IT1239745B - Impiego di a-amminofluorochetoni per la preparazione di medicamenti ad attivita' cardiovascolare e antipertensiva. - Google Patents
Impiego di a-amminofluorochetoni per la preparazione di medicamenti ad attivita' cardiovascolare e antipertensiva.Info
- Publication number
- IT1239745B IT1239745B IT47551A IT4755190A IT1239745B IT 1239745 B IT1239745 B IT 1239745B IT 47551 A IT47551 A IT 47551A IT 4755190 A IT4755190 A IT 4755190A IT 1239745 B IT1239745 B IT 1239745B
- Authority
- IT
- Italy
- Prior art keywords
- fluoroketones
- medications
- cardiovascular
- amino
- preparation
- Prior art date
Links
- 230000003276 anti-hypertensive effect Effects 0.000 title 1
- 229940079593 drug Drugs 0.000 title 1
- 239000003814 drug Substances 0.000 title 1
- 230000002526 effect on cardiovascular system Effects 0.000 title 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/005—Enzyme inhibitors
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Epidemiology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Immunology (AREA)
- Cardiology (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Heart & Thoracic Surgery (AREA)
- Organic Chemistry (AREA)
- Gastroenterology & Hepatology (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Hydrogenated Pyridines (AREA)
- Pyrrole Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CH23889 | 1989-01-26 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| IT9047551A0 IT9047551A0 (it) | 1990-01-22 |
| IT9047551A1 IT9047551A1 (it) | 1990-07-27 |
| IT1239745B true IT1239745B (it) | 1993-11-15 |
Family
ID=4182438
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IT47551A IT1239745B (it) | 1989-01-26 | 1990-01-22 | Impiego di a-amminofluorochetoni per la preparazione di medicamenti ad attivita' cardiovascolare e antipertensiva. |
Country Status (6)
| Country | Link |
|---|---|
| JP (1) | JPH02247123A (fr) |
| BE (1) | BE1003340A3 (fr) |
| DE (1) | DE4001087A1 (fr) |
| FR (1) | FR2641972A1 (fr) |
| GB (1) | GB2227411A (fr) |
| IT (1) | IT1239745B (fr) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5101068A (en) * | 1990-02-16 | 1992-03-31 | Prototek Inc. | Magnesium fluoromalonates |
| JP3228347B2 (ja) * | 1991-06-25 | 2001-11-12 | 三菱化学株式会社 | シクロプロペノン誘導体 |
| US5395958A (en) * | 1992-09-30 | 1995-03-07 | Mitsubishi Kasei Corporation | Cyclopropene derivatives |
| DE69610978D1 (de) * | 1995-03-31 | 2000-12-21 | Naeja Pharmaceutical Inc | 4-substituierte-3-peptidyl-azetidin-2-on-derivate als cystein-proteinase inhibitoren |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4518528A (en) * | 1983-05-19 | 1985-05-21 | Rasnick David W | α Amino fluoro ketones |
-
1990
- 1990-01-17 DE DE4001087A patent/DE4001087A1/de not_active Withdrawn
- 1990-01-22 GB GB9001453A patent/GB2227411A/en not_active Withdrawn
- 1990-01-22 IT IT47551A patent/IT1239745B/it active IP Right Grant
- 1990-01-22 FR FR9000777A patent/FR2641972A1/fr active Pending
- 1990-01-22 BE BE9000075A patent/BE1003340A3/fr not_active IP Right Cessation
- 1990-01-25 JP JP2015948A patent/JPH02247123A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| JPH02247123A (ja) | 1990-10-02 |
| GB2227411A (en) | 1990-08-01 |
| BE1003340A3 (fr) | 1992-03-03 |
| IT9047551A0 (it) | 1990-01-22 |
| GB9001453D0 (en) | 1990-03-21 |
| IT9047551A1 (it) | 1990-07-27 |
| FR2641972A1 (fr) | 1990-07-27 |
| DE4001087A1 (de) | 1990-08-02 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| 0001 | Granted | ||
| TA | Fee payment date (situation as of event date), data collected since 19931001 |
Effective date: 19940224 |