JP2017530193A5 - - Google Patents
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- Publication number
- JP2017530193A5 JP2017530193A5 JP2017535616A JP2017535616A JP2017530193A5 JP 2017530193 A5 JP2017530193 A5 JP 2017530193A5 JP 2017535616 A JP2017535616 A JP 2017535616A JP 2017535616 A JP2017535616 A JP 2017535616A JP 2017530193 A5 JP2017530193 A5 JP 2017530193A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- heteroaryl
- heterocycloalkyl
- aryl
- cycloalkyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- RXYPXQSKLGGKOL-UHFFFAOYSA-N CN1CCN(C)CC1 Chemical compound CN1CCN(C)CC1 RXYPXQSKLGGKOL-UHFFFAOYSA-N 0.000 description 2
- TZYFCEGYHDNOFE-UHFFFAOYSA-N CC(CC1N(C)CCCC1)[n]1nncc1 Chemical compound CC(CC1N(C)CCCC1)[n]1nncc1 TZYFCEGYHDNOFE-UHFFFAOYSA-N 0.000 description 1
- PAMIQIKDUOTOBW-UHFFFAOYSA-N CN1CCCCC1 Chemical compound CN1CCCCC1 PAMIQIKDUOTOBW-UHFFFAOYSA-N 0.000 description 1
- JWAWEQBUZOGIBZ-UHFFFAOYSA-N C[n]1nncc1 Chemical compound C[n]1nncc1 JWAWEQBUZOGIBZ-UHFFFAOYSA-N 0.000 description 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201462053389P | 2014-09-22 | 2014-09-22 | |
| US62/053,389 | 2014-09-22 | ||
| PCT/US2015/051143 WO2016048861A2 (en) | 2014-09-22 | 2015-09-21 | Heterocyclic compounds and use thereof |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2017530193A JP2017530193A (ja) | 2017-10-12 |
| JP2017530193A5 true JP2017530193A5 (2) | 2018-11-01 |
| JP6615207B2 JP6615207B2 (ja) | 2019-12-04 |
Family
ID=55525127
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2017535616A Active JP6615207B2 (ja) | 2014-09-22 | 2015-09-21 | 複素環式化合物及びその使用 |
Country Status (12)
| Country | Link |
|---|---|
| US (2) | US9862703B2 (2) |
| EP (1) | EP3197885B1 (2) |
| JP (1) | JP6615207B2 (2) |
| KR (1) | KR102509431B1 (2) |
| CN (1) | CN107207465B (2) |
| AU (1) | AU2015321654B2 (2) |
| BR (1) | BR112017005713B1 (2) |
| CA (1) | CA2962329C (2) |
| ES (1) | ES2849998T3 (2) |
| RU (1) | RU2704008C2 (2) |
| TW (1) | TWI598348B (2) |
| WO (1) | WO2016048861A2 (2) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| RU2756055C2 (ru) * | 2017-01-10 | 2021-09-24 | Нэшнл Хелт Рисерч Инститьютс | Гетероциклические соединения и их применение |
| KR20240151869A (ko) * | 2017-09-08 | 2024-10-18 | 더 보드 어브 트러스티스 어브 더 리랜드 스탠포드 주니어 유니버시티 | Enpp1 저해제 및 암의 치료용의 이의 용도 |
| EP3842435A4 (en) | 2018-09-20 | 2022-05-11 | Hanmi Pharm. Co., Ltd. | NOVEL SULFONAMIDE DERIVATIVE WITH FUSED PYRIMIDINE FRAMEWORK WITH INHIBITING ACTIVITY ON EPIDERMAL GROWTH FACTOR RECEPTOR MUTATIONS |
| JP7777332B2 (ja) * | 2019-02-01 | 2025-11-28 | ザ ボード オブ トラスティーズ オブ ザ レランド スタンフォード ジュニア ユニバーシティー | 免疫応答をモジュレートするｅｎｐｐ１阻害剤および方法 |
| CN111138417B (zh) * | 2019-12-18 | 2021-03-23 | 浙江工业大学 | 一种三氮唑修饰的5-氟-2,4-嘧啶二胺类化合物及其应用 |
| CA3228210A1 (en) * | 2021-08-02 | 2023-02-09 | National Health Research Institutes | Pyrimidine compounds and use thereof |
| IL320644A (en) * | 2022-11-07 | 2025-07-01 | Univ Kyoto | Quinazoline derivatives |
| UY40657A (es) | 2023-03-01 | 2024-09-13 | Novartis Ag | Derivados de hidroquinazolina para el tratamiento de una enfermedad o un trastorno |
Family Cites Families (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS4936700A (2) * | 1972-08-16 | 1974-04-05 | ||
| ES2150941T3 (es) * | 1992-04-03 | 2000-12-16 | Upjohn Co | Aminas biciclicas-heterociclicas eficaces farmaceuticamente. |
| US6156758A (en) * | 1999-09-08 | 2000-12-05 | Isis Pharmaceuticals, Inc. | Antibacterial quinazoline compounds |
| EP2043651A2 (en) * | 2006-07-05 | 2009-04-08 | Exelixis, Inc. | Methods of using igf1r and abl kinase modulators |
| BRPI0909375A2 (pt) * | 2008-03-28 | 2015-08-04 | Altiris Therapeutics | Moduladores de receptores de quimiocinas |
| CN102046609B (zh) * | 2008-03-31 | 2014-05-14 | 全药工业株式会社 | 具有细胞保护效果的嘧啶衍生物及其应用 |
| DK2268635T3 (en) | 2008-04-21 | 2015-09-14 | Taigen Biotechnology Co Ltd | Heterocyclic Compounds |
| WO2010046780A2 (en) | 2008-10-22 | 2010-04-29 | Institut Pasteur Korea | Anti viral compounds |
| GB201015411D0 (en) | 2010-09-15 | 2010-10-27 | Univ Leuven Kath | Anti-cancer activity of novel bicyclic heterocycles |
| BR112014007310A2 (pt) | 2011-09-27 | 2017-04-04 | Novartis Ag | 3-pirimidin-4-il-oxazolidin-2-onas como inibidores de idh mutante |
| WO2013155123A1 (en) | 2012-04-10 | 2013-10-17 | Georgia State University Research Foundation, Inc. | Compositions and methods for treating otitis media and other conditions with inhibitors of cyld |
| DK2906563T3 (en) | 2012-10-10 | 2018-06-06 | Janssen Sciences Ireland Uc | PYRROLO [3,2-D] PYRIMIDINE DERIVATIVES FOR TREATING VIRUS INFECTIONS AND OTHER DISEASES |
| US20150259649A1 (en) * | 2012-11-08 | 2015-09-17 | Emory University | Cellular compositions used to restore stem cell or progenitor cell function and methods related thereto |
-
2015
- 2015-09-21 ES ES15844487T patent/ES2849998T3/es active Active
- 2015-09-21 JP JP2017535616A patent/JP6615207B2/ja active Active
- 2015-09-21 BR BR112017005713-1A patent/BR112017005713B1/pt active IP Right Grant
- 2015-09-21 US US14/860,033 patent/US9862703B2/en active Active
- 2015-09-21 AU AU2015321654A patent/AU2015321654B2/en active Active
- 2015-09-21 RU RU2017109355A patent/RU2704008C2/ru active
- 2015-09-21 EP EP15844487.7A patent/EP3197885B1/en active Active
- 2015-09-21 CN CN201580050829.5A patent/CN107207465B/zh active Active
- 2015-09-21 WO PCT/US2015/051143 patent/WO2016048861A2/en not_active Ceased
- 2015-09-21 CA CA2962329A patent/CA2962329C/en active Active
- 2015-09-21 KR KR1020177010762A patent/KR102509431B1/ko active Active
- 2015-09-22 TW TW104131241A patent/TWI598348B/zh active
-
2017
- 2017-09-22 US US15/712,978 patent/US9926298B2/en active Active
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