JP2015509104A - 神経変性障害を治療するためのジアジリジン - Google Patents

神経変性障害を治療するためのジアジリジン Download PDF

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JP2015509104A
JP2015509104A JP2014553849A JP2014553849A JP2015509104A JP 2015509104 A JP2015509104 A JP 2015509104A JP 2014553849 A JP2014553849 A JP 2014553849A JP 2014553849 A JP2014553849 A JP 2014553849A JP 2015509104 A JP2015509104 A JP 2015509104A
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disorder
syndrome
disease
psychosis
sleep
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JP2015509104A5 (fr
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エヌ． マクホバ ニナ
エヌ． マクホバ ニナ
ワイ． ペトウクホバ ベラ
ワイ． ペトウクホバ ベラ
ブイ． シェブトソブ アレクアンドル
ブイ． シェブトソブ アレクアンドル
ブイ． ノバコブスクイイ ブライドイミル
ブイ． ノバコブスクイイ ブライドイミル
ブラドイミロビク クズネトソブ ブライドイミル
ブラドイミロビク クズネトソブ ブライドイミル
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D229/00—Heterocyclic compounds containing rings of less than five members having two nitrogen atoms as the only ring hetero atoms
    • C07D229/02—Heterocyclic compounds containing rings of less than five members having two nitrogen atoms as the only ring hetero atoms containing three-membered rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/396—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having three-membered rings, e.g. aziridine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
    • A61K31/4188—1,3-Diazoles condensed with other heterocyclic ring systems, e.g. biotin, sorbinil
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4192—1,2,3-Triazoles
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    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
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    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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    • C07D491/10—Spiro-condensed systems
    • C07D491/107—Spiro-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring
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  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
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  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Chemical Kinetics & Catalysis (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
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  • Epidemiology (AREA)
  • Psychiatry (AREA)
  • Addiction (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Psychology (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Pain & Pain Management (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Hospice & Palliative Care (AREA)
  • Ophthalmology & Optometry (AREA)
  • Anesthesiology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
JP2014553849A 2012-01-26 2013-01-26 神経変性障害を治療するためのジアジリジン Pending JP2015509104A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201261591176P 2012-01-26 2012-01-26
US61/591,176 2012-01-26
PCT/IB2013/050681 WO2013111117A2 (fr) 2012-01-26 2013-01-26 Agents pour le traitement de troubles mentaux

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Publication Number Publication Date
JP2015509104A true JP2015509104A (ja) 2015-03-26
JP2015509104A5 JP2015509104A5 (fr) 2016-03-17

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JP2014553849A Pending JP2015509104A (ja) 2012-01-26 2013-01-26 神経変性障害を治療するためのジアジリジン

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EP (1) EP2807150A2 (fr)
JP (1) JP2015509104A (fr)
WO (1) WO2013111117A2 (fr)

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* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2012042502A1 (fr) 2010-09-29 2012-04-05 Pharmdiscovery Llp Dérivés de diazaridine utiles dans le traitement des troubles mentaux

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WO2013111117A3 (fr) 2013-10-31
EP2807150A2 (fr) 2014-12-03
WO2013111117A2 (fr) 2013-08-01

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