IL98428A - 3-(1,2,4-oxadiazolyl) imidazo [1,5-a] quinazolineamine and quinoxalineamine compounds, their preparation and pharmaceutical compositions containing them - Google Patents
3-(1,2,4-oxadiazolyl) imidazo [1,5-a] quinazolineamine and quinoxalineamine compounds, their preparation and pharmaceutical compositions containing themInfo
- Publication number
- IL98428A IL98428A IL9842891A IL9842891A IL98428A IL 98428 A IL98428 A IL 98428A IL 9842891 A IL9842891 A IL 9842891A IL 9842891 A IL9842891 A IL 9842891A IL 98428 A IL98428 A IL 98428A
- Authority
- IL
- Israel
- Prior art keywords
- compound
- imidazo
- cyclopropyl
- set forth
- forth above
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Life Sciences & Earth Sciences (AREA)
- Neurology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Lubricants (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Plural Heterocyclic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DK151890A DK151890D0 (da) | 1990-06-22 | 1990-06-22 | Heterocykliske forbindelser deres fremstilling og brug |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| IL98428A0 IL98428A0 (en) | 1992-07-15 |
| IL98428A true IL98428A (en) | 1995-07-31 |
Family
ID=8105671
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL9842891A IL98428A (en) | 1990-06-22 | 1991-06-10 | 3-(1,2,4-oxadiazolyl) imidazo [1,5-a] quinazolineamine and quinoxalineamine compounds, their preparation and pharmaceutical compositions containing them |
Country Status (18)
| Country | Link |
|---|---|
| EP (1) | EP0535104B1 (ja) |
| JP (1) | JPH05507708A (ja) |
| KR (1) | KR930701442A (ja) |
| AT (1) | ATE142209T1 (ja) |
| AU (1) | AU662293B2 (ja) |
| CA (1) | CA2085591A1 (ja) |
| DE (1) | DE69121894T2 (ja) |
| DK (2) | DK151890D0 (ja) |
| ES (1) | ES2092571T3 (ja) |
| FI (1) | FI101072B (ja) |
| GR (1) | GR3021810T3 (ja) |
| IE (1) | IE911946A1 (ja) |
| IL (1) | IL98428A (ja) |
| NO (1) | NO302298B1 (ja) |
| NZ (1) | NZ238638A (ja) |
| PT (1) | PT98063B (ja) |
| WO (1) | WO1992000298A1 (ja) |
| ZA (1) | ZA914530B (ja) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DK204291D0 (da) * | 1991-12-20 | 1991-12-20 | Novo Nordisk As | Heterocykliske forbindelser deres fremstilling og anvendelse |
| US5792766A (en) | 1996-03-13 | 1998-08-11 | Neurogen Corporation | Imidazo 1,5-c! quinazolines; a new class of GABA brain receptor ligands |
| CN1052724C (zh) * | 1996-07-01 | 2000-05-24 | 瑞安大药厂股份有限公司 | 新的光学活性的2,3-二氢咪唑并[1,2-c]喹唑啉衍生物及其制备方法和用途 |
| ZA985870B (en) * | 1997-07-15 | 1999-01-27 | Dainippon Pharmaceutical Co | 5-substituted-3-oxadiazolyl-1, 6-naphthyridin-2(1H)-one derivatives |
| US6235740B1 (en) * | 1997-08-25 | 2001-05-22 | Bristol-Myers Squibb Co. | Imidazoquinoxaline protein tyrosine kinase inhibitors |
| US6635626B1 (en) * | 1997-08-25 | 2003-10-21 | Bristol-Myers Squibb Co. | Imidazoquinoxaline protein tyrosine kinase inhibitors |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DK476885D0 (da) * | 1985-10-17 | 1985-10-17 | Ferrosan As | Heterocycliske forbindelser og fremgangsmaader til fremstilling heraf |
| ATE44381T1 (de) * | 1985-10-17 | 1989-07-15 | Ferrosan As | Heterocyclische verbindungen und ihre herstellung und verwendung. |
| DK155524C (da) * | 1987-03-18 | 1989-09-11 | Ferrosan As | Kondenserede imidazolderivater og farmaceutiske praeparater indeholdende disse |
| DK160876C (da) * | 1987-12-08 | 1991-10-14 | Novo Nordisk As | Imidazoquinoxalinforbindelser, fremgangsmaade til deres fremstilling, anvendelse af forbindelserne og farmaceutiske praeparater, hvori forbindelserne indgaar |
| IL90315A0 (en) * | 1988-06-01 | 1989-12-15 | Ferrosan As | Imidazoquinoxaline compounds,their preparation and pharmaceutical compositions containing them |
| DK161148C (da) * | 1988-06-14 | 1991-11-18 | Novo Nordisk As | Imidazoquinoxalinforbindelser, fremgangsmaade til fremstilling deraf samt farmaceutiske praeprater indeholdende forbindelserne |
| DK588489D0 (da) * | 1989-11-22 | 1989-11-22 | Ferrosan As | Heterocykliske forbindelser, deres fremstilling og anvendelse |
| DK204291D0 (da) * | 1991-12-20 | 1991-12-20 | Novo Nordisk As | Heterocykliske forbindelser deres fremstilling og anvendelse |
| AU8396491A (en) * | 1990-09-04 | 1992-03-30 | Upjohn Company, The | Oxygenated quinoxalines |
-
1990
- 1990-06-22 DK DK151890A patent/DK151890D0/da not_active IP Right Cessation
-
1991
- 1991-06-07 IE IE194691A patent/IE911946A1/en unknown
- 1991-06-10 IL IL9842891A patent/IL98428A/en not_active IP Right Cessation
- 1991-06-13 ZA ZA914530A patent/ZA914530B/xx unknown
- 1991-06-20 NZ NZ238638A patent/NZ238638A/xx unknown
- 1991-06-21 DK DK91911908.1T patent/DK0535104T3/da active
- 1991-06-21 KR KR1019920703302A patent/KR930701442A/ko not_active Ceased
- 1991-06-21 DE DE69121894T patent/DE69121894T2/de not_active Expired - Fee Related
- 1991-06-21 WO PCT/DK1991/000170 patent/WO1992000298A1/en not_active Ceased
- 1991-06-21 AT AT91911908T patent/ATE142209T1/de not_active IP Right Cessation
- 1991-06-21 EP EP91911908A patent/EP0535104B1/en not_active Expired - Lifetime
- 1991-06-21 PT PT98063A patent/PT98063B/pt not_active IP Right Cessation
- 1991-06-21 AU AU80633/91A patent/AU662293B2/en not_active Ceased
- 1991-06-21 ES ES91911908T patent/ES2092571T3/es not_active Expired - Lifetime
- 1991-06-21 JP JP91511051A patent/JPH05507708A/ja active Pending
- 1991-06-21 CA CA002085591A patent/CA2085591A1/en not_active Abandoned
-
1992
- 1992-12-16 FI FI925718A patent/FI101072B/fi active
- 1992-12-18 NO NO924930A patent/NO302298B1/no unknown
-
1996
- 1996-11-28 GR GR960403201T patent/GR3021810T3/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| AU8063391A (en) | 1992-01-23 |
| ZA914530B (en) | 1993-02-24 |
| DK0535104T3 (da) | 1997-01-13 |
| PT98063A (pt) | 1992-03-31 |
| FI101072B (fi) | 1998-04-15 |
| NO924930D0 (no) | 1992-12-18 |
| WO1992000298A1 (en) | 1992-01-09 |
| JPH05507708A (ja) | 1993-11-04 |
| IE911946A1 (en) | 1992-01-01 |
| DK151890D0 (da) | 1990-06-22 |
| PT98063B (pt) | 1998-12-31 |
| EP0535104A1 (en) | 1993-04-07 |
| ATE142209T1 (de) | 1996-09-15 |
| DE69121894T2 (de) | 1997-02-06 |
| AU662293B2 (en) | 1995-08-31 |
| IL98428A0 (en) | 1992-07-15 |
| KR930701442A (ko) | 1993-06-11 |
| NO302298B1 (no) | 1998-02-16 |
| EP0535104B1 (en) | 1996-09-04 |
| ES2092571T3 (es) | 1996-12-01 |
| FI925718A0 (fi) | 1992-12-16 |
| GR3021810T3 (en) | 1997-02-28 |
| FI925718L (fi) | 1992-12-16 |
| DE69121894D1 (de) | 1996-10-10 |
| NZ238638A (en) | 1993-09-27 |
| NO924930L (no) | 1992-12-18 |
| CA2085591A1 (en) | 1991-12-23 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| KB | Patent renewed | ||
| MM9K | Patent not in force due to non-payment of renewal fees |