IT1400964B1 - Procedimento per la preparazione di derivati pteridinici - Google Patents
Procedimento per la preparazione di derivati pteridiniciInfo
- Publication number
- IT1400964B1 IT1400964B1 ITMI2010A001076A ITMI20101076A IT1400964B1 IT 1400964 B1 IT1400964 B1 IT 1400964B1 IT MI2010A001076 A ITMI2010A001076 A IT MI2010A001076A IT MI20101076 A ITMI20101076 A IT MI20101076A IT 1400964 B1 IT1400964 B1 IT 1400964B1
- Authority
- IT
- Italy
- Prior art keywords
- procedure
- preparation
- pteridine derivatives
- pteridine
- derivatives
- Prior art date
Links
- CPNGPNLZQNNVQM-UHFFFAOYSA-N pteridine Chemical class N1=CN=CC2=NC=CN=C21 CPNGPNLZQNNVQM-UHFFFAOYSA-N 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D475/00—Heterocyclic compounds containing pteridine ring systems
- C07D475/02—Heterocyclic compounds containing pteridine ring systems with an oxygen atom directly attached in position 4
- C07D475/04—Heterocyclic compounds containing pteridine ring systems with an oxygen atom directly attached in position 4 with a nitrogen atom directly attached in position 2
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
- C07D333/08—Hydrogen atoms or radicals containing only hydrogen and carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D337/00—Heterocyclic compounds containing rings of more than six members having one sulfur atom as the only ring hetero atom
- C07D337/02—Seven-membered rings
- C07D337/04—Seven-membered rings not condensed with other rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D337/00—Heterocyclic compounds containing rings of more than six members having one sulfur atom as the only ring hetero atom
- C07D337/02—Seven-membered rings
- C07D337/06—Seven-membered rings condensed with carbocyclic rings or ring systems
- C07D337/08—Seven-membered rings condensed with carbocyclic rings or ring systems condensed with one six-membered ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D339/00—Heterocyclic compounds containing rings having two sulfur atoms as the only ring hetero atoms
- C07D339/02—Five-membered rings
- C07D339/06—Five-membered rings having the hetero atoms in positions 1 and 3, e.g. cyclic dithiocarbonates
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D339/00—Heterocyclic compounds containing rings having two sulfur atoms as the only ring hetero atoms
- C07D339/08—Six-membered rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H3/00—Compounds containing only hydrogen atoms and saccharide radicals having only carbon, hydrogen, and oxygen atoms
- C07H3/02—Monosaccharides
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H9/00—Compounds containing a hetero ring sharing at least two hetero atoms with a saccharide radical
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Health & Medical Sciences (AREA)
- Biochemistry (AREA)
- Biotechnology (AREA)
- General Health & Medical Sciences (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Saccharide Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Catalysts (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Priority Applications (9)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ITMI2010A001076A IT1400964B1 (it) | 2010-06-15 | 2010-06-15 | Procedimento per la preparazione di derivati pteridinici |
| US13/703,932 US8809553B2 (en) | 2010-06-15 | 2011-06-13 | Process for the preparation of pteridine derivatives |
| PL11730560T PL2582711T3 (pl) | 2010-06-15 | 2011-06-13 | Sposób wytwarzania pochodnych pterydyny |
| ES11730560.7T ES2525357T3 (es) | 2010-06-15 | 2011-06-13 | Proceso para la preparación de derivados de pteridina |
| CN201180029143.XA CN102939298B (zh) | 2010-06-15 | 2011-06-13 | 制备蝶啶衍生物的方法 |
| AU2011267471A AU2011267471B8 (en) | 2010-06-15 | 2011-06-13 | Process for the preparation of pteridine derivatives |
| EP11730560.7A EP2582711B1 (en) | 2010-06-15 | 2011-06-13 | Process for the preparation of pteridine derivatives |
| JP2013514578A JP5972867B2 (ja) | 2010-06-15 | 2011-06-13 | プテリジン誘導体の調製方法 |
| PCT/EP2011/002896 WO2011157388A1 (en) | 2010-06-15 | 2011-06-13 | Process for the preparation of pteridine derivatives |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ITMI2010A001076A IT1400964B1 (it) | 2010-06-15 | 2010-06-15 | Procedimento per la preparazione di derivati pteridinici |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| ITMI20101076A1 ITMI20101076A1 (it) | 2011-12-16 |
| IT1400964B1 true IT1400964B1 (it) | 2013-07-05 |
Family
ID=43332261
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ITMI2010A001076A IT1400964B1 (it) | 2010-06-15 | 2010-06-15 | Procedimento per la preparazione di derivati pteridinici |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US8809553B2 (it) |
| EP (1) | EP2582711B1 (it) |
| JP (1) | JP5972867B2 (it) |
| CN (1) | CN102939298B (it) |
| AU (1) | AU2011267471B8 (it) |
| ES (1) | ES2525357T3 (it) |
| IT (1) | IT1400964B1 (it) |
| PL (1) | PL2582711T3 (it) |
| WO (1) | WO2011157388A1 (it) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN102627644B (zh) * | 2012-04-10 | 2014-04-16 | 凯莱英医药集团（天津）股份有限公司 | 一种通过直接手性合成方法制备二盐酸沙丙蝶呤的方法 |
| WO2016101211A1 (zh) * | 2014-12-25 | 2016-06-30 | 北京卡威生物医药科技有限公司 | 一种盐酸沙丙喋呤的制备方法 |
| CN107353314A (zh) * | 2016-05-10 | 2017-11-17 | 江苏福锌雨医药科技有限公司 | 一种5-脱氧-l-阿拉伯糖的合成方法 |
| CN106117097B (zh) * | 2016-06-20 | 2017-12-05 | 四川大学 | L‑鼠李糖二烷基缩硫醛类化合物的制备方法 |
| CN109776540B (zh) * | 2017-11-15 | 2021-07-06 | 北京启慧生物医药有限公司 | 一种盐酸沙丙蝶呤的制备方法 |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3505329A (en) * | 1968-02-06 | 1970-04-07 | Smithkline Corp | Process for the synthesis of biopterin |
| JPS60169493A (ja) * | 1984-02-14 | 1985-09-02 | Suntory Ltd | ５−デオキシ−ｌ−アラビノ−スの製造法 |
| US4713454A (en) | 1985-01-28 | 1987-12-15 | Shiratori Pharmaceutical Co., Ltd. | Preparation process of (6R)-tetrahydro-L-biopterin |
| JPS62175495A (ja) * | 1986-01-27 | 1987-08-01 | Noguchi Kenkyusho | 糖ジチオアセタ−ル誘導体の製造方法 |
| JPH0723367B2 (ja) * | 1986-02-27 | 1995-03-15 | サントリー株式会社 | オキサビシクロヘプタン誘導体 |
| US5502073A (en) * | 1987-06-05 | 1996-03-26 | The Wellcome Foundation | Heterocyclic pesticidal compounds |
| JPH09132589A (ja) * | 1995-09-08 | 1997-05-20 | Microbial Chem Res Found | 糖部分の水酸基をモノ−または−ジ−ｏ−アミノアルカノイル化された含フッ素アンスラサイクリン誘導体 |
| WO2006070862A1 (ja) * | 2004-12-28 | 2006-07-06 | Asubio Pharma Co., Ltd. | アルドース類の減炭素化合物の製造方法 |
-
2010
- 2010-06-15 IT ITMI2010A001076A patent/IT1400964B1/it active
-
2011
- 2011-06-13 JP JP2013514578A patent/JP5972867B2/ja active Active
- 2011-06-13 CN CN201180029143.XA patent/CN102939298B/zh not_active Expired - Fee Related
- 2011-06-13 ES ES11730560.7T patent/ES2525357T3/es active Active
- 2011-06-13 PL PL11730560T patent/PL2582711T3/pl unknown
- 2011-06-13 EP EP11730560.7A patent/EP2582711B1/en active Active
- 2011-06-13 AU AU2011267471A patent/AU2011267471B8/en not_active Ceased
- 2011-06-13 US US13/703,932 patent/US8809553B2/en active Active
- 2011-06-13 WO PCT/EP2011/002896 patent/WO2011157388A1/en not_active Ceased
Also Published As
| Publication number | Publication date |
|---|---|
| CN102939298A (zh) | 2013-02-20 |
| EP2582711B1 (en) | 2014-11-12 |
| ITMI20101076A1 (it) | 2011-12-16 |
| US8809553B2 (en) | 2014-08-19 |
| CN102939298B (zh) | 2015-11-25 |
| ES2525357T3 (es) | 2014-12-22 |
| AU2011267471B8 (en) | 2014-09-11 |
| PL2582711T3 (pl) | 2015-04-30 |
| JP5972867B2 (ja) | 2016-08-17 |
| JP2013531654A (ja) | 2013-08-08 |
| WO2011157388A1 (en) | 2011-12-22 |
| EP2582711A1 (en) | 2013-04-24 |
| AU2011267471A1 (en) | 2013-01-10 |
| US20130090474A1 (en) | 2013-04-11 |
| AU2011267471B2 (en) | 2014-08-28 |
| WO2011157388A8 (en) | 2012-03-15 |
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