IS6732A - Bísýklísk heteróarómatísk efnasambönd - Google Patents

Bísýklísk heteróarómatísk efnasambönd

Info

Publication number: IS6732A
Authority: IS; Iceland
Prior art keywords: heteroaromatic compounds; bicyclic heteroaromatic; bicyclic; compounds; heteroaromatic
Prior art date: 2000-09-22

Application number

IS6732A

Other languages

English (en)

Other versions

IS2531B (is

Inventor

Marius Timmers Cornelis

Frederik Johan Karstens Willem

Original Assignee

Akzo Nobel N.V.

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-09-22

Filing date

2003-02-28

Publication date

2003-02-28

2003-02-28 Application filed by Akzo Nobel N.V. filed Critical Akzo Nobel N.V.

2003-02-28 Publication of IS6732A publication Critical patent/IS6732A/is

2009-07-15 Publication of IS2531B publication Critical patent/IS2531B/is

Links

-1 Bicyclic heteroaromatic compounds Chemical class 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/06—Drugs for disorders of the endocrine system of the anterior pituitary hormones, e.g. TSH, ACTH, FSH, LH, PRL, GH
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
- C07D239/72—Quinazolines; Hydrogenated quinazolines
- C07D239/78—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 2
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Bioinformatics & Cheminformatics (AREA)
Pharmacology & Pharmacy (AREA)
Engineering & Computer Science (AREA)
Animal Behavior & Ethology (AREA)
Chemical Kinetics & Catalysis (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Endocrinology (AREA)
Diabetes (AREA)
Reproductive Health (AREA)
Gynecology & Obstetrics (AREA)
Pregnancy & Childbirth (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)

IS6732A 2000-09-22 2003-02-28 Bísýklísk heteróarómatísk efnasambönd IS2531B (is)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
EP00203287		2000-09-22
PCT/EP2001/010743 WO2002024703A1 (en)	2000-09-22	2001-09-17	Bicyclic heteroaromatic compounds

Publications (2)

Publication Number	Publication Date
IS6732A true IS6732A (is)	2003-02-28
IS2531B IS2531B (is)	2009-07-15

Family

ID=8172046

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
IS6732A IS2531B (is)	2000-09-22	2003-02-28	Bísýklísk heteróarómatísk efnasambönd

Country Status (31)

Country	Link
US (2)	US7229990B2 (is)
EP (2)	EP1322651B1 (is)
JP (1)	JP4977940B2 (is)
KR (1)	KR100860040B1 (is)
CN (1)	CN1247594C (is)
AR (1)	AR030784A1 (is)
AT (1)	ATE384726T1 (is)
AU (2)	AU2002213929B2 (is)
BR (1)	BR0113987A (is)
CA (1)	CA2422054C (is)
CY (1)	CY1107308T1 (is)
CZ (1)	CZ297136B6 (is)
DE (1)	DE60132607T2 (is)
DK (1)	DK1322651T3 (is)
EC (1)	ECSP034523A (is)
ES (1)	ES2299524T3 (is)
HR (1)	HRP20030220B1 (is)
HU (1)	HU229422B1 (is)
IL (2)	IL154624A0 (is)
IS (1)	IS2531B (is)
MX (1)	MXPA03002478A (is)
NO (1)	NO328683B1 (is)
NZ (1)	NZ524444A (is)
PE (1)	PE20020537A1 (is)
PL (1)	PL207755B1 (is)
PT (1)	PT1322651E (is)
RU (1)	RU2271360C2 (is)
SK (1)	SK287554B6 (is)
TW (1)	TWI290143B (is)
WO (1)	WO2002024703A1 (is)
ZA (1)	ZA200301588B (is)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
EP1322651B1 (en) *	2000-09-22	2008-01-23	N.V. Organon	Bicyclic heteroaromatic compounds
TW200407127A (en)	2002-08-21	2004-05-16	Astrazeneca Ab	Chemical compounds
US7674822B2 (en)	2004-11-24	2010-03-09	Wyeth	PTP1b inhibitors
US7737155B2 (en) *	2005-05-17	2010-06-15	Schering Corporation	Nitrogen-containing heterocyclic compounds and methods of use thereof
JP4975739B2 (ja) *	2005-05-17	2012-07-11	シェーリングコーポレイション	脂質異常症の処置のための、ニコチン酸受容体アゴニストとしての複素環
AU2007254165A1 (en) *	2006-05-17	2007-11-29	Forschungsverbund Berlin E.V.	Pyrimidine low molecular weight ligands for modulating hormone receptors
CN102015704A (zh)	2008-04-29	2011-04-13	霍夫曼-拉罗奇有限公司	Jnk的嘧啶基吡啶酮抑制剂
EP2358684B8 (en)	2008-10-20	2014-10-22	The Government of the United States of America as represented by the Secretary of the Department of Health and Human Services	Low molecular weight thyroid stimulating hormone receptor (tshr) agonists
CN102791705B (zh)	2010-04-08	2016-08-03	美国政府(由卫生和人类服务部的部长所代表)	用于tsh受体的反向激动剂和中性拮抗剂
DK3392252T3 (da) *	2011-08-23	2024-01-08	Libertas Bio Inc	Pyrimido-pyridazinonforbindelser og deres anvendelse
CN113680386B (zh) *	2021-08-23	2023-08-11	深圳湾实验室坪山生物医药研发转化中心	氮杂环卡宾-方酰胺双功能催化剂及其制备方法

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
RU2127736C1 (ru) *	1992-06-22	1999-03-20	Берингер Ингельгейм КГ	Производные анеллированного дигидропиридина или их соли с физиологически переносимыми кислотами и средство, блокирующее неселективные катионные каналы
TW276256B (is) *	1993-08-26	1996-05-21	Takeda Pharm Industry Co Ltd
NZ284846A (en) *	1994-06-16	1998-12-23	Pfizer	1-substituted-pyrazolo[3,4-b]pyridin-5-carboxylic acid derivatives, preparation, use, intermediates and pharmaceutical compositions thereof
AU712019B2 (en) *	1996-05-20	1999-10-28	Merck & Co., Inc.	Antagonists of gonadotropin releasing hormone
TW564247B (en) *	1999-04-08	2003-12-01	Akzo Nobel Nv	Bicyclic heteraromatic compound
EP1322651B1 (en) *	2000-09-22	2008-01-23	N.V. Organon	Bicyclic heteroaromatic compounds

2001
- 2001-09-17 EP EP01982306A patent/EP1322651B1/en not_active Expired - Lifetime
- 2001-09-17 PL PL360675A patent/PL207755B1/pl unknown
- 2001-09-17 ES ES01982306T patent/ES2299524T3/es not_active Expired - Lifetime
- 2001-09-17 CA CA2422054A patent/CA2422054C/en not_active Expired - Fee Related
- 2001-09-17 RU RU2003111463/04A patent/RU2271360C2/ru not_active IP Right Cessation
- 2001-09-17 DE DE60132607T patent/DE60132607T2/de not_active Expired - Lifetime
- 2001-09-17 AU AU2002213929A patent/AU2002213929B2/en not_active Ceased
- 2001-09-17 CZ CZ20030828A patent/CZ297136B6/cs not_active IP Right Cessation
- 2001-09-17 AT AT01982306T patent/ATE384726T1/de active
- 2001-09-17 CN CNB018160670A patent/CN1247594C/zh not_active Expired - Fee Related
- 2001-09-17 IL IL15462401A patent/IL154624A0/xx unknown
- 2001-09-17 KR KR1020037004132A patent/KR100860040B1/ko not_active Expired - Fee Related
- 2001-09-17 NZ NZ524444A patent/NZ524444A/en not_active IP Right Cessation
- 2001-09-17 DK DK01982306T patent/DK1322651T3/da active
- 2001-09-17 HU HU0302648A patent/HU229422B1/hu not_active IP Right Cessation
- 2001-09-17 PT PT01982306T patent/PT1322651E/pt unknown
- 2001-09-17 BR BR0113987-8A patent/BR0113987A/pt not_active IP Right Cessation
- 2001-09-17 HR HR20030220A patent/HRP20030220B1/xx not_active IP Right Cessation
- 2001-09-17 US US10/381,248 patent/US7229990B2/en not_active Expired - Lifetime
- 2001-09-17 WO PCT/EP2001/010743 patent/WO2002024703A1/en not_active Ceased
- 2001-09-17 AU AU1392902A patent/AU1392902A/xx active Pending
- 2001-09-17 SK SK331-2003A patent/SK287554B6/sk not_active IP Right Cessation
- 2001-09-17 JP JP2002529113A patent/JP4977940B2/ja not_active Expired - Fee Related
- 2001-09-17 EP EP07113490A patent/EP1886999A3/en not_active Withdrawn
- 2001-09-17 MX MXPA03002478A patent/MXPA03002478A/es active IP Right Grant
- 2001-09-19 TW TW090123098A patent/TWI290143B/zh not_active IP Right Cessation
- 2001-09-21 PE PE2001000954A patent/PE20020537A1/es not_active Application Discontinuation
- 2001-09-21 AR ARP010104458A patent/AR030784A1/es active IP Right Grant
2003
- 2003-02-26 IL IL154624A patent/IL154624A/en not_active IP Right Cessation
- 2003-02-26 ZA ZA200301588A patent/ZA200301588B/en unknown
- 2003-02-28 IS IS6732A patent/IS2531B/is unknown
- 2003-03-21 EC EC2003004523A patent/ECSP034523A/es unknown
- 2003-03-21 NO NO20031314A patent/NO328683B1/no not_active IP Right Cessation
2007
- 2007-04-23 US US11/788,886 patent/US7618963B2/en not_active Expired - Lifetime
2008
- 2008-03-18 CY CY20081100301T patent/CY1107308T1/el unknown

Also Published As

Publication number	Publication date
HU229422B1 (hu)	2013-12-30
HRP20030220A2 (en)	2003-06-30
DE60132607T2 (de)	2009-01-29
NO20031314D0 (no)	2003-03-21
HRP20030220B1 (en)	2011-10-31
ATE384726T1 (de)	2008-02-15
HUP0302648A2 (hu)	2003-11-28
JP4977940B2 (ja)	2012-07-18
AU2002213929B2 (en)	2006-04-13
US7229990B2 (en)	2007-06-12
IL154624A (en)	2009-09-01
CZ2003828A3 (cs)	2003-08-13
CZ297136B6 (cs)	2006-09-13
WO2002024703A1 (en)	2002-03-28
KR100860040B1 (ko)	2008-09-25
HUP0302648A3 (en)	2004-11-29
CA2422054C (en)	2011-01-11
PT1322651E (pt)	2008-02-28
HK1054942A1 (en)	2003-12-19
US20030225113A1 (en)	2003-12-04
MXPA03002478A (es)	2004-05-05
AU1392902A (en)	2002-04-02
EP1886999A2 (en)	2008-02-13
CN1247594C (zh)	2006-03-29
EP1322651B1 (en)	2008-01-23
ECSP034523A (es)	2003-04-25
JP2004509896A (ja)	2004-04-02
PL360675A1 (en)	2004-09-20
CN1462273A (zh)	2003-12-17
NZ524444A (en)	2004-03-26
RU2271360C2 (ru)	2006-03-10
EP1886999A8 (en)	2010-08-04
CA2422054A1 (en)	2002-03-28
US7618963B2 (en)	2009-11-17
KR20030040483A (ko)	2003-05-22
PE20020537A1 (es)	2002-06-20
ZA200301588B (en)	2004-06-22
IL154624A0 (en)	2003-09-17
TWI290143B (en)	2007-11-21
CY1107308T1 (el)	2012-11-21
EP1886999A3 (en)	2008-03-12
BR0113987A (pt)	2003-08-12
DK1322651T3 (da)	2008-06-02
AR030784A1 (es)	2003-09-03
NO328683B1 (no)	2010-04-26
ES2299524T3 (es)	2008-06-01
IS2531B (is)	2009-07-15
PL207755B1 (pl)	2011-01-31
SK3312003A3 (en)	2003-08-05
SK287554B6 (sk)	2011-01-04
EP1322651A1 (en)	2003-07-02
US20070197527A1 (en)	2007-08-23
DE60132607D1 (de)	2008-03-13
NO20031314L (no)	2003-03-21

Publication	Publication Date	Title
CY2015035I2 (el)	2016-04-13	Ενωσεις πυριμιδινης
NO20026196L (no)	2003-02-24	Kinazolinditosylatsalt-forbindelser
NO20024127L (no)	2002-08-29	Pyrimidin-forbindelser
DK1619192T3 (da)	2010-03-29	Arylkondeserede azapolycykliske forbindelser
AR027983A1 (es)	2003-04-23	Novedosos compuestos
IS2531B (is)	2009-07-15	Bísýklísk heteróarómatísk efnasambönd
IS6657A (is)	2002-12-17	Ný efnasambönd
ATE372338T1 (de)	2007-09-15	Deshalogenverbindungen
AR028220A1 (es)	2003-04-30	Novedosos compuestos
NO20030303L (no)	2003-03-20	Kalsilytiske forbindelser
NO20031837L (no)	2003-06-20	Kalsilytiske forbindelser
NO20023508L (no)	2002-07-23	Kalsilyttiske forbindelser
ATE360010T1 (de)	2007-05-15	Heterocyclische retioidverbindungen
SE0003477D0 (sv)	2000-09-28	Compounds
SE0004611D0 (sv)	2000-12-13	Novel Compounds
SE0002234D0 (sv)	2000-06-14	Novel compounds
SE0003979D0 (sv)	2000-10-31	Novel Compounds
SE0004824D0 (sv)	2000-12-22	Novel compounds
SE0003437D0 (sv)	2000-09-26	Novel compounds
SE0003436D0 (sv)	2000-09-26	Novel compounds
SE0003203D0 (sv)	2000-09-08	Novel compounds
SE0003641D0 (sv)	2000-10-09	Novel compounds
SE0000620D0 (sv)	2000-02-25	Novel compounds
SE0002331D0 (sv)	2000-06-20	Novel compounds
FI20050832L (fi)	2005-08-17	Uudet yhdisteet