IS2916B - P38 kínasatálmar að stofni til úr 5 hluta heteróhring - Google Patents
P38 kínasatálmar að stofni til úr 5 hluta heteróhringInfo
- Publication number
- IS2916B IS2916B IS8255A IS8255A IS2916B IS 2916 B IS2916 B IS 2916B IS 8255 A IS8255 A IS 8255A IS 8255 A IS8255 A IS 8255A IS 2916 B IS2916 B IS 2916B
- Authority
- IS
- Iceland
- Prior art keywords
- kinase
- heterocycle
- parts
- kinase inhibitors
- inhibitors
- Prior art date
Links
- 125000000623 heterocyclic group Chemical group 0.000 title abstract 2
- 229940043355 kinase inhibitor Drugs 0.000 title abstract 2
- 239000003757 phosphotransferase inhibitor Substances 0.000 title abstract 2
- 102000002574 p38 Mitogen-Activated Protein Kinases Human genes 0.000 abstract 4
- RAXXELZNTBOGNW-UHFFFAOYSA-N imidazole Natural products C1=CNC=N1 RAXXELZNTBOGNW-UHFFFAOYSA-N 0.000 abstract 3
- 150000001875 compounds Chemical class 0.000 abstract 2
- 208000027866 inflammatory disease Diseases 0.000 abstract 2
- 102000001253 Protein Kinase Human genes 0.000 abstract 1
- WTKZEGDFNFYCGP-UHFFFAOYSA-N Pyrazole Chemical compound C=1C=NNC=1 WTKZEGDFNFYCGP-UHFFFAOYSA-N 0.000 abstract 1
- 208000037765 diseases and disorders Diseases 0.000 abstract 1
- 239000003112 inhibitor Substances 0.000 abstract 1
- 230000001404 mediated effect Effects 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 230000002265 prevention Effects 0.000 abstract 1
- 108060006633 protein kinase Proteins 0.000 abstract 1
- 208000024891 symptom Diseases 0.000 abstract 1
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- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
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- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/10—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing aromatic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
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Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US48342803P | 2003-06-26 | 2003-06-26 | |
| US49905403P | 2003-08-29 | 2003-08-29 | |
| US56048104P | 2004-04-07 | 2004-04-07 | |
| PCT/US2004/020384 WO2005009973A1 (en) | 2003-06-26 | 2004-06-24 | 5-membered heterocycle-based p38 kinase inhibitors |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| IS8255A IS8255A (is) | 2006-01-23 |
| IS2916B true IS2916B (is) | 2014-12-15 |
Family
ID=34108816
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IS8255A IS2916B (is) | 2003-06-26 | 2006-01-23 | P38 kínasatálmar að stofni til úr 5 hluta heteróhring |
| IS9037A IS2984B (is) | 2003-06-26 | 2014-01-28 | P38 kínasatálmar að stofni til úr 5 hluta heteróhring |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IS9037A IS2984B (is) | 2003-06-26 | 2014-01-28 | P38 kínasatálmar að stofni til úr 5 hluta heteróhring |
Country Status (26)
| Country | Link |
|---|---|
| US (4) | US7863314B2 (is) |
| EP (2) | EP1641764B1 (is) |
| JP (1) | JP4838121B2 (is) |
| KR (1) | KR101120857B1 (is) |
| CN (1) | CN1832928B (is) |
| AT (1) | ATE517872T1 (is) |
| AU (1) | AU2004259662B2 (is) |
| BR (1) | BRPI0411825B8 (is) |
| CA (1) | CA2526455C (is) |
| CY (2) | CY1111985T1 (is) |
| DK (2) | DK2298743T3 (is) |
| EC (2) | ECSP056206A (is) |
| ES (1) | ES2393950T3 (is) |
| HR (2) | HRP20110757T1 (is) |
| IL (1) | IL172182A (is) |
| IS (2) | IS2916B (is) |
| MA (1) | MA27888A1 (is) |
| MX (1) | MXPA05013824A (is) |
| MY (1) | MY158162A (is) |
| NO (1) | NO334947B1 (is) |
| NZ (1) | NZ544230A (is) |
| PL (2) | PL1641764T3 (is) |
| PT (2) | PT2298743E (is) |
| SI (2) | SI1641764T1 (is) |
| TW (2) | TWI452035B (is) |
| WO (1) | WO2005009973A1 (is) |
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| EP1992344A1 (en) | 2007-05-18 | 2008-11-19 | Institut Curie | P38 alpha as a therapeutic target in pathologies linked to FGFR3 mutation |
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-
2004
- 2004-06-24 HR HR20110757T patent/HRP20110757T1/hr unknown
- 2004-06-24 SI SI200431766T patent/SI1641764T1/sl unknown
- 2004-06-24 PT PT101643674T patent/PT2298743E/pt unknown
- 2004-06-24 AT AT04777075T patent/ATE517872T1/de active
- 2004-06-24 WO PCT/US2004/020384 patent/WO2005009973A1/en not_active Ceased
- 2004-06-24 EP EP04777075A patent/EP1641764B1/en not_active Expired - Lifetime
- 2004-06-24 PL PL04777075T patent/PL1641764T3/pl unknown
- 2004-06-24 BR BRPI0411825A patent/BRPI0411825B8/pt not_active IP Right Cessation
- 2004-06-24 ES ES10164367T patent/ES2393950T3/es not_active Expired - Lifetime
- 2004-06-24 MX MXPA05013824A patent/MXPA05013824A/es active IP Right Grant
- 2004-06-24 TW TW093118259A patent/TWI452035B/zh not_active IP Right Cessation
- 2004-06-24 JP JP2006517650A patent/JP4838121B2/ja not_active Expired - Lifetime
- 2004-06-24 EP EP10164367A patent/EP2298743B1/en not_active Expired - Lifetime
- 2004-06-24 CA CA2526455A patent/CA2526455C/en not_active Expired - Lifetime
- 2004-06-24 SI SI200431950T patent/SI2298743T1/sl unknown
- 2004-06-24 NZ NZ544230A patent/NZ544230A/en not_active IP Right Cessation
- 2004-06-24 DK DK10164367.4T patent/DK2298743T3/da active
- 2004-06-24 KR KR1020057024679A patent/KR101120857B1/ko not_active Expired - Lifetime
- 2004-06-24 TW TW100114024A patent/TWI449696B/zh not_active IP Right Cessation
- 2004-06-24 AU AU2004259662A patent/AU2004259662B2/en not_active Expired
- 2004-06-24 PL PL10164367T patent/PL2298743T3/pl unknown
- 2004-06-24 DK DK04777075.5T patent/DK1641764T3/da active
- 2004-06-24 CN CN2004800180564A patent/CN1832928B/zh not_active Expired - Lifetime
- 2004-06-24 PT PT04777075T patent/PT1641764E/pt unknown
- 2004-06-25 MY MYPI20042496A patent/MY158162A/en unknown
- 2004-06-25 US US10/877,534 patent/US7863314B2/en not_active Expired - Lifetime
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2005
- 2005-11-24 IL IL172182A patent/IL172182A/en active IP Right Grant
- 2005-12-08 EC EC2005006206A patent/ECSP056206A/es unknown
- 2005-12-21 MA MA28678A patent/MA27888A1/fr unknown
-
2006
- 2006-01-23 IS IS8255A patent/IS2916B/is unknown
- 2006-01-26 NO NO20060424A patent/NO334947B1/no unknown
-
2010
- 2010-11-19 US US12/950,649 patent/US8242117B2/en not_active Expired - Lifetime
-
2011
- 2011-10-27 CY CY20111101022T patent/CY1111985T1/el unknown
-
2012
- 2012-02-07 EC ECSP12006206 patent/ECSP12006206A/es unknown
- 2012-06-22 US US13/530,919 patent/US8410160B2/en not_active Expired - Fee Related
- 2012-11-08 CY CY20121101064T patent/CY1113313T1/el unknown
- 2012-11-08 HR HRP20120900TT patent/HRP20120900T1/hr unknown
-
2013
- 2013-02-25 US US13/775,963 patent/US8580838B2/en not_active Expired - Fee Related
-
2014
- 2014-01-28 IS IS9037A patent/IS2984B/is unknown
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