JP2004507465A - エストロゲン受容体陽性癌腫の治療方法 - Google Patents

エストロゲン受容体陽性癌腫の治療方法 Download PDF

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Publication number
JP2004507465A
JP2004507465A JP2002518948A JP2002518948A JP2004507465A JP 2004507465 A JP2004507465 A JP 2004507465A JP 2002518948 A JP2002518948 A JP 2002518948A JP 2002518948 A JP2002518948 A JP 2002518948A JP 2004507465 A JP2004507465 A JP 2004507465A
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JP
Japan
Prior art keywords
rapamycin
carbon atoms
estrogen
hydroxy
pharmaceutically acceptable
Prior art date
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Withdrawn
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JP2002518948A
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English (en)
Japanese (ja)
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JP2004507465A5 (2
Inventor
イシャン・ジャン
タミー・ミシェル・サドラー
フィリップ・フロスト
リー・マーティン・グリーンバーガー
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Wyeth LLC
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Wyeth LLC
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=22840171&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=JP2004507465(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Wyeth LLC filed Critical Wyeth LLC
Publication of JP2004507465A publication Critical patent/JP2004507465A/ja
Publication of JP2004507465A5 publication Critical patent/JP2004507465A5/ja
Withdrawn legal-status Critical Current

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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/4738Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/4745Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems condensed with ring systems having nitrogen as a ring hetero atom, e.g. phenantrolines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/24Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/32Antioestrogens

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Molecular Biology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
JP2002518948A 2000-08-11 2001-08-06 エストロゲン受容体陽性癌腫の治療方法 Withdrawn JP2004507465A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US22432600P 2000-08-11 2000-08-11
PCT/US2001/024615 WO2002013802A2 (en) 2000-08-11 2001-08-06 Method of treating estrogen receptor positive carcinoma

Publications (2)

Publication Number Publication Date
JP2004507465A true JP2004507465A (ja) 2004-03-11
JP2004507465A5 JP2004507465A5 (2) 2008-09-25

Family

ID=22840171

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2002518948A Withdrawn JP2004507465A (ja) 2000-08-11 2001-08-06 エストロゲン受容体陽性癌腫の治療方法

Country Status (14)

Country Link
US (1) US6511986B2 (2)
EP (1) EP1318837B1 (2)
JP (1) JP2004507465A (2)
CN (1) CN100448487C (2)
AR (1) AR033555A1 (2)
AT (1) ATE278421T1 (2)
AU (1) AU2001283139A1 (2)
CA (1) CA2416976C (2)
DE (1) DE60106281T2 (2)
DK (1) DK1318837T3 (2)
ES (1) ES2228932T3 (2)
MX (1) MXPA03001245A (2)
PT (1) PT1318837E (2)
WO (1) WO2002013802A2 (2)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2022552132A (ja) * 2019-10-01 2022-12-15 サノフイ 新規の置換6,7-ジヒドロ-5h-ベンゾ[7]アンヌレン化合物、その製造方法およびその治療的使用

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Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2022552132A (ja) * 2019-10-01 2022-12-15 サノフイ 新規の置換6,7-ジヒドロ-5h-ベンゾ[7]アンヌレン化合物、その製造方法およびその治療的使用
JP7680438B2 (ja) 2019-10-01 2025-05-20 サノフイ 新規の置換6,7-ジヒドロ-5h-ベンゾ[7]アンヌレン化合物、その製造方法およびその治療的使用

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EP1318837B1 (en) 2004-10-06
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US20020045638A1 (en) 2002-04-18
ES2228932T3 (es) 2005-04-16
CN100448487C (zh) 2009-01-07
MXPA03001245A (es) 2003-05-27
HK1056687A1 (en) 2004-02-27
DE60106281T2 (de) 2005-02-24
US6511986B2 (en) 2003-01-28
CA2416976A1 (en) 2002-02-21
AU2001283139A1 (en) 2002-02-25
DE60106281D1 (de) 2004-11-11
DK1318837T3 (da) 2005-01-10
WO2002013802A3 (en) 2003-03-27
EP1318837A2 (en) 2003-06-18
ATE278421T1 (de) 2004-10-15
PT1318837E (pt) 2004-12-31
CN1446106A (zh) 2003-10-01
WO2002013802A2 (en) 2002-02-21

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