IN2012DN00602A - - Google Patents
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- Publication number
- IN2012DN00602A IN2012DN00602A IN602DEN2012A IN2012DN00602A IN 2012DN00602 A IN2012DN00602 A IN 2012DN00602A IN 602DEN2012 A IN602DEN2012 A IN 602DEN2012A IN 2012DN00602 A IN2012DN00602 A IN 2012DN00602A
- Authority
- IN
- India
- Prior art keywords
- phenylpiperidin
- exploration
- pharmacologically
- biologically
- oxo
- Prior art date
Links
- LRAPFVNQEPAVQK-UHFFFAOYSA-N O=C1C(NS(=O)=O)CCCN1C1=CC=CC=C1 Chemical class O=C1C(NS(=O)=O)CCCN1C1=CC=CC=C1 LRAPFVNQEPAVQK-UHFFFAOYSA-N 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 208000037765 diseases and disorders Diseases 0.000 abstract 1
- 230000005714 functional activity Effects 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/68—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
- C07D211/72—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D211/74—Oxygen atoms
- C07D211/76—Oxygen atoms attached in position 2 or 6
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ES200901515 | 2009-06-25 | ||
| PCT/IB2010/052856 WO2010150204A1 (en) | 2009-06-25 | 2010-06-23 | N-(2-oxo-1-phenylpiperidin-3-yl) sulfonamides for the identification of biological and pharmacological activity |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| IN2012DN00602A true IN2012DN00602A (de) | 2015-06-12 |
Family
ID=42797604
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IN602DEN2012 IN2012DN00602A (de) | 2009-06-25 | 2010-06-23 |
Country Status (4)
| Country | Link |
|---|---|
| US (1) | US8569507B2 (de) |
| EP (1) | EP2445879A1 (de) |
| IN (1) | IN2012DN00602A (de) |
| WO (1) | WO2010150204A1 (de) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ES2350548B1 (es) | 2009-06-25 | 2011-09-29 | Institut Univ. De Ciència I Tecnologia, S.A. | N-fenil-1-sulfonil-2-pirrolidinacarboxamidas para la identificacion de actividad biologica y farmacologica. |
| IN2012DN00602A (de) | 2009-06-25 | 2015-06-12 | Inst Univ De Ciencia I Technologia S A | |
| ES2352398B1 (es) | 2009-06-25 | 2011-09-29 | Institut Univ. De Ciencia I Tecnologia S.A. | N-fenetilsulfonamidas-n-sustituidas para la identificacion de actividad biologica y farmacologica. |
| ES2354550B1 (es) * | 2009-06-26 | 2011-11-15 | Institut Univ. De Ciència I Tecnologia, S.A. | Biblioteca de n-(1-fenil-2-oxo-3-piperidil)sulfonamidas para el descubrimiento de fármacos. |
| MD3762368T2 (ro) | 2018-03-08 | 2022-07-31 | Incyte Corp | Compuși diol aminopirazină ca inhibitori ai PI3K-Y |
| EP3587416A1 (de) * | 2018-06-29 | 2020-01-01 | Institut Univ. de Ciència i Tecnologia, S.A. | 2-oxopiperidin-3-yl-derivate und verwendung davon |
| US11046658B2 (en) | 2018-07-02 | 2021-06-29 | Incyte Corporation | Aminopyrazine derivatives as PI3K-γ inhibitors |
Family Cites Families (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6939973B1 (en) | 1999-02-09 | 2005-09-06 | The Scripps Research Institute | Glycoluril core molecules for combinatorial libraries |
| US6710058B2 (en) | 2000-11-06 | 2004-03-23 | Bristol-Myers Squibb Pharma Company | Monocyclic or bicyclic carbocycles and heterocycles as factor Xa inhibitors |
| TW200307667A (en) * | 2002-05-06 | 2003-12-16 | Bristol Myers Squibb Co | Sulfonylaminovalerolactams and derivatives thereof as factor Xa inhibitors |
| DE102004059219A1 (de) * | 2004-12-09 | 2006-06-14 | Bayer Healthcare Ag | Pyrazindicarbonsäureamide und ihre Verwendung |
| US7979558B2 (en) | 2008-08-06 | 2011-07-12 | Futurewei Technologies, Inc. | Remote session control |
| ES2350548B1 (es) | 2009-06-25 | 2011-09-29 | Institut Univ. De Ciència I Tecnologia, S.A. | N-fenil-1-sulfonil-2-pirrolidinacarboxamidas para la identificacion de actividad biologica y farmacologica. |
| IN2012DN00602A (de) | 2009-06-25 | 2015-06-12 | Inst Univ De Ciencia I Technologia S A | |
| ES2352398B1 (es) | 2009-06-25 | 2011-09-29 | Institut Univ. De Ciencia I Tecnologia S.A. | N-fenetilsulfonamidas-n-sustituidas para la identificacion de actividad biologica y farmacologica. |
| ES2354550B1 (es) | 2009-06-26 | 2011-11-15 | Institut Univ. De Ciència I Tecnologia, S.A. | Biblioteca de n-(1-fenil-2-oxo-3-piperidil)sulfonamidas para el descubrimiento de fármacos. |
| ES2351323B1 (es) | 2009-06-26 | 2011-10-05 | Institut Univ. De Ciència I Tecnologia, S.A. | Bibliotecas de n-fenil-1-sulfonil-2-pirrolidinacarboxamidas para el descubrimiento de farmacos. |
| US20120122920A1 (en) | 2009-06-26 | 2012-05-17 | Josep Castells Boliart | Libraries of n-substituted-n-phenylethylsulfonamides for drug discovery |
| US20120122710A1 (en) | 2009-07-01 | 2012-05-17 | Josep Castells Boliart | Libraries of n-substituted-n-phenylethylsulfonamides for the identification of biological and pharmacological activity |
| ES2351452B1 (es) | 2009-07-01 | 2011-10-05 | Institut Univ. De Ciència I Tecnologia, S.A. | Bibliotecas de n-fenil-1-sulfonil-2-pirrolidinacarboxamidas para la identificacion de actividad biologica y farmacologica. |
| ES2354551B1 (es) | 2009-07-01 | 2011-11-15 | Institut Univ. De Ciencia I Tecnologia S.A. | Bibliotecas de n-(1-fenil-2-oxo-3-piperidil)sulfonamidas para la identificación de actividad biológica y farmacológica. |
-
2010
- 2010-06-23 IN IN602DEN2012 patent/IN2012DN00602A/en unknown
- 2010-06-23 WO PCT/IB2010/052856 patent/WO2010150204A1/en not_active Ceased
- 2010-06-23 EP EP10731803A patent/EP2445879A1/de not_active Ceased
-
2011
- 2011-12-21 US US13/332,625 patent/US8569507B2/en active Active
Also Published As
| Publication number | Publication date |
|---|---|
| US20120142930A1 (en) | 2012-06-07 |
| US8569507B2 (en) | 2013-10-29 |
| EP2445879A1 (de) | 2012-05-02 |
| WO2010150204A1 (en) | 2010-12-29 |
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