IT1223327B - Composti eterociclici alifatici n sostituiti atti a facilitare il passaggio di sostanze attive attraverso le barrierefisiologiche - Google Patents

Composti eterociclici alifatici n sostituiti atti a facilitare il passaggio di sostanze attive attraverso le barrierefisiologiche

Info

Publication number
IT1223327B
IT1223327B IT22423/87A IT2242387A IT1223327B IT 1223327 B IT1223327 B IT 1223327B IT 22423/87 A IT22423/87 A IT 22423/87A IT 2242387 A IT2242387 A IT 2242387A IT 1223327 B IT1223327 B IT 1223327B
Authority
IT
Italy
Prior art keywords
substituted
facilitate
passage
active substances
heterocyclic compounds
Prior art date
Application number
IT22423/87A
Other languages
English (en)
Other versions
IT8722423A0 (it
Inventor
C Meroni
S Maiorana
P L Rugarli
P G Pagella
Original Assignee
Mediolanum Farmaceutici Srl
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Mediolanum Farmaceutici Srl filed Critical Mediolanum Farmaceutici Srl
Priority to IT22423/87A priority Critical patent/IT1223327B/it
Publication of IT8722423A0 publication Critical patent/IT8722423A0/it
Priority to EP88117557A priority patent/EP0314008A3/en
Priority to KR1019880014068A priority patent/KR890006607A/ko
Priority to JP63271111A priority patent/JPH01151566A/ja
Application granted granted Critical
Publication of IT1223327B publication Critical patent/IT1223327B/it

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/02—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms containing only hydrogen and carbon atoms in addition to the ring hetero elements
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
    • C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
    • C07D295/182—Radicals derived from carboxylic acids
    • C07D295/185—Radicals derived from carboxylic acids from aliphatic carboxylic acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/02—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms containing only hydrogen and carbon atoms in addition to the ring hetero elements
    • C07D295/027—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms containing only hydrogen and carbon atoms in addition to the ring hetero elements containing only one hetero ring
    • C07D295/03—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms containing only hydrogen and carbon atoms in addition to the ring hetero elements containing only one hetero ring with the ring nitrogen atoms directly attached to acyclic carbon atoms

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Pulmonology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
IT22423/87A 1987-10-28 1987-10-28 Composti eterociclici alifatici n sostituiti atti a facilitare il passaggio di sostanze attive attraverso le barrierefisiologiche IT1223327B (it)

Priority Applications (4)

Application Number Priority Date Filing Date Title
IT22423/87A IT1223327B (it) 1987-10-28 1987-10-28 Composti eterociclici alifatici n sostituiti atti a facilitare il passaggio di sostanze attive attraverso le barrierefisiologiche
EP88117557A EP0314008A3 (en) 1987-10-28 1988-10-21 N-substituted aliphatic heterocyclic compounds able to facilitate the passage of active substances through physiological barriers
KR1019880014068A KR890006607A (ko) 1987-10-28 1988-10-28 생리학적 장벽을 통한 활성물질의 통과를 용이하게 할 수 있는 n-치환된 지방족 헤테로 사이클릭 화합물
JP63271111A JPH01151566A (ja) 1987-10-28 1988-10-28 活性物質の生理的障壁通過を促進するｎ−置換脂肪族複素環式化合物

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT22423/87A IT1223327B (it) 1987-10-28 1987-10-28 Composti eterociclici alifatici n sostituiti atti a facilitare il passaggio di sostanze attive attraverso le barrierefisiologiche

Publications (2)

Publication Number Publication Date
IT8722423A0 IT8722423A0 (it) 1987-10-28
IT1223327B true IT1223327B (it) 1990-09-19

Family

ID=11196109

Family Applications (1)

Application Number Title Priority Date Filing Date
IT22423/87A IT1223327B (it) 1987-10-28 1987-10-28 Composti eterociclici alifatici n sostituiti atti a facilitare il passaggio di sostanze attive attraverso le barrierefisiologiche

Country Status (4)

Country Link
EP (1) EP0314008A3 (it)
JP (1) JPH01151566A (it)
KR (1) KR890006607A (it)
IT (1) IT1223327B (it)

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2947649A1 (de) * 1979-11-27 1981-08-06 C.F. Spiess & Sohn GmbH & Co, 6719 Kleinkarlbach Insektizide mittel
DE2947648A1 (de) * 1979-11-27 1981-08-06 C.F. Spiess & Sohn GmbH & Co, 6719 Kleinkarlbach Verwendung tertiaerer heterocyclischer amine als potenzierungsmittel fuer insektizide
CA1308352C (en) * 1986-08-15 1992-10-06 James V. Peck Compositions comprising 1-oxohydrocarbyl-substituted azacyclohexanes
CA1319613C (en) * 1986-10-07 1993-06-29 Gevork Minaskanian Penetration enhancers for transdermal delivery of systemic agents
JPS63301812A (ja) * 1987-06-01 1988-12-08 Nichibai Boeki Kk 抗齲蝕剤
JPS6445302A (en) * 1987-08-13 1989-02-17 Yoshinori Tsuda Vermicide

Also Published As

Publication number Publication date
JPH01151566A (ja) 1989-06-14
EP0314008A3 (en) 1990-07-25
IT8722423A0 (it) 1987-10-28
EP0314008A2 (en) 1989-05-03
KR890006607A (ko) 1989-06-14

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