JP2009503025A5 - - Google Patents

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Publication number
JP2009503025A5
JP2009503025A5 JP2008524509A JP2008524509A JP2009503025A5 JP 2009503025 A5 JP2009503025 A5 JP 2009503025A5 JP 2008524509 A JP2008524509 A JP 2008524509A JP 2008524509 A JP2008524509 A JP 2008524509A JP 2009503025 A5 JP2009503025 A5 JP 2009503025A5
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JP
Japan
Prior art keywords
alkyl
use according
hydrogen
het
halo
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Application number
JP2008524509A
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English (en)
Japanese (ja)
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JP2009503025A (ja
JP5302680B2 (ja
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Application filed filed Critical
Priority claimed from PCT/EP2006/064858 external-priority patent/WO2007014941A2/en
Publication of JP2009503025A publication Critical patent/JP2009503025A/ja
Publication of JP2009503025A5 publication Critical patent/JP2009503025A5/ja
Application granted granted Critical
Publication of JP5302680B2 publication Critical patent/JP5302680B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2008524509A 2005-08-03 2006-07-31 抗バクテリア剤としてのキノリン誘導体 Expired - Fee Related JP5302680B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP05107164 2005-08-03
EP05107164.5 2005-08-03
PCT/EP2006/064858 WO2007014941A2 (en) 2005-08-03 2006-07-31 Quinoline derivatives as antibacterial agents

Publications (3)

Publication Number Publication Date
JP2009503025A JP2009503025A (ja) 2009-01-29
JP2009503025A5 true JP2009503025A5 (2) 2009-09-17
JP5302680B2 JP5302680B2 (ja) 2013-10-02

Family

ID=35744723

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2008524509A Expired - Fee Related JP5302680B2 (ja) 2005-08-03 2006-07-31 抗バクテリア剤としてのキノリン誘導体

Country Status (30)

Country Link
US (1) US8802671B2 (2)
EP (1) EP1912648B1 (2)
JP (1) JP5302680B2 (2)
KR (1) KR101413997B1 (2)
CN (2) CN101277696B8 (2)
AP (1) AP2654A (2)
AR (1) AR054890A1 (2)
AU (1) AU2006274880B2 (2)
BR (1) BRPI0614493B8 (2)
CA (1) CA2615903C (2)
CY (1) CY1114318T1 (2)
DK (1) DK1912648T3 (2)
EA (1) EA014833B1 (2)
ES (1) ES2414956T3 (2)
HR (1) HRP20130540T1 (2)
IL (1) IL189142A0 (2)
JO (1) JO2855B1 (2)
ME (1) ME01616B (2)
MX (1) MX2008001603A (2)
MY (1) MY159560A (2)
NO (1) NO341242B1 (2)
NZ (1) NZ565947A (2)
PL (1) PL1912648T3 (2)
PT (1) PT1912648E (2)
RS (1) RS52808B (2)
SI (1) SI1912648T1 (2)
TW (1) TWI422374B (2)
UA (1) UA95915C2 (2)
WO (1) WO2007014941A2 (2)
ZA (1) ZA200801110B (2)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2004186452A (ja) 2002-12-04 2004-07-02 Renesas Technology Corp 不揮発性半導体記憶装置およびその製造方法
JO2683B1 (en) * 2006-12-06 2013-03-03 جانسين فارماسوتيكا ان. في Quinoline antibacterial derivatives
JO3271B1 (ar) * 2006-12-06 2018-09-16 Janssen Pharmaceutica Nv مشتقات الكوينولين المضادة للجراثيم
CA2869453C (en) 2012-04-27 2021-03-02 Janssen Pharmaceutica Nv Antibacterial quinoline derivatives
KR102110355B1 (ko) 2012-04-27 2020-05-14 얀센 파마슈티카 엔.브이. 항균성 퀴놀린 유도체
US9290476B2 (en) 2012-10-16 2016-03-22 Janssen Pharmaceutica Nv Methylene linked quinolinyl modulators of RORγt
CN104884448A (zh) 2012-10-16 2015-09-02 詹森药业有限公司 Rorγt的杂芳基连接的喹啉基调节剂
CN105073729A (zh) 2012-10-16 2015-11-18 詹森药业有限公司 RORγt的苯基连接的喹啉基调节剂
US10555941B2 (en) 2013-10-15 2020-02-11 Janssen Pharmaceutica Nv Alkyl linked quinolinyl modulators of RORγt
US9403816B2 (en) 2013-10-15 2016-08-02 Janssen Pharmaceutica Nv Phenyl linked quinolinyl modulators of RORγt
US9221804B2 (en) 2013-10-15 2015-12-29 Janssen Pharmaceutica Nv Secondary alcohol quinolinyl modulators of RORγt
BR112016008258A2 (pt) 2013-10-15 2017-10-10 Janssen Pharmaceutica Nv moduladores de ror?t de quinolinila
US9328095B2 (en) 2013-10-15 2016-05-03 Janssen Pharmaceutica Nv Heteroaryl linked quinolinyl modulators of RORgammat
BR112016008215A2 (pt) 2013-10-15 2017-09-26 Janssen Pharmaceutica Nv moduladores de quinolinila ligados por alquila de roryt
US9284308B2 (en) 2013-10-15 2016-03-15 Janssen Pharmaceutica Nv Methylene linked quinolinyl modulators of RORγt
CN109111397B (zh) * 2018-08-28 2021-12-10 广东工业大学 一种喹啉芳香乙烯类衍生物及其制备方法和应用
CN109111396B (zh) * 2018-08-28 2021-09-03 广东工业大学 一种喹啉芳香乙烯衍生物及其制备方法和应用
CN112110907B (zh) * 2020-10-09 2021-12-21 中央民族大学 一种含1,4-二氧六环二聚双噻吩结构的化合物及其制备方法和应用
CN112079825B (zh) * 2020-10-09 2021-12-21 中央民族大学 含1,3-二氧戊环二聚双噻吩结构的化合物及其制备方法和应用

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB807750A (en) 1956-06-15 1959-01-21 Rhone Poulenc Sa Improvements in or relating to piperazine derivatives
GB9317491D0 (en) * 1993-08-23 1993-10-06 Fujisawa Pharmaceutical Co New compound and a process for preparation thereof
US5965572A (en) * 1996-10-28 1999-10-12 The United States Of America As Respresented By The Secretary Of The Army Methods for treating antibiotic-resistant infections
US6103905A (en) * 1997-06-19 2000-08-15 Sepracor, Inc. Quinoline-indole antimicrobial agents, uses and compositions related thereto
AR040336A1 (es) * 2002-06-26 2005-03-30 Glaxo Group Ltd Compuesto de piperidina, uso del mismo para la fabricacion de un medicamento, composicion farmaceutica que lo comprende y procedimiento para preparar dicho compuesto
DK1527050T3 (da) * 2002-07-25 2010-07-19 Janssen Pharmaceutica Nv Quinolin-derivater og deres anvendelse som mycobakterielle inhibitorer
PL360102A3 (en) 2003-05-13 2004-11-15 "ENERGOMAR-NORD" Sp.z o.o. Method for manufacturing highly reactive calcium sorbing agents and facility designed for manufacturing highly reactive calcium sorbing agents
EA011277B1 (ru) 2004-01-23 2009-02-27 Янссен Фармацевтика Н.В. Производные хинолина и их применение в качестве ингибиторов микобактерий
AP2188A (en) 2004-01-23 2010-12-14 Janssen Pharmaceutica Nv Substituted quinolines and their use as mycobacterial inhibitors.
EA011572B9 (ru) * 2004-01-29 2018-01-31 Янссен Фармацевтика Н.В. Производные хинолина для применения в качестве микобактериальных ингибиторов
CA2528849C (en) * 2005-06-08 2014-01-14 Janssen Pharmaceutica N.V. Quinoline derivatives as antibacterial agents
US20070018948A1 (en) 2005-07-22 2007-01-25 Elaine Chen Apparatus for stabilizing an electronic device during data input and device control

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