IS7891A - Skiptitengd þrísýklísk gamma-karbólín sem serótónín viðtaka gerandefni og mótverkunarefni - Google Patents

Skiptitengd þrísýklísk gamma-karbólín sem serótónín viðtaka gerandefni og mótverkunarefni

Info

Publication number
IS7891A
IS7891A IS7891A IS7891A IS7891A IS 7891 A IS7891 A IS 7891A IS 7891 A IS7891 A IS 7891A IS 7891 A IS7891 A IS 7891A IS 7891 A IS7891 A IS 7891A
Authority
IS
Iceland
Prior art keywords
sup
antagonists
receptor agonists
serotonin receptor
novel compounds
Prior art date
Application number
IS7891A
Other languages
English (en)
Inventor
Lee Taekyu
Chen Wenting
Deng Wei
Robichaud Albert
Wexler Ruth
Original Assignee
Bristol-Myers Squibb Company
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol-Myers Squibb Company filed Critical Bristol-Myers Squibb Company
Publication of IS7891A publication Critical patent/IS7891A/is

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Obesity (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Child & Adolescent Psychology (AREA)
  • Cardiology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
IS7891A 2002-12-19 2005-06-10 Skiptitengd þrísýklísk gamma-karbólín sem serótónín viðtaka gerandefni og mótverkunarefni IS7891A (is)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US43476002P 2002-12-19 2002-12-19
PCT/US2003/041447 WO2004056324A2 (en) 2002-12-19 2003-12-19 Substituted tricyclic gamma-carbolines as serotonin receptor agonists and antagonists

Publications (1)

Publication Number Publication Date
IS7891A true IS7891A (is) 2005-06-10

Family

ID=32682101

Family Applications (1)

Application Number Title Priority Date Filing Date
IS7891A IS7891A (is) 2002-12-19 2005-06-10 Skiptitengd þrísýklísk gamma-karbólín sem serótónín viðtaka gerandefni og mótverkunarefni

Country Status (10)

Country Link
US (1) US7109339B2 (is)
EP (1) EP1581221B1 (is)
JP (1) JP4486505B2 (is)
AT (1) ATE509929T1 (is)
AU (1) AU2003303210A1 (is)
ES (1) ES2364046T3 (is)
IS (1) IS7891A (is)
NO (1) NO20052728L (is)
PL (1) PL377426A1 (is)
WO (1) WO2004056324A2 (is)

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Also Published As

Publication number Publication date
WO2004056324A3 (en) 2004-09-02
JP2006511568A (ja) 2006-04-06
ES2364046T3 (es) 2011-08-23
JP4486505B2 (ja) 2010-06-23
EP1581221A2 (en) 2005-10-05
AU2003303210A1 (en) 2004-07-14
NO20052728L (no) 2005-08-23
WO2004056324A2 (en) 2004-07-08
ATE509929T1 (de) 2011-06-15
NO20052728D0 (no) 2005-06-07
EP1581221A4 (en) 2008-11-26
PL377426A1 (pl) 2006-02-06
US20040180875A1 (en) 2004-09-16
AU2003303210A8 (en) 2004-07-14
US7109339B2 (en) 2006-09-19
EP1581221B1 (en) 2011-05-18

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