IS8147A - New lincomycin derivatives possessing antimicrobial activity - Google Patents

New lincomycin derivatives possessing antimicrobial activity

Info

Publication number: IS8147A
Authority: IS; Iceland
Prior art keywords: new; antimicrobial activity; derivatives possessing; lincomycin derivatives; possessing antimicrobial
Prior art date: 2003-06-17

Application number

IS8147A

Other languages

Icelandic (is)

Inventor

Gustaf Lewis Jason

Anandan Sampath-Kumar

Fremont

O'dowd Hardwin

Federovich Gordeev Mikhail

Original Assignee

Vicuron Pharmaceuticals Inc.

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2003-06-17

Filing date

2005-11-24

Publication date

2005-11-24

2003-08-15 Priority claimed from US10/642,807 external-priority patent/US7164011B2/en

2004-02-11 Priority claimed from US10/777,455 external-priority patent/US7199105B2/en

2005-11-24 Application filed by Vicuron Pharmaceuticals Inc. filed Critical Vicuron Pharmaceuticals Inc.

2005-11-24 Publication of IS8147A publication Critical patent/IS8147A/en

Links

230000000845 anti-microbial effect Effects 0.000 title 1
OJMMVQQUTAEWLP-KIDUDLJLSA-N lincomycin Chemical class CN1C[C@H](CCC)C[C@H]1C(=O)N[C@H]([C@@H](C)O)[C@@H]1[C@H](O)[C@H](O)[C@@H](O)[C@@H](SC)O1 OJMMVQQUTAEWLP-KIDUDLJLSA-N 0.000 title 1

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
- A61K31/7052—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
- C07H15/02—Acyclic radicals, not substituted by cyclic structures
- C07H15/14—Acyclic radicals, not substituted by cyclic structures attached to a sulfur, selenium or tellurium atom of a saccharide radical
- C07H15/16—Lincomycin; Derivatives thereof

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Molecular Biology (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Engineering & Computer Science (AREA)
Biochemistry (AREA)
Epidemiology (AREA)
Genetics & Genomics (AREA)
Biotechnology (AREA)
Crystallography & Structural Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Bioinformatics & Cheminformatics (AREA)
Communicable Diseases (AREA)
Oncology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Preparation Of Compounds By Using Micro-Organisms (AREA)
Saccharide Compounds (AREA)

IS8147A 2003-06-17 2005-11-24 New lincomycin derivatives possessing antimicrobial activity IS8147A (en)

Applications Claiming Priority (5)

Application Number	Priority Date	Filing Date	Title
US47950203P	2003-06-17	2003-06-17
US47929603P	2003-06-17	2003-06-17
US10/642,807 US7164011B2 (en)	2002-08-15	2003-08-15	Lincomycin derivatives possessing antibacterial activity
US10/777,455 US7199105B2 (en)	2002-08-15	2004-02-11	Lincomycin derivatives possessing antibacterial activity
PCT/US2004/019689 WO2005012320A2 (en)	2003-06-17	2004-06-17	Novel lincomycin derivatives possessing antimicrobial activity

Publications (1)

Publication Number	Publication Date
IS8147A true IS8147A (en)	2005-11-24

Family

ID=40203032

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
IS8147A IS8147A (en)	2003-06-17	2005-11-24	New lincomycin derivatives possessing antimicrobial activity

Country Status (16)

Country	Link
EP (1)	EP1644393A2 (en)
JP (1)	JP2007516172A (en)
KR (1)	KR20060091050A (en)
AU (1)	AU2004261550A1 (en)
BR (1)	BRPI0411534A (en)
CA (1)	CA2528592A1 (en)
EC (1)	ECSP056233A (en)
GE (1)	GEP20084437B (en)
IL (1)	IL172183A0 (en)
IS (1)	IS8147A (en)
MA (1)	MA27860A1 (en)
MX (1)	MXPA05013915A (en)
NO (1)	NO20055893L (en)
OA (1)	OA13179A (en)
RS (1)	RS20050931A (en)
WO (1)	WO2005012320A2 (en)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US7199105B2 (en)	2002-08-15	2007-04-03	Vicuron Pharmaceuticals, Inc.	Lincomycin derivatives possessing antibacterial activity
KR20050056195A (en)	2002-08-15	2005-06-14	비큐론 파마슈티컬스 인코포레이티드	Lincomycin derivatives possessing antibacterial activity
US7256177B2 (en)	2003-06-17	2007-08-14	Vicuron Pharmaceuticals, Inc.	Lincomycin derivatives possessing antibacterial activity
CA2528596A1 (en) *	2003-06-17	2005-01-27	Vicuron Pharmaceuticals Inc.	Lincomycin derivatives possessing antibacterial activity
US7199106B2 (en)	2003-06-17	2007-04-03	Vicuron Pharmaceuticals, Inc.	Lincomycin derivatives possessing antimicrobial activity
US7361743B2 (en) *	2004-02-11	2008-04-22	Pfizer Inc	Lincomycin derivatives possessing antibacterial activity
BRPI0615300A2 (en) *	2005-08-31	2009-07-14	Wyeth Corp	compound; pharmaceutical composition; method for the preparation, treatment or control of bacterial infections in warm-blooded animals; use of a compound; and method for preparing compounds represented by formula (i)
EP1970377A4 (en)	2005-12-09	2013-02-27	Meiji Seika Kaisha	Lincomycin derivative and antibacterial agent containing the same as active ingredient
WO2008146919A1 (en)	2007-05-31	2008-12-04	Meiji Seika Kaisha, Ltd.	Lincosamide derivative, and antibacterial agent comprising the same as active ingredient
EP2151447A4 (en) *	2007-05-31	2012-09-05	Meiji Seika Kaisha	Lincomycin derivatives and antibacterial agents containing the same as the active ingredient
US20130267699A1 (en)	2011-06-24	2013-10-10	California Institute Of Technology	Quaternary heteroatom containing compounds
US8822679B2 (en) *	2011-06-24	2014-09-02	California Institute Of Technology	Quaternary heteroatom containing compounds
US10421696B2 (en)	2014-12-18	2019-09-24	California Institute Of Technology	Enantioselective synthesis of α-quaternary mannich adducts by palladium-catalyzed allylic alkylation
US10106479B2 (en)	2015-03-27	2018-10-23	California Institute Of Technology	Asymmetric catalytic decarboxylative alkyl alkylation using low catalyst concentrations and a robust precatalyst
EP3426391A4 (en)	2016-03-11	2019-08-28	California Institute of Technology	COMPOSITIONS AND METHODS FOR ACYLATION OF LACTAMS
EP3480190B1 (en)	2017-11-01	2023-01-04	California Institute of Technology	Methods for enantioselective allylic alkylation of esters, lactones, and lactams with unactivated allylic alcohols
EP3699173A1 (en)	2018-10-18	2020-08-26	California Institute of Technology	Gem-disubstituted pyrrolidines, piperazines, and diazepanes, and compositions and methods of making the same
CN110357839A (en) *	2019-08-29	2019-10-22	重庆经致制药技术开发有限公司	The preparation method of Bu Waxitan chiral intermediate

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3268556A (en) *	1964-04-13	1966-08-23	Upjohn Co	Novel lincomycin derivatives
NL128232C (en) *	1964-04-13
NL146501C (en) *	1964-07-01
US3282917A (en) *	1964-08-17	1966-11-01	Upjohn Co	Methyl n-(1-alkyl-4-alkoxy-prolyl)-alpha-thiolincosaminide compounds and process therefor
NL140527B (en) *	1965-02-08	1973-12-17	Upjohn Co	PROCESS FOR PREPARING LINCOMYCIN RELATED COMPOUNDS.
US3496163A (en) *	1965-02-08	1970-02-17	Upjohn Co	7-halo-7-deoxylincomycins and process for preparing the same
US3555007A (en) *	1968-07-22	1971-01-12	Upjohn Co	7-deoxy-7-halo lincomycin d derivatives
US3549615A (en) *	1968-10-17	1970-12-22	Upjohn Co	Lincomycin derivatives and process for producing the same
DE2118636A1 (en) *	1970-04-20	1971-11-04	The Upjohn Co., Kalamazoo, Mich. (V.StA.)	3-nucleotides of lincomycin and their analogues, processes for their preparation and their use in therapeutic preparations
US3787390A (en) *	1971-06-23	1974-01-22	Upjohn Co	Analogs of lincomycin and process
US3849396A (en) *	1973-01-08	1974-11-19	Upjohn Co	Lincomycin and clindamycin 1-o-ethers
US3923602A (en) *	1973-10-25	1975-12-02	Upjohn Co	Composition of matter and process
JPS5641239A (en) *	1979-09-13	1981-04-17	Hitachi Cable Ltd	Flame-retardant composition
US4278789A (en) *	1979-11-23	1981-07-14	The Upjohn Company	Lincomycin compounds
KR20050056195A (en) *	2002-08-15	2005-06-14	비큐론 파마슈티컬스 인코포레이티드	Lincomycin derivatives possessing antibacterial activity
BRPI0411537A (en) *	2003-06-17	2006-08-01	Vicuron Pharm Inc	lincomycin derivatives that have antibacterial activity

2004
- 2004-06-17 OA OA1200500364A patent/OA13179A/en unknown
- 2004-06-17 CA CA002528592A patent/CA2528592A1/en not_active Abandoned
- 2004-06-17 RS YUP-2005/0931A patent/RS20050931A/en unknown
- 2004-06-17 GE GEAP20049117A patent/GEP20084437B/en unknown
- 2004-06-17 AU AU2004261550A patent/AU2004261550A1/en not_active Abandoned
- 2004-06-17 BR BRPI0411534-1A patent/BRPI0411534A/en not_active IP Right Cessation
- 2004-06-17 EP EP04776816A patent/EP1644393A2/en not_active Withdrawn
- 2004-06-17 JP JP2006517464A patent/JP2007516172A/en active Pending
- 2004-06-17 MX MXPA05013915A patent/MXPA05013915A/en unknown
- 2004-06-17 WO PCT/US2004/019689 patent/WO2005012320A2/en not_active Ceased
- 2004-06-17 KR KR1020057024291A patent/KR20060091050A/en not_active Ceased
2005
- 2005-11-24 IL IL172183A patent/IL172183A0/en unknown
- 2005-11-24 IS IS8147A patent/IS8147A/en unknown
- 2005-12-12 NO NO20055893A patent/NO20055893L/en not_active Application Discontinuation
- 2005-12-16 MA MA28672A patent/MA27860A1/en unknown
- 2005-12-16 EC EC2005006233A patent/ECSP056233A/en unknown

Also Published As

Publication number	Publication date
CA2528592A1 (en)	2005-02-10
HK1090061A1 (en)	2006-12-15
JP2007516172A (en)	2007-06-21
EP1644393A2 (en)	2006-04-12
NO20055893L (en)	2006-03-14
RS20050931A (en)	2008-04-04
WO2005012320A3 (en)	2005-10-20
MA27860A1 (en)	2006-04-03
BRPI0411534A (en)	2006-08-22
OA13179A (en)	2006-12-13
WO2005012320A2 (en)	2005-02-10
KR20060091050A (en)	2006-08-17
AU2004261550A1 (en)	2005-02-10
ECSP056233A (en)	2006-04-19
GEP20084437B (en)	2008-07-25
MXPA05013915A (en)	2006-07-03
IL172183A0 (en)	2011-08-01

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PT3127553T (en)	2022-01-24	CALIQUEAMICIN DERIVATIVE CONJUGATES - CARRIER
EP1537195A4 (en)	2008-05-21	DISINFECTANT COMPOSITION
ATE383771T1 (en)	2008-02-15	FUNGICIDAL ACTIVE COMBINATIONS
IS8147A (en)	2005-11-24	New lincomycin derivatives possessing antimicrobial activity
EP1970377A4 (en)	2013-02-27	Lincomycin derivative and antibacterial agent containing the same as active ingredient
ATE392813T1 (en)	2008-05-15	FUNGICIDAL ACTIVE COMBINATION
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PT1381609E (en)	2005-05-31	5-HALOGEN-6-PHENYL-7-FLUOROALQUILAMINO-TRIAZOLOPYRIMIDINES AS FUNGICIDES
IL166476A0 (en)	2006-01-15	Lincomycin derivatives possessing antibacterial activity
IS7795A (en)	2005-04-11	Pyrrole derivatives as compounds against fungal bacteria
ATA17802003A (en)	2005-11-15	FURNITURE ARRANGEMENT
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ZA200602947B (en)	2007-09-26	Pyrrol derivatives with antibacterial activity
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EP1483253A4 (en)	2007-03-21	ANTIMICROBIAL AGENT