IT1126577B - 4(3h)-chinazolinoni sostituiti nella meta' 3-aromatica,procedimento per la loro produzione e loro impiego - Google Patents

4(3h)-chinazolinoni sostituiti nella meta' 3-aromatica,procedimento per la loro produzione e loro impiego

Info

Publication number
IT1126577B
IT1126577B IT28062/79A IT2806279A IT1126577B IT 1126577 B IT1126577 B IT 1126577B IT 28062/79 A IT28062/79 A IT 28062/79A IT 2806279 A IT2806279 A IT 2806279A IT 1126577 B IT1126577 B IT 1126577B
Authority
IT
Italy
Prior art keywords
chinazolinones
replaced
procedure
production
aromatic
Prior art date
Application number
IT28062/79A
Other languages
English (en)
Other versions
IT7928062A0 (it
Inventor
Masayuki Ishikawa
Hiromichi Tanaka
Yukuo Eguchi
Shigeru Ito
Yishimi Takashima
Masahiko Kobayashi
Original Assignee
Masayuki Ishikawa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP15576478A external-priority patent/JPS5583761A/ja
Priority claimed from JP12673879A external-priority patent/JPS5651461A/ja
Priority claimed from JP13358279A external-priority patent/JPS5657768A/ja
Priority claimed from JP14198779A external-priority patent/JPS5665877A/ja
Application filed by Masayuki Ishikawa filed Critical Masayuki Ishikawa
Publication of IT7928062A0 publication Critical patent/IT7928062A0/it
Application granted granted Critical
Publication of IT1126577B publication Critical patent/IT1126577B/it

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72—Quinazolines; Hydrogenated quinazolines
    • C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/88—Oxygen atoms
    • C07D239/91—Oxygen atoms with aryl or aralkyl radicals attached in position 2 or 3

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Furan Compounds (AREA)
IT28062/79A 1978-12-19 1979-12-17 4(3h)-chinazolinoni sostituiti nella meta' 3-aromatica,procedimento per la loro produzione e loro impiego IT1126577B (it)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
JP15576478A JPS5583761A (en) 1978-12-19 1978-12-19 Novel 3-phenyl-4-quinazolone derivative
JP12673879A JPS5651461A (en) 1979-10-03 1979-10-03 Novel 3-phenyl-4-quinazolone derivative
JP13358279A JPS5657768A (en) 1979-10-18 1979-10-18 Novel 4-quinazolone derivative substituted by aromatic residue at 3-position
JP14198779A JPS5665877A (en) 1979-11-05 1979-11-05 Preparation of 4-quinazolone derivative

Publications (2)

Publication Number Publication Date
IT7928062A0 IT7928062A0 (it) 1979-12-17
IT1126577B true IT1126577B (it) 1986-05-21

Family

ID=27471233

Family Applications (1)

Application Number Title Priority Date Filing Date
IT28062/79A IT1126577B (it) 1978-12-19 1979-12-17 4(3h)-chinazolinoni sostituiti nella meta' 3-aromatica,procedimento per la loro produzione e loro impiego

Country Status (16)

Country Link
US (1) US4276295A (it)
AR (1) AR225028A1 (it)
AU (1) AU526309B2 (it)
CH (1) CH644112A5 (it)
DD (1) DD150462A5 (it)
DE (1) DE2950376A1 (it)
DK (1) DK539979A (it)
FR (1) FR2444671A1 (it)
GB (1) GB2040927B (it)
HU (1) HU182733B (it)
IT (1) IT1126577B (it)
NL (1) NL7909118A (it)
NO (1) NO794135L (it)
NZ (1) NZ192392A (it)
SE (1) SE7910376L (it)
YU (1) YU306379A (it)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1161036A (en) * 1980-05-15 1984-01-24 Masayuki Ishikawa Quinazoline-dione compounds, process for production thereof and pharmaceutical use thereof
AU543928B2 (en) * 1981-01-16 1985-05-09 Masayuki Ishikawa 4(311)-quinazolinone derivatives
US4419357A (en) * 1982-01-18 1983-12-06 The Dow Chemical Company 3-(1H-Tetrazol-5-yl)-4(3H)-quinazolinones
US4684654A (en) * 1985-08-14 1987-08-04 American Cyanamid Company 3-heteroalkyl-2,4-quinzaolinediones
EP0293500A1 (en) * 1987-06-01 1988-12-07 American Cyanamid Company 3-heteroalkyl-2,4.quinzaoline-diones
WO1991012001A1 (en) * 1990-02-13 1991-08-22 Merck & Co., Inc. Angiotensin ii antagonists incorporating a substituted benzyl element
US5075313A (en) * 1990-09-13 1991-12-24 Eli Lilly And Company 3-aryl-4(3H)quinazolinone CCK antagonists and pharmaceutical formulations thereof
US5283247A (en) * 1991-02-06 1994-02-01 Research Corporation Technologies, Inc. Anticonvulsant substituted quinazolones
WO1992013535A1 (en) * 1991-02-06 1992-08-20 Research Corporation Technologies, Inc. Anticonvulsant substituted quinazolones
RU2139862C1 (ru) * 1993-05-12 1999-10-20 Е.И. Дю Пон де Немурс энд Компани Замещенные 4(3н)-хиназолиноны, обладающие фунгицидными свойствами, композиции на их основе и способы борьбы с мучнистой росой
US5756502A (en) * 1994-08-08 1998-05-26 Warner-Lambert Company Quinazolinone derivatives as cholyecystokinin (CCK) ligands
US6255311B1 (en) * 1998-01-14 2001-07-03 E. I. Du Pont De Nemours And Company Fungicidal fused bicyclic pyrimidinones
WO2002026718A2 (en) * 2000-09-29 2002-04-04 Millennium Pharmaceutical, Inc. Bicyclic pyrimidin-4-one based inhibitors of factor xa
AU2007202781B2 (en) * 2002-02-06 2010-09-09 Novartis Ag Quinazolinone derivatives and their use as CB agonists
TW200306839A (en) * 2002-02-06 2003-12-01 Novartis Ag Quinazolinone derivatives and their use as CB agonists
BRPI0507629A (pt) * 2004-02-13 2007-07-03 Banyu Pharma Co Ltd composto, antagonista do receptor e agonista inverso do receptor da histamina h3, agente profilático ou terapêutico para uma doença metabólica, uma doença circulatória ou uma doença do sistema nervoso, ou um seu sal farmaceuticamente aceitável
JP6258918B2 (ja) * 2012-04-10 2018-01-10 アンジー ファーマスーティカル カンパニー リミテッドAnnji Pharamaceutical Co., Ltd. ヒストンデアセチラーゼ(hdacs)阻害剤

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3047462A (en) * 1959-03-06 1962-07-31 Lab Jacques Logeais Soc D Expl Quinazolone anti-inflammatory composition
DE1695799C3 (de) * 1967-01-23 1974-10-17 Sumitomo Chemical Co., Ltd., Osaka (Japan) 5-Chlor-3- eckige Klammer auf pyridin-2'-yl eckige Klammer zu -4-(3H)- chinazolinone
JPS5516425B2 (it) * 1972-09-19 1980-05-01
JPS5521748B2 (it) * 1972-09-19 1980-06-12

Also Published As

Publication number Publication date
IT7928062A0 (it) 1979-12-17
AU526309B2 (en) 1983-01-06
NZ192392A (en) 1983-02-15
GB2040927A (en) 1980-09-03
US4276295A (en) 1981-06-30
AR225028A1 (es) 1982-02-15
YU306379A (en) 1983-12-31
DD150462A5 (de) 1981-09-02
GB2040927B (en) 1983-01-26
FR2444671B1 (it) 1983-06-10
HU182733B (en) 1984-03-28
SE7910376L (sv) 1980-06-20
NO794135L (no) 1980-06-20
NL7909118A (nl) 1980-06-23
FR2444671A1 (fr) 1980-07-18
CH644112A5 (de) 1984-07-13
AU5393279A (en) 1980-06-26
DE2950376A1 (de) 1980-07-10
DK539979A (da) 1980-06-20

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