IS6524A - 5-alkýlpyrídó(3-3-D)pyrimídín týrósín kínasa tálmar - Google Patents

5-alkýlpyrídó(3-3-D)pyrimídín týrósín kínasa tálmar

Info

Publication number
IS6524A
IS6524A IS6524A IS6524A IS6524A IS 6524 A IS6524 A IS 6524A IS 6524 A IS6524 A IS 6524A IS 6524 A IS6524 A IS 6524A IS 6524 A IS6524 A IS 6524A
Authority
IS
Iceland
Prior art keywords
alkylpyrido
tyrosine kinase
kinase inhibitors
pyrimidine
pyrimidine tyrosine
Prior art date
Application number
IS6524A
Other languages
English (en)
Icelandic (is)
Inventor
John Booth Richard
Myra Dobrusin Ellen
Laurence Toogood Peter
Norman Vanderwel Scott
Original Assignee
Warner-Lambert Company
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Warner-Lambert Company filed Critical Warner-Lambert Company
Publication of IS6524A publication Critical patent/IS6524A/is

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/06Antipsoriatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A61P29/02Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID] without antiinflammatory effect
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Dermatology (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
IS6524A 2000-03-06 2002-08-23 5-alkýlpyrídó(3-3-D)pyrimídín týrósín kínasa tálmar IS6524A (is)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US18712400P 2000-03-06 2000-03-06
PCT/US2001/002657 WO2001070741A1 (en) 2000-03-06 2001-01-29 5-alkylpyrido[2,3-d]pyrimidines tyrosine kinase inhibitors

Publications (1)

Publication Number Publication Date
IS6524A true IS6524A (is) 2002-08-23

Family

ID=22687699

Family Applications (1)

Application Number Title Priority Date Filing Date
IS6524A IS6524A (is) 2000-03-06 2002-08-23 5-alkýlpyrídó(3-3-D)pyrimídín týrósín kínasa tálmar

Country Status (37)

Country Link
EP (1) EP1268476A1 (es)
JP (1) JP2003528101A (es)
KR (1) KR20020075805A (es)
CN (1) CN1422268A (es)
AP (1) AP2002002643A0 (es)
AR (1) AR034119A1 (es)
AU (1) AU2001233028A1 (es)
BG (1) BG107161A (es)
BR (1) BR0109056A (es)
CA (1) CA2401368A1 (es)
CO (1) CO5280200A1 (es)
CR (1) CR6736A (es)
CZ (1) CZ20022929A3 (es)
DZ (1) DZ3308A1 (es)
EA (1) EA200200802A1 (es)
EE (1) EE200200506A (es)
GT (1) GT200100037A (es)
HN (1) HN2001000040A (es)
HR (1) HRP20020798A2 (es)
HU (1) HUP0300136A2 (es)
IL (1) IL151480A0 (es)
IS (1) IS6524A (es)
MA (1) MA26881A1 (es)
MX (1) MXPA02008535A (es)
NO (1) NO20024235L (es)
NZ (1) NZ520962A (es)
OA (1) OA12227A (es)
PA (1) PA8513201A1 (es)
PE (1) PE20011177A1 (es)
PL (1) PL358271A1 (es)
PY (1) PY0104899A (es)
SK (1) SK12472002A3 (es)
SV (1) SV2001000338A (es)
TN (1) TNSN01036A1 (es)
WO (1) WO2001070741A1 (es)
YU (1) YU66502A (es)
ZA (1) ZA200207110B (es)

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US7235551B2 (en) 2000-03-02 2007-06-26 Smithkline Beecham Corporation 1,5-disubstituted-3,4-dihydro-1h-pyrimido[4,5-d]pyrimidin-2-one compounds and their use in treating csbp/p38 kinase mediated diseases
JP4524072B2 (ja) 2000-10-23 2010-08-11 グラクソスミスクライン・リミテッド・ライアビリティ・カンパニー 新規化合物
CZ20032416A3 (cs) * 2001-02-12 2004-07-14 F. Hoffmann-La Roche Ag 6-Substituované pyridopyrimidiny
JP4166991B2 (ja) * 2001-02-26 2008-10-15 田辺三菱製薬株式会社 ピリドピリミジンまたはナフチリジン誘導体
AU2002324450A1 (en) * 2001-06-21 2003-01-08 Ariad Pharmaceuticals, Inc. Novel pyridopyrimidines and uses thereof
US20030100572A1 (en) * 2001-06-21 2003-05-29 Ariad Pharmaceuticals,Inc. Novel pyridopyrimidones and uses thereof
DE60303009T2 (de) 2002-01-22 2006-07-13 Warner-Lambert Co. Llc 2-(pyridin-2-ylamino)-pyrido[2,3-d]pyrimidin-7-one
MXPA04010267A (es) 2002-04-19 2005-02-03 Smithkline Beecham Corp Compuestos novedosos.
EP1542989B1 (en) 2002-07-31 2007-04-18 Critical Outcome Technologies, Inc. Protein tyrosine kinase inhibitors
AU2003273675A1 (en) 2002-10-09 2004-05-04 Wayne R. Danter Protein tyrosine kinase inhibitors
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DE102004029784A1 (de) 2004-06-21 2006-01-05 Boehringer Ingelheim Pharma Gmbh & Co. Kg Neue 2-Benzylaminodihydropteridinone, Verfahren zur deren Herstellung und deren Verwendung als Arzneimittel
DE102004033670A1 (de) 2004-07-09 2006-02-02 Boehringer Ingelheim Pharma Gmbh & Co. Kg Neue Pyridodihydropyrazinone, Verfahren zu Ihrer Herstellung und Ihre Verwendung als Arzneimittel
FR2873118B1 (fr) 2004-07-15 2007-11-23 Sanofi Synthelabo Derives de pyrido-pyrimidine, leur application en therapeutique
US20060035903A1 (en) 2004-08-14 2006-02-16 Boehringer Ingelheim International Gmbh Storage stable perfusion solution for dihydropteridinones
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US7759485B2 (en) 2004-08-14 2010-07-20 Boehringer Ingelheim International Gmbh Process for the manufacture of dihydropteridinones
US7728134B2 (en) 2004-08-14 2010-06-01 Boehringer Ingelheim International Gmbh Hydrates and polymorphs of 4[[(7R)-8-cyclopentyl-7-ethyl-5,6,7,8-tetrahydro-5-methyl-6-oxo-2-pteridinyl]amino]-3-methoxy-N-(1-methyl-4-piperidinyl)-benzamide, process for their manufacture and their use as medicament
US20060074088A1 (en) 2004-08-14 2006-04-06 Boehringer Ingelheim International Gmbh Dihydropteridinones for the treatment of cancer diseases
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US20080114007A1 (en) * 2006-10-31 2008-05-15 Player Mark R 5-oxo-5,8-dihydro-pyrido-pyrimidines as inhibitors of c-fms kinase
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WO2008124323A1 (en) * 2007-04-03 2008-10-16 Array Biopharma Inc. Imidazo[1,2-a]pyridine compounds as receptor tyrosine kinase inhibitors
CN101784551A (zh) * 2007-06-15 2010-07-21 万有制药株式会社 二环苯胺衍生物
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WO2020114519A1 (zh) * 2018-12-07 2020-06-11 杭州英创医药科技有限公司 作为cdk-hdac双通路抑制剂的杂环化合物
CN112759589B (zh) * 2019-11-01 2022-04-08 暨南大学 嘧啶并吡啶酮类化合物及其应用
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JP7756374B2 (ja) * 2021-03-08 2025-10-20 曁南大学 ピリドピリミジン系化合物及びその使用
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CN117720531A (zh) * 2022-09-16 2024-03-19 华东师范大学 作为rsk抑制剂的吡啶酮并嘧啶衍生物及其应用
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US5620981A (en) * 1995-05-03 1997-04-15 Warner-Lambert Company Pyrido [2,3-D]pyrimidines for inhibiting protein tyrosine kinase mediated cellular proliferation
DE69839338T2 (de) * 1997-02-05 2008-07-10 Warner-Lambert Company Llc Pyrido (2,3-d) pyrimidine und 4-amino-pyrimidine als inhibitoren der zellulären proliferation
EE200000706A (et) * 1998-05-26 2002-06-17 Warner-Lambert Company Bitsüklilised pürimidiinid ja bitsüklilised 3,4-dihüdropürimidiinid kui rakkude proliferatsiooni inhibiitorid

Also Published As

Publication number Publication date
PY0104899A (es) 2003-11-03
CZ20022929A3 (cs) 2003-02-12
AU2001233028A1 (en) 2001-10-03
NO20024235D0 (no) 2002-09-05
MXPA02008535A (es) 2002-12-13
NZ520962A (en) 2003-09-26
NO20024235L (no) 2002-11-05
OA12227A (en) 2004-03-18
YU66502A (sh) 2005-09-19
EE200200506A (et) 2004-02-16
HN2001000040A (es) 2001-09-06
EA200200802A1 (ru) 2003-02-27
CA2401368A1 (en) 2001-09-27
BR0109056A (pt) 2003-06-03
ZA200207110B (en) 2003-12-04
TNSN01036A1 (en) 2005-11-10
CN1422268A (zh) 2003-06-04
IL151480A0 (en) 2003-04-10
CR6736A (es) 2004-03-10
PE20011177A1 (es) 2001-11-23
HUP0300136A2 (en) 2003-05-28
MA26881A1 (fr) 2004-12-20
JP2003528101A (ja) 2003-09-24
BG107161A (bg) 2003-06-30
EP1268476A1 (en) 2003-01-02
SK12472002A3 (sk) 2003-04-01
SV2001000338A (es) 2001-11-30
KR20020075805A (ko) 2002-10-05
GT200100037A (es) 2002-03-04
DZ3308A1 (fr) 2001-09-27
HRP20020798A2 (en) 2004-02-29
WO2001070741A1 (en) 2001-09-27
CO5280200A1 (es) 2003-05-30
PL358271A1 (pl) 2004-08-09
AP2002002643A0 (en) 2002-12-31
PA8513201A1 (es) 2003-06-30
AR034119A1 (es) 2004-02-04

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