IN2012DN05125A - - Google Patents

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Publication number
IN2012DN05125A
IN2012DN05125A IN5125DEN2012A IN2012DN05125A IN 2012DN05125 A IN2012DN05125 A IN 2012DN05125A IN 5125DEN2012 A IN5125DEN2012 A IN 5125DEN2012A IN 2012DN05125 A IN2012DN05125 A IN 2012DN05125A
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India
Prior art keywords
sphingosine
modulators
pharmaceuticals
preparing
processes
Prior art date
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English (en)
Inventor
M Heidelbaugh Todd
X Nguyen Phong
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Allergan Inc
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Publication of IN2012DN05125A publication Critical patent/IN2012DN05125A/en

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    • C07D307/34—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D307/38—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms
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HUE039931T2 (hu) 2013-02-20 2019-02-28 Lg Chemical Ltd Szfingozin-1-foszfát receptor agonisták, azok elkészítési eljárásai, és azokat aktív ágensként tartalmazó gyógyszerészeti készítmények
US20140256945A1 (en) * 2013-03-07 2014-09-11 Allergan, Inc. Phosphonic acid compounds as sphingosine-1-phosphate receptor modulators
US20150045328A1 (en) * 2013-08-08 2015-02-12 Allergan, Inc. Disubstituted aryl oxy derivatives as sphingosine-1 phosphate receptors modulators
US20150045341A1 (en) * 2013-08-08 2015-02-12 Allergan, Inc. Disubstituted aryl azetidine derivatives as sphingosine-1 phosphate receptors modulators
WO2015073547A1 (en) * 2013-11-13 2015-05-21 Allergan, Inc. Disubstituted phenoxy azetidine derivatives as sphingosine-1-phosphate (s1p) receptor modulators
MX2020007948A (es) 2018-02-02 2020-12-10 Univ Kyoto Medicamento para prevenir o tratar una enfermedad oftalmica asociada con neovascularizacion intraocular mejorada y/o permeabilidad vascular intraocular.
TWI894459B (zh) * 2021-04-14 2025-08-21 南韓商Lg化學股份有限公司 製備用於合成鞘胺醇—1—磷酸酯受體促效劑之中間體的方法
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JP5939158B2 (ja) 2016-06-22
EP2504323A1 (en) 2012-10-03
WO2011066179A1 (en) 2011-06-03
IN2012DN05171A (th) 2015-10-23
ZA201203524B (en) 2013-01-30
JP2013512243A (ja) 2013-04-11
RU2012125184A (ru) 2013-12-27
AU2010324988A1 (en) 2012-06-07
EP2504323B1 (en) 2017-03-15
US20140107075A1 (en) 2014-04-17
US8440644B2 (en) 2013-05-14
CL2012001352A1 (es) 2012-08-31
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IL219759A0 (en) 2012-07-31
CA2780908A1 (en) 2011-06-03
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KR20120098796A (ko) 2012-09-05
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CA2780987C (en) 2018-03-06
US8703745B1 (en) 2014-04-22
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ZA201203523B (en) 2013-01-31
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