ATE427948T1 - Folat-mimetika und deren folatrezeptorbindende konjugate - Google Patents
Folat-mimetika und deren folatrezeptorbindende konjugateInfo
- Publication number
- ATE427948T1 ATE427948T1 AT02731495T AT02731495T ATE427948T1 AT E427948 T1 ATE427948 T1 AT E427948T1 AT 02731495 T AT02731495 T AT 02731495T AT 02731495 T AT02731495 T AT 02731495T AT E427948 T1 ATE427948 T1 AT E427948T1
- Authority
- AT
- Austria
- Prior art keywords
- folate
- mimetics
- receptor
- binding conjugates
- disclosure relates
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D475/00—Heterocyclic compounds containing pteridine ring systems
- C07D475/02—Heterocyclic compounds containing pteridine ring systems with an oxygen atom directly attached in position 4
- C07D475/04—Heterocyclic compounds containing pteridine ring systems with an oxygen atom directly attached in position 4 with a nitrogen atom directly attached in position 2
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K51/00—Preparations containing radioactive substances for use in therapy or testing in vivo
- A61K51/02—Preparations containing radioactive substances for use in therapy or testing in vivo characterised by the carrier, i.e. characterised by the agent or material covalently linked or complexing the radioactive nucleus
- A61K51/04—Organic compounds
- A61K51/0497—Organic compounds conjugates with a carrier being an organic compounds
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Physics & Mathematics (AREA)
- Optics & Photonics (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
- Peptides Or Proteins (AREA)
- Saccharide Compounds (AREA)
- Medicines Containing Material From Animals Or Micro-Organisms (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US28608201P | 2001-04-24 | 2001-04-24 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE427948T1 true ATE427948T1 (de) | 2009-04-15 |
Family
ID=23096986
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT02731495T ATE427948T1 (de) | 2001-04-24 | 2002-04-24 | Folat-mimetika und deren folatrezeptorbindende konjugate |
Country Status (5)
| Country | Link |
|---|---|
| US (2) | US7875612B2 (de) |
| EP (1) | EP1389209B1 (de) |
| AT (1) | ATE427948T1 (de) |
| DE (1) | DE60231868D1 (de) |
| WO (1) | WO2002085908A1 (de) |
Families Citing this family (97)
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-
2002
- 2002-04-24 AT AT02731495T patent/ATE427948T1/de not_active IP Right Cessation
- 2002-04-24 US US10/475,876 patent/US7875612B2/en not_active Expired - Lifetime
- 2002-04-24 DE DE60231868T patent/DE60231868D1/de not_active Expired - Lifetime
- 2002-04-24 EP EP02731495A patent/EP1389209B1/de not_active Expired - Lifetime
- 2002-04-24 WO PCT/US2002/013045 patent/WO2002085908A1/en not_active Ceased
-
2010
- 2010-05-07 US US12/775,824 patent/US8470822B2/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| US7875612B2 (en) | 2011-01-25 |
| EP1389209B1 (de) | 2009-04-08 |
| US8470822B2 (en) | 2013-06-25 |
| US20040242582A1 (en) | 2004-12-02 |
| EP1389209A1 (de) | 2004-02-18 |
| US20050227985A9 (en) | 2005-10-13 |
| WO2002085908A1 (en) | 2002-10-31 |
| US20110028714A1 (en) | 2011-02-03 |
| DE60231868D1 (de) | 2009-05-20 |
| EP1389209A4 (de) | 2005-04-13 |
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