IN2012DN00602A - - Google Patents
Download PDFInfo
- Publication number
- IN2012DN00602A IN2012DN00602A IN602DEN2012A IN2012DN00602A IN 2012DN00602 A IN2012DN00602 A IN 2012DN00602A IN 602DEN2012 A IN602DEN2012 A IN 602DEN2012A IN 2012DN00602 A IN2012DN00602 A IN 2012DN00602A
- Authority
- IN
- India
- Prior art keywords
- phenylpiperidin
- exploration
- pharmacologically
- biologically
- oxo
- Prior art date
Links
- LRAPFVNQEPAVQK-UHFFFAOYSA-N O=C1C(NS(=O)=O)CCCN1C1=CC=CC=C1 Chemical class O=C1C(NS(=O)=O)CCCN1C1=CC=CC=C1 LRAPFVNQEPAVQK-UHFFFAOYSA-N 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 208000037765 diseases and disorders Diseases 0.000 abstract 1
- 230000005714 functional activity Effects 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/68—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
- C07D211/72—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D211/74—Oxygen atoms
- C07D211/76—Oxygen atoms attached in position 2 or 6
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ES200901515 | 2009-06-25 | ||
| PCT/IB2010/052856 WO2010150204A1 (fr) | 2009-06-25 | 2010-06-23 | N-(2-oxo-1-phénylpipéridin-3-yl)sulfonamides pour l'identification d'une activité biologique et pharmacologique |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| IN2012DN00602A true IN2012DN00602A (fr) | 2015-06-12 |
Family
ID=42797604
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IN602DEN2012 IN2012DN00602A (fr) | 2009-06-25 | 2010-06-23 |
Country Status (4)
| Country | Link |
|---|---|
| US (1) | US8569507B2 (fr) |
| EP (1) | EP2445879A1 (fr) |
| IN (1) | IN2012DN00602A (fr) |
| WO (1) | WO2010150204A1 (fr) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ES2352398B1 (es) | 2009-06-25 | 2011-09-29 | Institut Univ. De Ciencia I Tecnologia S.A. | N-fenetilsulfonamidas-n-sustituidas para la identificacion de actividad biologica y farmacologica. |
| ES2350548B1 (es) | 2009-06-25 | 2011-09-29 | Institut Univ. De Ciència I Tecnologia, S.A. | N-fenil-1-sulfonil-2-pirrolidinacarboxamidas para la identificacion de actividad biologica y farmacologica. |
| IN2012DN00602A (fr) | 2009-06-25 | 2015-06-12 | Inst Univ De Ciencia I Technologia S A | |
| ES2354550B1 (es) * | 2009-06-26 | 2011-11-15 | Institut Univ. De Ciència I Tecnologia, S.A. | Biblioteca de n-(1-fenil-2-oxo-3-piperidil)sulfonamidas para el descubrimiento de fármacos. |
| TWI903299B (zh) | 2018-03-08 | 2025-11-01 | 美商英塞特公司 | 作為PI3K-γ抑制劑之胺基吡嗪二醇化合物 |
| EP3587416A1 (fr) * | 2018-06-29 | 2020-01-01 | Institut Univ. de Ciència i Tecnologia, S.A. | Dérivés de 2-oxopiperidin-3-yl et leurs utilisations |
| WO2020010003A1 (fr) | 2018-07-02 | 2020-01-09 | Incyte Corporation | DÉRIVÉS D'AMINOPYRAZINE UTILISÉS EN TANT QU'INHIBITEURS DE PI3K-γ |
Family Cites Families (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6939973B1 (en) | 1999-02-09 | 2005-09-06 | The Scripps Research Institute | Glycoluril core molecules for combinatorial libraries |
| US6710058B2 (en) | 2000-11-06 | 2004-03-23 | Bristol-Myers Squibb Pharma Company | Monocyclic or bicyclic carbocycles and heterocycles as factor Xa inhibitors |
| TW200307667A (en) | 2002-05-06 | 2003-12-16 | Bristol Myers Squibb Co | Sulfonylaminovalerolactams and derivatives thereof as factor Xa inhibitors |
| DE102004059219A1 (de) * | 2004-12-09 | 2006-06-14 | Bayer Healthcare Ag | Pyrazindicarbonsäureamide und ihre Verwendung |
| US7979558B2 (en) | 2008-08-06 | 2011-07-12 | Futurewei Technologies, Inc. | Remote session control |
| ES2352398B1 (es) | 2009-06-25 | 2011-09-29 | Institut Univ. De Ciencia I Tecnologia S.A. | N-fenetilsulfonamidas-n-sustituidas para la identificacion de actividad biologica y farmacologica. |
| ES2350548B1 (es) | 2009-06-25 | 2011-09-29 | Institut Univ. De Ciència I Tecnologia, S.A. | N-fenil-1-sulfonil-2-pirrolidinacarboxamidas para la identificacion de actividad biologica y farmacologica. |
| IN2012DN00602A (fr) | 2009-06-25 | 2015-06-12 | Inst Univ De Ciencia I Technologia S A | |
| US20120122920A1 (en) | 2009-06-26 | 2012-05-17 | Josep Castells Boliart | Libraries of n-substituted-n-phenylethylsulfonamides for drug discovery |
| ES2351323B1 (es) | 2009-06-26 | 2011-10-05 | Institut Univ. De Ciència I Tecnologia, S.A. | Bibliotecas de n-fenil-1-sulfonil-2-pirrolidinacarboxamidas para el descubrimiento de farmacos. |
| ES2354550B1 (es) | 2009-06-26 | 2011-11-15 | Institut Univ. De Ciència I Tecnologia, S.A. | Biblioteca de n-(1-fenil-2-oxo-3-piperidil)sulfonamidas para el descubrimiento de fármacos. |
| US20120122710A1 (en) | 2009-07-01 | 2012-05-17 | Josep Castells Boliart | Libraries of n-substituted-n-phenylethylsulfonamides for the identification of biological and pharmacological activity |
| ES2351452B1 (es) | 2009-07-01 | 2011-10-05 | Institut Univ. De Ciència I Tecnologia, S.A. | Bibliotecas de n-fenil-1-sulfonil-2-pirrolidinacarboxamidas para la identificacion de actividad biologica y farmacologica. |
| ES2354551B1 (es) | 2009-07-01 | 2011-11-15 | Institut Univ. De Ciencia I Tecnologia S.A. | Bibliotecas de n-(1-fenil-2-oxo-3-piperidil)sulfonamidas para la identificación de actividad biológica y farmacológica. |
-
2010
- 2010-06-23 IN IN602DEN2012 patent/IN2012DN00602A/en unknown
- 2010-06-23 WO PCT/IB2010/052856 patent/WO2010150204A1/fr not_active Ceased
- 2010-06-23 EP EP10731803A patent/EP2445879A1/fr not_active Ceased
-
2011
- 2011-12-21 US US13/332,625 patent/US8569507B2/en active Active
Also Published As
| Publication number | Publication date |
|---|---|
| US8569507B2 (en) | 2013-10-29 |
| EP2445879A1 (fr) | 2012-05-02 |
| US20120142930A1 (en) | 2012-06-07 |
| WO2010150204A1 (fr) | 2010-12-29 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| EA200971077A1 (ru) | Гетероциклические модуляторы киназы | |
| IN2012DN00602A (fr) | ||
| EA200970738A1 (ru) | Ингибиторы активности akt | |
| MX2009010517A (es) | Moduladores de cinasa aurora y metodos de uso. | |
| EA200901157A1 (ru) | Конденсированные кольцевые гетероциклические модуляторы киназы | |
| EA201291107A1 (ru) | Соединения, ингибирующие металлоферменты | |
| TW200745109A (en) | Pyrrolo-pyridine kinase modulators | |
| EA201691121A1 (ru) | Гидроксиамидные соединения пиримидина в качестве ингибиторов деацетилаз белков и способы их применения | |
| BR112013027774A2 (pt) | novos compostos como moduladores de proteína quinases | |
| TN2012000081A1 (en) | Compounds and compositions as protein kinase inhibitors | |
| EA200900779A1 (ru) | Производные дигидропиридина, полезные как ингибиторы протеинкиназы | |
| EA200900959A1 (ru) | Ингибиторы мек | |
| MX2009011210A (es) | Inhibidores de mcl1 de indol 7-no sustituido. | |
| BRPI0808775A2 (pt) | compostos e composições como moduladores de atividade de gpr119 | |
| MY156274A (en) | COMPOUNDS FOR THE REDUCTION OF ß-AMYLOID PRODUCTION | |
| WO2008124849A3 (fr) | Modulateurs de pyrrolo-pyridine kinase | |
| EA200970403A1 (ru) | Бициклические триазолы в качестве модуляторов протеинкиназы | |
| BR112012011528A2 (pt) | métodos para inibir uma proteína quinase e para tratar uma doença associada com atividade de quinase, e, composto | |
| BR112012008004A2 (pt) | compostos e composições como moduladores da atividade de gpr119 | |
| MA32349B1 (fr) | Antagonistes de la voie hedgehog a base de phtalazines disubstituees | |
| EA201171063A1 (ru) | Фармацевтические составы олмесартана | |
| UY31760A (es) | Tiazolopiridin-2-iloxi-fenil y tiazolopirazin-2-iloxi-fenil aminas como moduladores de leucotrieno a4 hidrolasa | |
| MX2009007911A (es) | Inhibidores de proteina tirosina fosfatasa 1b aromaticos fusionados. | |
| EA200901042A1 (ru) | Производные 1-бензенсульфонил-1h-индола в качестве ингибиторов активности ccr9 | |
| BRPI0820668A2 (pt) | Derivados de oxindol substituídos por 5-halogênio e seu uso para tratar doenças dependentes de vasopressina |