JP2017522300A5 - - Google Patents
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- Publication number
- JP2017522300A5 JP2017522300A5 JP2016575499A JP2016575499A JP2017522300A5 JP 2017522300 A5 JP2017522300 A5 JP 2017522300A5 JP 2016575499 A JP2016575499 A JP 2016575499A JP 2016575499 A JP2016575499 A JP 2016575499A JP 2017522300 A5 JP2017522300 A5 JP 2017522300A5
- Authority
- JP
- Japan
- Prior art keywords
- dihydro
- benzoxazin
- oxo
- carbonyl
- acetamide
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201462018790P | 2014-06-30 | 2014-06-30 | |
| US62/018,790 | 2014-06-30 | ||
| PCT/GB2015/051860 WO2016001631A1 (en) | 2014-06-30 | 2015-06-26 | Benzoxazinone amides as mineralocorticoid receptor modulators |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2017522300A JP2017522300A (ja) | 2017-08-10 |
| JP2017522300A5 true JP2017522300A5 (2) | 2018-07-19 |
| JP6368383B2 JP6368383B2 (ja) | 2018-08-01 |
Family
ID=53539739
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2016575499A Active JP6368383B2 (ja) | 2014-06-30 | 2015-06-26 | 鉱質コルチコイド受容体修飾因子としてのベンゾオキサジノンアミド |
Country Status (26)
| Country | Link |
|---|---|
| US (2) | US10017502B2 (2) |
| EP (1) | EP3160948B1 (2) |
| JP (1) | JP6368383B2 (2) |
| KR (1) | KR102012222B1 (2) |
| CN (1) | CN106536491B (2) |
| AR (1) | AR101036A1 (2) |
| AU (1) | AU2015282450C1 (2) |
| CA (1) | CA2953655C (2) |
| CY (1) | CY1121596T1 (2) |
| DK (1) | DK3160948T3 (2) |
| EA (1) | EA029518B1 (2) |
| ES (1) | ES2707726T3 (2) |
| HR (1) | HRP20190147T1 (2) |
| HU (1) | HUE042370T2 (2) |
| LT (1) | LT3160948T (2) |
| ME (1) | ME03316B (2) |
| MX (1) | MX367404B (2) |
| PL (1) | PL3160948T3 (2) |
| PT (1) | PT3160948T (2) |
| RS (1) | RS58274B1 (2) |
| SI (1) | SI3160948T1 (2) |
| SM (1) | SMT201900039T1 (2) |
| TR (1) | TR201900659T4 (2) |
| TW (1) | TWI677498B (2) |
| UY (1) | UY36195A (2) |
| WO (1) | WO2016001631A1 (2) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MX367404B (es) * | 2014-06-30 | 2019-08-20 | Astrazeneca Ab | Amidas de benzoxazinona como moduladores del receptor de mineralocorticoides. |
| BR112021000139A2 (pt) | 2018-07-19 | 2021-04-06 | Astrazeneca Ab | Métodos de tratamento da hfpef empregando dapagliflozina e composições compreendendo a mesma |
| CN112107568B (zh) * | 2019-06-19 | 2022-03-25 | 北京龙嘉博创医药科技有限公司 | 二芳基酰胺类化合物及其应用 |
| WO2021037400A1 (en) * | 2019-08-30 | 2021-03-04 | Astrazeneca Ab | Methods of treating heart failure with reduced ejection fraction with dapagliflozin |
| TW202220672A (zh) | 2020-07-27 | 2022-06-01 | 瑞典商阿斯特捷利康公司 | 用達格列淨治療慢性腎臟病之方法 |
| AU2021202643B2 (en) | 2020-07-27 | 2023-02-02 | Astrazeneca Ab | Methods of treating chronic kidney disease with dapagliflozin |
| CA3222502A1 (en) | 2021-06-15 | 2022-12-22 | Lingyun Wu | Benzoxazinone derivatives |
| TW202409023A (zh) | 2022-07-14 | 2024-03-01 | 美商富曼西公司 | 除草苯并𠯤 |
| CR20250112A (es) | 2022-09-01 | 2025-08-18 | Aztrazeneca Ab | Combinación de ihnibidores de sglt2 y moduladores del receptor mineralcorticoide para usar en el tratamiento de enfermedades cardiorrenales |
| CN120344508A (zh) * | 2022-12-15 | 2025-07-18 | 正大天晴药业集团股份有限公司 | 苯并恶嗪酮类化合物的结晶及其制备 |
| WO2025111184A1 (en) | 2023-11-21 | 2025-05-30 | Fmc Corporation | Substituted tetrahydroquinoline and tetrahydroquinoxaline herbicides |
Family Cites Families (23)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2004528335A (ja) * | 2001-04-23 | 2004-09-16 | アストラゼネカ アクチボラグ | 血管新生の治療に使用のベンゾオキサジノン誘導体 |
| AU2003303231A1 (en) * | 2002-12-20 | 2004-07-14 | Warner-Lambert Company Llc | Benzoxazines and derivatives thereof as inhibitors of pi3ks |
| BRPI0513119A (pt) * | 2004-07-14 | 2008-04-29 | Ligand Pharm Inc | compostos e métodos modulares de receptores intracelulares |
| RU2007107177A (ru) * | 2004-07-28 | 2008-09-10 | Айрм Ллк (Bm) | Соединения и композиции, как модуляторы ядерных рецепторов стероидных гормонов |
| CA2635541A1 (en) | 2005-12-28 | 2007-07-12 | Takeda Pharmaceutical Company Limited | Fused heterocyclic compounds and their use as mineralocorticoid receptor ligands |
| TWI385161B (zh) | 2006-02-02 | 2013-02-11 | Mitsubishi Tanabe Pharma Corp | 含氮雜雙環化合物 |
| SI2089367T1 (sl) | 2006-10-31 | 2012-02-29 | Pfizer Prod Inc | Spojine pirazolina kot antagonisti mineralokortikoidnih receptorjev |
| DE102007009494A1 (de) | 2007-02-27 | 2008-08-28 | Bayer Healthcare Ag | Substituierte 4-Aryl-1, 4-dihydro-1,6-naphthyridinamide und ihre Verwendung |
| WO2008118319A2 (en) | 2007-03-23 | 2008-10-02 | Merck & Co., Inc. | Mineralocorticoid receptor modulators |
| CN101679243B (zh) | 2007-04-09 | 2012-09-26 | 第一三共株式会社 | 吡咯衍生物的阻转异构体 |
| US8258131B2 (en) | 2007-08-01 | 2012-09-04 | Mitsubishi Tanabe Pharma Corporation | Fused bicyclic compound |
| JP5173653B2 (ja) * | 2007-08-01 | 2013-04-03 | 田辺三菱製薬株式会社 | 医薬組成物 |
| TWI431010B (zh) | 2007-12-19 | 2014-03-21 | Lilly Co Eli | 礦皮質素受體拮抗劑及使用方法 |
| WO2009154557A1 (en) * | 2008-06-18 | 2009-12-23 | Astrazeneca Ab | Benzoxazinone derivatives acting as beta2-adrenoreceptor agonist for the treatment of respiratory disorders |
| US20100094000A1 (en) | 2008-09-03 | 2010-04-15 | Takeda Pharmaceutical Company Limited | Pyrazole compounds |
| WO2010098286A1 (ja) | 2009-02-25 | 2010-09-02 | 第一三共株式会社 | ミネラルコルチコイド受容体拮抗薬を含有する医薬 |
| AU2010222902B2 (en) | 2009-03-12 | 2013-04-18 | Eli Lilly And Company | Mineralocorticoid receptor antagonist and methods of use |
| US20120022058A1 (en) | 2009-04-10 | 2012-01-26 | Pfizer Inc. | 4,5-dihydro-1h-pyrazole compounds and their pharmaceutical uses |
| CN102906495B (zh) | 2010-05-11 | 2016-08-24 | 皇家飞利浦电子股份有限公司 | 照明模块 |
| WO2011141848A1 (en) | 2010-05-11 | 2011-11-17 | Pfizer Inc. | Morpholine compounds as mineralocorticoid receptor antagonists |
| TW201216957A (en) | 2010-07-13 | 2012-05-01 | Dainippon Sumitomo Pharma Co | Biarylamide derivative or a pharmaceutically acceptable salt thereof |
| EP2638012A1 (en) | 2010-11-10 | 2013-09-18 | Boehringer Ingelheim International GmbH | Pyridyl ureas as mineralocorticoid receptor antagonists |
| MX367404B (es) * | 2014-06-30 | 2019-08-20 | Astrazeneca Ab | Amidas de benzoxazinona como moduladores del receptor de mineralocorticoides. |
-
2015
- 2015-06-26 MX MX2017000183A patent/MX367404B/es active IP Right Grant
- 2015-06-26 EP EP15736015.7A patent/EP3160948B1/en active Active
- 2015-06-26 CA CA2953655A patent/CA2953655C/en active Active
- 2015-06-26 WO PCT/GB2015/051860 patent/WO2016001631A1/en not_active Ceased
- 2015-06-26 SM SM20190039T patent/SMT201900039T1/it unknown
- 2015-06-26 US US15/320,379 patent/US10017502B2/en active Active
- 2015-06-26 PL PL15736015T patent/PL3160948T3/pl unknown
- 2015-06-26 RS RS20190085A patent/RS58274B1/sr unknown
- 2015-06-26 AU AU2015282450A patent/AU2015282450C1/en active Active
- 2015-06-26 KR KR1020177002518A patent/KR102012222B1/ko active Active
- 2015-06-26 ME MEP-2019-19A patent/ME03316B/me unknown
- 2015-06-26 EA EA201790046A patent/EA029518B1/ru not_active IP Right Cessation
- 2015-06-26 DK DK15736015.7T patent/DK3160948T3/en active
- 2015-06-26 TR TR2019/00659T patent/TR201900659T4/tr unknown
- 2015-06-26 PT PT15736015T patent/PT3160948T/pt unknown
- 2015-06-26 JP JP2016575499A patent/JP6368383B2/ja active Active
- 2015-06-26 HR HRP20190147TT patent/HRP20190147T1/hr unknown
- 2015-06-26 HU HUE15736015A patent/HUE042370T2/hu unknown
- 2015-06-26 UY UY0001036195A patent/UY36195A/es not_active Application Discontinuation
- 2015-06-26 ES ES15736015T patent/ES2707726T3/es active Active
- 2015-06-26 SI SI201530572T patent/SI3160948T1/sl unknown
- 2015-06-26 LT LTEP15736015.7T patent/LT3160948T/lt unknown
- 2015-06-26 CN CN201580035032.8A patent/CN106536491B/zh active Active
- 2015-06-29 TW TW104120998A patent/TWI677498B/zh active
- 2015-06-29 US US14/753,239 patent/US9394291B2/en active Active
- 2015-06-30 AR ARP150102098A patent/AR101036A1/es active IP Right Grant
-
2019
- 2019-01-24 CY CY20191100097T patent/CY1121596T1/el unknown
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