JP4820094B2 - ヒスタミン−３受容体リガンドとしての２環式置換アミン - Google Patents

ヒスタミン−３受容体リガンドとしての２環式置換アミン Download PDF

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JP4820094B2
JP4820094B2 JP2004551799A JP2004551799A JP4820094B2 JP 4820094 B2 JP4820094 B2 JP 4820094B2 JP 2004551799 A JP2004551799 A JP 2004551799A JP 2004551799 A JP2004551799 A JP 2004551799A JP 4820094 B2 JP4820094 B2 JP 4820094B2
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ethyl
methyl
pyrrolidinyl
formula
naphthalen
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JP2004551799A
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JP2006514926A (ja
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アルテンバツク，ロバート・ジエイ
ブラツク，ローレンス・エイ
チヤン，ソウ−ジエン
コワート，マーロン・デイー
フアギー，ラミン
グフエサー，グレゴリー・エイ
クー，イー−イン
リウ，ホアチン
ルーキン，キリル・エイ
ナーセシアン，ダイアナ・エル
プ，ユ−ミン
シヤルマ，パダム・エヌ
ベンナニ，ユセフ・エル
カーテイス，マイケル・ピー
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Abbott Laboratories
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Abbott Laboratories
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Priority claimed from US10/292,422 external-priority patent/US20040092521A1/en
Priority claimed from US10/689,735 external-priority patent/US7153889B2/en
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Publication of JP2006514926A publication Critical patent/JP2006514926A/ja
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US20040224952A1 (en) * 2003-05-07 2004-11-11 Cowart Marlon D. Fused bicyclic-substituted amines as histamine-3 receptor ligands
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US20050256118A1 (en) * 2004-05-12 2005-11-17 Altenbach Robert J Bicyclic-substituted amines having cyclic-substituted monocyclic substituents
US7205316B2 (en) 2004-05-12 2007-04-17 Abbott Laboratories Tri- and bi-cyclic heteroaryl histamine-3 receptor ligands
US20050256309A1 (en) * 2004-05-12 2005-11-17 Altenbach Robert J Tri-and bi-cyclic heteroaryl histamine-3 receptor ligands
US7098222B2 (en) 2004-05-12 2006-08-29 Abbott Laboratories Bicyclic-substituted amines having cyclic-substituted monocyclic substituents
CA2566526C (en) * 2004-06-02 2012-10-23 F. Hoffmann-La Roche Ag Naphthaline derivatives useful as histamine-3-receptor ligands
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