IT8847794A0 - Derivati dell'acido furanuronico, loro preparazione e loro impiego come medicamenti - Google Patents

Derivati dell'acido furanuronico, loro preparazione e loro impiego come medicamenti

Info

Publication number
IT8847794A0
IT8847794A0 IT8847794A IT4779488A IT8847794A0 IT 8847794 A0 IT8847794 A0 IT 8847794A0 IT 8847794 A IT8847794 A IT 8847794A IT 4779488 A IT4779488 A IT 4779488A IT 8847794 A0 IT8847794 A0 IT 8847794A0
Authority
IT
Italy
Prior art keywords
medicines
derivatives
preparation
furanuronic
acid
Prior art date
Application number
IT8847794A
Other languages
English (en)
Other versions
IT1219892B (it
Inventor
Gadient Fulvio
Vogel Arnold
Original Assignee
Sandoz Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sandoz Ag filed Critical Sandoz Ag
Publication of IT8847794A0 publication Critical patent/IT8847794A0/it
Application granted granted Critical
Publication of IT1219892B publication Critical patent/IT1219892B/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/16Purine radicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Animal Behavior & Ethology (AREA)
  • Cardiology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
IT47794/88A 1987-04-06 1988-03-30 Derivati dell' acido furanuronico,loro preparazione e loro impiego come medicamenti IT1219892B (it)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
DE3711563 1987-04-06
DE3711561 1987-04-06
DE3711564 1987-04-06
DE3711562 1987-04-06

Publications (2)

Publication Number Publication Date
IT8847794A0 true IT8847794A0 (it) 1988-03-30
IT1219892B IT1219892B (it) 1990-05-24

Family

ID=27433888

Family Applications (1)

Application Number Title Priority Date Filing Date
IT47794/88A IT1219892B (it) 1987-04-06 1988-03-30 Derivati dell' acido furanuronico,loro preparazione e loro impiego come medicamenti

Country Status (22)

Country Link
JP (1) JPS63258892A (it)
KR (1) KR880012629A (it)
AT (1) AT393507B (it)
AU (1) AU609109B2 (it)
BE (1) BE1002151A5 (it)
CA (1) CA1326017C (it)
CH (1) CH676121A5 (it)
DK (1) DK183488A (it)
ES (1) ES2007177A6 (it)
FI (1) FI87463C (it)
FR (1) FR2613367A1 (it)
GB (1) GB2203149B (it)
HU (1) HU201955B (it)
IL (1) IL85969A (it)
IT (1) IT1219892B (it)
LU (1) LU87181A1 (it)
MY (1) MY102323A (it)
NL (1) NL8800862A (it)
NZ (1) NZ224131A (it)
PH (1) PH25424A (it)
PT (1) PT87153B (it)
SE (1) SE8801236L (it)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4755594A (en) * 1986-01-31 1988-07-05 Warner-Lambert Company N6 -substituted adenosines
US5063233A (en) * 1986-11-14 1991-11-05 Ciba-Geigy Corporation N9 -cyclopentyl-substituted adenine derivatives useful as adenosine receptor agonists
US4954504A (en) * 1986-11-14 1990-09-04 Ciba-Geigy Corporation N9 -cyclopentyl-substituted adenine derivatives having adenosine-2 receptor stimulating activity
HU198950B (en) * 1986-12-15 1989-12-28 Sandoz Ag Process for producing new furanuronic acid derivatives and pharmaceutical compositions comprising such compounds
US4968697A (en) * 1987-02-04 1990-11-06 Ciba-Geigy Corporation 2-substituted adenosine 5'-carboxamides as antihypertensive agents
EP0277917A3 (en) * 1987-02-04 1990-03-28 Ciba-Geigy Ag Certain adenosine 5'-carboxamide derivatives
USRE36494E (en) * 1990-02-20 2000-01-11 Discovery Therapeutics, Inc. 2-aralkoxy and 2-alkoxy adenosine derivatives as coronary vasodilators and antihypertensive agents
US5140015A (en) * 1990-02-20 1992-08-18 Whitby Research, Inc. 2-aralkoxy and 2-alkoxy adenosine derivatives as coronary vasodilators and antihypertensive agents
IT1254915B (it) * 1992-04-24 1995-10-11 Gloria Cristalli Derivati di adenosina ad attivita' a2 agonista
GB9301000D0 (en) * 1993-01-20 1993-03-10 Glaxo Group Ltd Chemical compounds
TW528755B (en) 1996-12-24 2003-04-21 Glaxo Group Ltd 2-(purin-9-yl)-tetrahydrofuran-3,4-diol derivatives
YU44900A (sh) 1998-01-31 2003-01-31 Glaxo Group Limited Derivati 2-(purin-9-il)tetrahidrofuran-3,4-diola
JP3933870B2 (ja) 1998-06-23 2007-06-20 グラクソ グループ リミテッド 2−(プリン−9−イル)−テトラヒドロフラン−3,4−ジオール誘導体
AR023463A1 (es) 1999-04-16 2002-09-04 Schering Corp Uso de compuestos de azetidinona
US20050033044A1 (en) 2003-05-19 2005-02-10 Bristol-Myers Squibb Pharma Company Methods for preparing 2-alkynyladenosine derivatives
PE20060272A1 (es) 2004-05-24 2006-05-22 Glaxo Group Ltd (2r,3r,4s,5r,2'r,3'r,4's,5's)-2,2'-{trans-1,4-ciclohexanodiilbis-[imino(2-{[2-(1-metil-1h-imidazol-4-il)etil]amino}-9h-purin-6,9-diil)]}bis[5-(2-etil-2h-tetrazol-5-il)tetrahidro-3,4-furanodiol] como agonista a2a
MX2007003271A (es) * 2004-09-20 2007-06-05 Inotek Pharmaceuticals Corp Derivados de purina y metodos de uso de los mismos.
GB0514809D0 (en) 2005-07-19 2005-08-24 Glaxo Group Ltd Compounds

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH606084A5 (en) * 1975-02-18 1978-10-13 Hoffmann La Roche (Di) nitrates of adenosine -5'-carboxylic acid derivs
US4167565A (en) * 1976-11-08 1979-09-11 Abbott Laboratories Adenosine-5'-carboxamides and method of use
DE3406533A1 (de) * 1984-02-23 1985-08-29 Boehringer Mannheim Gmbh, 6800 Mannheim Verwendung von adenosin-derivaten als antiallergica und arzneimittel, die diese enthalten
HU198950B (en) * 1986-12-15 1989-12-28 Sandoz Ag Process for producing new furanuronic acid derivatives and pharmaceutical compositions comprising such compounds
EP0277917A3 (en) * 1987-02-04 1990-03-28 Ciba-Geigy Ag Certain adenosine 5'-carboxamide derivatives

Also Published As

Publication number Publication date
BE1002151A5 (fr) 1990-08-07
KR880012629A (ko) 1988-11-28
MY102323A (en) 1992-05-28
PT87153A (pt) 1988-05-01
DK183488A (da) 1988-10-07
CH676121A5 (it) 1990-12-14
AU609109B2 (en) 1991-04-26
IL85969A (en) 1992-03-29
AT393507B (de) 1991-11-11
HUT48902A (en) 1989-07-28
SE8801236A0 (sv) 1988-10-17
NL8800862A (nl) 1988-11-01
ES2007177A6 (es) 1989-06-01
HU201955B (en) 1991-01-28
IT1219892B (it) 1990-05-24
DK183488D0 (da) 1988-04-05
FR2613367A1 (fr) 1988-10-07
ATA87388A (de) 1991-04-15
FI881571A0 (fi) 1988-04-05
FI87463C (fi) 1993-01-11
FI87463B (fi) 1992-09-30
CA1326017C (en) 1994-01-11
FI881571L (fi) 1988-10-07
LU87181A1 (fr) 1988-11-17
PH25424A (it) 1991-07-01
SE8801236D0 (sv) 1988-04-05
GB2203149A (en) 1988-10-12
GB8807750D0 (en) 1988-05-05
SE8801236L (sv) 1988-10-17
JPS63258892A (ja) 1988-10-26
AU1415188A (en) 1988-10-06
IL85969A0 (en) 1988-09-30
PT87153B (pt) 1992-07-31
GB2203149B (en) 1991-02-13
NZ224131A (en) 1991-12-23

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TA Fee payment date (situation as of event date), data collected since 19931001

Effective date: 19940328