 (es) 1999-11-01
DE69131546T2 (de) 2000-03-23
JP3090500B2 (ja) 2000-09-18
FI912499L (fi) 1991-11-26
ZA913951B (en) 1992-03-25
AU638572B2 (en) 1993-07-01
IL98231A0 (en) 1992-06-21
KR910020018A (ko) 1991-12-19
PT97762B (pt) 1998-10-30
US5015637A (en) 1991-05-14
HU911755D0 (en) 1991-12-30
NO911998D0 (no) 1991-05-24
FI912499A0 (fi) 1991-05-23
KR100286405B1 (ko) 2001-04-16
DK0458331T3 (da) 2000-03-13
HUT60744A (en) 1992-10-28

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Legal Events

Date Code Title Description
KB Patent renewed
HC Change of name of proprietor(s)