JP5669582B2 - グルカゴンアンタゴニスト - Google Patents

グルカゴンアンタゴニスト Download PDF

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Publication number
JP5669582B2
JP5669582B2 JP2010532154A JP2010532154A JP5669582B2 JP 5669582 B2 JP5669582 B2 JP 5669582B2 JP 2010532154 A JP2010532154 A JP 2010532154A JP 2010532154 A JP2010532154 A JP 2010532154A JP 5669582 B2 JP5669582 B2 JP 5669582B2
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JP
Japan
Prior art keywords
seq
amino acid
glucagon
acid
group
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Expired - Fee Related
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JP2010532154A
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English (en)
Japanese (ja)
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JP2011502155A5 (es
JP2011502155A (ja
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ディマルキ,リチャード,ディー.
ヤン,ビン
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Indiana University Research and Technology Corp
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Indiana University Research and Technology Corp
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Publication of JP2011502155A5 publication Critical patent/JP2011502155A5/ja
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K14/00Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/575Hormones
    • C07K14/605Glucagons
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Obesity (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Hematology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Toxicology (AREA)
  • Genetics & Genomics (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Zoology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Emergency Medicine (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicinal Preparation (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
JP2010532154A 2007-10-30 2008-10-23 グルカゴンアンタゴニスト Expired - Fee Related JP5669582B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US98378307P 2007-10-30 2007-10-30
US60/983,783 2007-10-30
PCT/US2008/080973 WO2009058662A2 (en) 2007-10-30 2008-10-23 Glucagon antagonists

Publications (3)

Publication Number Publication Date
JP2011502155A JP2011502155A (ja) 2011-01-20
JP2011502155A5 JP2011502155A5 (es) 2011-12-15
JP5669582B2 true JP5669582B2 (ja) 2015-02-12

Family

ID=40591715

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2010532154A Expired - Fee Related JP5669582B2 (ja) 2007-10-30 2008-10-23 グルカゴンアンタゴニスト

Country Status (12)

Country Link
US (1) US8981047B2 (es)
EP (1) EP2217701B9 (es)
JP (1) JP5669582B2 (es)
AR (1) AR069110A1 (es)
AU (1) AU2008318986B2 (es)
CA (1) CA2707861A1 (es)
CL (1) CL2008003222A1 (es)
ES (1) ES2509883T3 (es)
MX (1) MX2010004297A (es)
PE (1) PE20091393A1 (es)
TW (1) TW200920404A (es)
WO (1) WO2009058662A2 (es)

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US8981047B2 (en) 2015-03-17
US20120122783A1 (en) 2012-05-17
HK1143994A1 (en) 2011-01-21
CA2707861A1 (en) 2009-05-07
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EP2217701B9 (en) 2015-02-18
AU2008318986A1 (en) 2009-05-07
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TW200920404A (en) 2009-05-16
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