IN2012DN05125A - - Google Patents

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Publication number
IN2012DN05125A
IN2012DN05125A IN5125DEN2012A IN2012DN05125A IN 2012DN05125 A IN2012DN05125 A IN 2012DN05125A IN 5125DEN2012 A IN5125DEN2012 A IN 5125DEN2012A IN 2012DN05125 A IN2012DN05125 A IN 2012DN05125A
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India
Prior art keywords
sphingosine
modulators
pharmaceuticals
preparing
processes
Prior art date
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English (en)
Inventor
M Heidelbaugh Todd
X Nguyen Phong
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Allergan Inc
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Publication of IN2012DN05125A publication Critical patent/IN2012DN05125A/en

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    • C07D307/34—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D307/38—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms
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CA2865215A1 (fr) 2012-02-21 2013-08-29 Allergan, Inc. Derives de phenoxy-azetidine utilises comme modulateurs des recepteurs de la sphingosine 1-phosphate (s1p)
WO2014093253A1 (fr) * 2012-12-13 2014-06-19 Allergan, Inc. Nouveaux composés thio aromatiques utilisés en tant que modulateurs des récepteurs
SI2958913T1 (sl) 2013-02-20 2018-12-31 Lg Chem, Ltd. Sfingozin-1-fosfat receptor agonisti, postopki za njegovo pripravo in farmacevtski sestavki, ki ga vsebujejo kot aktivno sredstvo
US20140256945A1 (en) * 2013-03-07 2014-09-11 Allergan, Inc. Phosphonic acid compounds as sphingosine-1-phosphate receptor modulators
WO2015021112A1 (fr) * 2013-08-08 2015-02-12 Allergan, Inc. Dérivés aryloxy disubstitués à utiliser en tant que modulateurs des récepteurs de la sphingosine-1-phosphate
US20150045341A1 (en) * 2013-08-08 2015-02-12 Allergan, Inc. Disubstituted aryl azetidine derivatives as sphingosine-1 phosphate receptors modulators
WO2015073547A1 (fr) * 2013-11-13 2015-05-21 Allergan, Inc. Dérivés de phénoxy azétidine disubstitutés utilisés comme modulateurs du récepteur de la sphingosine 1-phosphate (s1p)
KR20200116953A (ko) 2018-02-02 2020-10-13 고쿠리츠 다이가쿠 호진 교토 다이가쿠 안내 혈관 신생 및/또는 안내 혈관 투과성 항진을 수반하는 안과 질환의 예방 또는 치료를 위한 의약
US20240217935A1 (en) * 2021-04-14 2024-07-04 Lg Chem, Ltd. Method for preparing intermediate for synthesis of sphingosine-1-phosphate receptor agonist
KR102802371B1 (ko) * 2021-04-14 2025-05-07 주식회사 엘지화학 스핑고신-1-인산 수용체 효능제의 신규한 제조방법
EP4306516A4 (fr) * 2021-04-14 2024-09-11 Lg Chem, Ltd. Nouveau procédé de préparation d'un agoniste du récepteur de la sphingosine-1-phosphate

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BR112012012259A2 (pt) 2019-09-24
EP2504323A1 (fr) 2012-10-03
ZA201203524B (en) 2013-01-30
JP5939158B2 (ja) 2016-06-22
RU2012122615A (ru) 2013-12-27
AU2010324988A1 (en) 2012-06-07
US8440644B2 (en) 2013-05-14
CA2780908A1 (fr) 2011-06-03
AU2010324988B2 (en) 2016-05-26
KR20120101686A (ko) 2012-09-14
CN102712618A (zh) 2012-10-03
EP2504323B1 (fr) 2017-03-15
KR20120098796A (ko) 2012-09-05
CN102712607B (zh) 2016-06-22
US8703745B1 (en) 2014-04-22
CL2012001352A1 (es) 2012-08-31
IN2012DN05171A (fr) 2015-10-23
AU2010324983A1 (en) 2012-06-07
NZ599966A (en) 2014-09-26
MX2012006022A (es) 2012-08-15
US8653062B2 (en) 2014-02-18
RU2012125184A (ru) 2013-12-27
US20110212925A1 (en) 2011-09-01
CN102712618B (zh) 2014-11-26
JP2013512243A (ja) 2013-04-11
CN102712607A (zh) 2012-10-03
JP2013512244A (ja) 2013-04-11
US20110152241A1 (en) 2011-06-23
IL219758A0 (en) 2012-07-31
MX2012006028A (es) 2012-06-19
US20140107075A1 (en) 2014-04-17
IL219759A0 (en) 2012-07-31
EP2504328A1 (fr) 2012-10-03
CA2780987A1 (fr) 2011-06-03
ZA201203523B (en) 2013-01-31
WO2011066179A1 (fr) 2011-06-03
CA2780987C (fr) 2018-03-06
BR112012012261A2 (pt) 2016-04-26

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