IT1239745B - Impiego di a-amminofluorochetoni per la preparazione di medicamenti ad attivita' cardiovascolare e antipertensiva. - Google Patents

Impiego di a-amminofluorochetoni per la preparazione di medicamenti ad attivita' cardiovascolare e antipertensiva.

Info

Publication number
IT1239745B
IT1239745B IT47551A IT4755190A IT1239745B IT 1239745 B IT1239745 B IT 1239745B IT 47551 A IT47551 A IT 47551A IT 4755190 A IT4755190 A IT 4755190A IT 1239745 B IT1239745 B IT 1239745B
Authority
IT
Italy
Prior art keywords
fluoroketones
medications
cardiovascular
amino
preparation
Prior art date
Application number
IT47551A
Other languages
English (en)
Italian (it)
Other versions
IT9047551A0 (it
IT9047551A1 (it
Inventor
Anis Khusro Mir
Original Assignee
Sandoz Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sandoz Ag filed Critical Sandoz Ag
Publication of IT9047551A0 publication Critical patent/IT9047551A0/it
Publication of IT9047551A1 publication Critical patent/IT9047551A1/it
Application granted granted Critical
Publication of IT1239745B publication Critical patent/IT1239745B/it

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/005Enzyme inhibitors
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/195Carboxylic acids, e.g. valproic acid having an amino group
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/04Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Immunology (AREA)
  • Cardiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Organic Chemistry (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Hydrogenated Pyridines (AREA)
  • Pyrrole Compounds (AREA)
IT47551A 1989-01-26 1990-01-22 Impiego di a-amminofluorochetoni per la preparazione di medicamenti ad attivita' cardiovascolare e antipertensiva. IT1239745B (it)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH23889 1989-01-26

Publications (3)

Publication Number Publication Date
IT9047551A0 IT9047551A0 (it) 1990-01-22
IT9047551A1 IT9047551A1 (it) 1990-07-27
IT1239745B true IT1239745B (it) 1993-11-15

Family

ID=4182438

Family Applications (1)

Application Number Title Priority Date Filing Date
IT47551A IT1239745B (it) 1989-01-26 1990-01-22 Impiego di a-amminofluorochetoni per la preparazione di medicamenti ad attivita' cardiovascolare e antipertensiva.

Country Status (6)

Country Link
JP (1) JPH02247123A (fr)
BE (1) BE1003340A3 (fr)
DE (1) DE4001087A1 (fr)
FR (1) FR2641972A1 (fr)
GB (1) GB2227411A (fr)
IT (1) IT1239745B (fr)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5101068A (en) * 1990-02-16 1992-03-31 Prototek Inc. Magnesium fluoromalonates
JP3228347B2 (ja) * 1991-06-25 2001-11-12 三菱化学株式会社 シクロプロペノン誘導体
US5395958A (en) * 1992-09-30 1995-03-07 Mitsubishi Kasei Corporation Cyclopropene derivatives
DE69610978D1 (de) * 1995-03-31 2000-12-21 Naeja Pharmaceutical Inc 4-substituierte-3-peptidyl-azetidin-2-on-derivate als cystein-proteinase inhibitoren

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4518528A (en) * 1983-05-19 1985-05-21 Rasnick David W α Amino fluoro ketones

Also Published As

Publication number Publication date
JPH02247123A (ja) 1990-10-02
GB2227411A (en) 1990-08-01
BE1003340A3 (fr) 1992-03-03
IT9047551A0 (it) 1990-01-22
GB9001453D0 (en) 1990-03-21
IT9047551A1 (it) 1990-07-27
FR2641972A1 (fr) 1990-07-27
DE4001087A1 (de) 1990-08-02

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Legal Events

Date Code Title Description
0001 Granted
TA Fee payment date (situation as of event date), data collected since 19931001

Effective date: 19940224