IS7891A - Skiptitengd þrísýklísk gamma-karbólín sem serótónín viðtaka gerandefni og mótverkunarefni - Google Patents

Skiptitengd þrísýklísk gamma-karbólín sem serótónín viðtaka gerandefni og mótverkunarefni

Info

Publication number: IS7891A
Authority: IS; Iceland
Prior art keywords: sup; antagonists; receptor agonists; serotonin receptor; novel compounds
Prior art date: 2002-12-19

Application number

IS7891A

Other languages

English (en)

Inventor

Lee Taekyu

Chen Wenting

Deng Wei

Robichaud Albert

Wexler Ruth

Original Assignee

Bristol-Myers Squibb Company

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2002-12-19

Filing date

2005-06-10

Publication date

2005-06-10

2005-06-10 Application filed by Bristol-Myers Squibb Company filed Critical Bristol-Myers Squibb Company

2005-06-10 Publication of IS7891A publication Critical patent/IS7891A/is

Links

RDMFHRSPDKWERA-UHFFFAOYSA-N 5H-Pyrido[4,3-b]indole Chemical compound C1=NC=C2C3=CC=CC=C3NC2=C1 RDMFHRSPDKWERA-UHFFFAOYSA-N 0.000 title 1
239000003420 antiserotonin agent Substances 0.000 title 1
239000000952 serotonin receptor agonist Substances 0.000 title 1
150000001875 compounds Chemical class 0.000 abstract 4
208000015114 central nervous system disease Diseases 0.000 abstract 2
102000040125 5-hydroxytryptamine receptor family Human genes 0.000 abstract 1
108091032151 5-hydroxytryptamine receptor family Proteins 0.000 abstract 1
208000019901 Anxiety disease Diseases 0.000 abstract 1
208000019695 Migraine disease Diseases 0.000 abstract 1
208000008589 Obesity Diseases 0.000 abstract 1
208000021384 Obsessive-Compulsive disease Diseases 0.000 abstract 1
208000028017 Psychotic disease Diseases 0.000 abstract 1
239000004480 active ingredient Substances 0.000 abstract 1
208000022531 anorexia Diseases 0.000 abstract 1
230000036506 anxiety Effects 0.000 abstract 1
206010061428 decreased appetite Diseases 0.000 abstract 1
238000009472 formulation Methods 0.000 abstract 1
206010027599 migraine Diseases 0.000 abstract 1
239000000203 mixture Substances 0.000 abstract 1
235000020824 obesity Nutrition 0.000 abstract 1
239000008194 pharmaceutical composition Substances 0.000 abstract 1
230000002265 prevention Effects 0.000 abstract 1
239000000018 receptor agonist Substances 0.000 abstract 1
229940044601 receptor agonist Drugs 0.000 abstract 1
239000002464 receptor antagonist Substances 0.000 abstract 1
229940044551 receptor antagonist Drugs 0.000 abstract 1
150000003839 salts Chemical class 0.000 abstract 1
201000000980 schizophrenia Diseases 0.000 abstract 1
208000012201 sexual and gender identity disease Diseases 0.000 abstract 1
208000015891 sexual disease Diseases 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Veterinary Medicine (AREA)
Life Sciences & Earth Sciences (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Bioinformatics & Cheminformatics (AREA)
Pharmacology & Pharmacy (AREA)
Chemical Kinetics & Catalysis (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Engineering & Computer Science (AREA)
Obesity (AREA)
Diabetes (AREA)
Hematology (AREA)
Heart & Thoracic Surgery (AREA)
Child & Adolescent Psychology (AREA)
Cardiology (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Endocrinology (AREA)
Reproductive Health (AREA)
Dermatology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)

IS7891A 2002-12-19 2005-06-10 Skiptitengd þrísýklísk gamma-karbólín sem serótónín viðtaka gerandefni og mótverkunarefni IS7891A (is)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US43476002P	2002-12-19	2002-12-19
PCT/US2003/041447 WO2004056324A2 (en)	2002-12-19	2003-12-19	Substituted tricyclic gamma-carbolines as serotonin receptor agonists and antagonists

Publications (1)

Publication Number	Publication Date
IS7891A true IS7891A (is)	2005-06-10

Family

ID=32682101

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
IS7891A IS7891A (is)	2002-12-19	2005-06-10	Skiptitengd þrísýklísk gamma-karbólín sem serótónín viðtaka gerandefni og mótverkunarefni

Country Status (10)

Country	Link
US (1)	US7109339B2 (is)
EP (1)	EP1581221B1 (is)
JP (1)	JP4486505B2 (is)
AT (1)	ATE509929T1 (is)
AU (1)	AU2003303210A1 (is)
ES (1)	ES2364046T3 (is)
IS (1)	IS7891A (is)
NO (1)	NO20052728L (is)
PL (1)	PL377426A1 (is)
WO (1)	WO2004056324A2 (is)

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2003
- 2003-12-19 ES ES03808574T patent/ES2364046T3/es not_active Expired - Lifetime
- 2003-12-19 JP JP2004561460A patent/JP4486505B2/ja not_active Expired - Fee Related
- 2003-12-19 AT AT03808574T patent/ATE509929T1/de not_active IP Right Cessation
- 2003-12-19 EP EP03808574A patent/EP1581221B1/en not_active Expired - Lifetime
- 2003-12-19 PL PL377426A patent/PL377426A1/pl not_active Application Discontinuation
- 2003-12-19 WO PCT/US2003/041447 patent/WO2004056324A2/en not_active Ceased
- 2003-12-19 US US10/743,449 patent/US7109339B2/en not_active Expired - Lifetime
- 2003-12-19 AU AU2003303210A patent/AU2003303210A1/en not_active Abandoned
2005
- 2005-06-07 NO NO20052728A patent/NO20052728L/no not_active Application Discontinuation
- 2005-06-10 IS IS7891A patent/IS7891A/is unknown

Also Published As

Publication number	Publication date
WO2004056324A3 (en)	2004-09-02
JP4486505B2 (ja)	2010-06-23
NO20052728L (no)	2005-08-23
ATE509929T1 (de)	2011-06-15
EP1581221A2 (en)	2005-10-05
EP1581221B1 (en)	2011-05-18
ES2364046T3 (es)	2011-08-23
NO20052728D0 (no)	2005-06-07
EP1581221A4 (en)	2008-11-26
AU2003303210A1 (en)	2004-07-14
US7109339B2 (en)	2006-09-19
AU2003303210A8 (en)	2004-07-14
PL377426A1 (pl)	2006-02-06
JP2006511568A (ja)	2006-04-06
US20040180875A1 (en)	2004-09-16
WO2004056324A2 (en)	2004-07-08

Publication	Publication Date	Title
AU2003303210A8 (en)	2004-07-14	Substituted tricyclic gamma-carbolines as serotonin receptor agonists and antagonists
WO2002059129A3 (en)	2003-01-30	Substituted tetracyclic pyridoindoles as serotonin agonists and antagonists
IL156261A0 (en)	2004-01-04	Pyrroloquinoline and pyridoquinoline derivatives and pharmaceutical compositions containing the same
HK1043112A1 (zh)	2002-09-06	取代的稠杂环γ-咔啉
NO20080317L (no)	2008-02-21	Substituerte tetrahydro-1H-Pyrido[4,3-B]Indoler som serotonin reseptor-agonister og antagonister
MX2007013021A (es)	2008-01-11	Derivados de benzofuranil-alcanamina y usos de los mismos como agonistas de 5-ht2c.
EA200901162A1 (ru)	2010-04-30	Производные 1,4-дизамещённого 3-цианопиридона и их применение в качестве положительных модуляторов рецептора mglur2
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