JPS53127491A - 33*22aminoethylthio**66ethyll77oxoo 11azabicyclo*3*2*0*heptaa22enee22 carboxylate - Google Patents

33*22aminoethylthio**66ethyll77oxoo 11azabicyclo*3*2*0*heptaa22enee22 carboxylate

Info

Publication number
JPS53127491A
JPS53127491A JP4045678A JP4045678A JPS53127491A JP S53127491 A JPS53127491 A JP S53127491A JP 4045678 A JP4045678 A JP 4045678A JP 4045678 A JP4045678 A JP 4045678A JP S53127491 A JPS53127491 A JP S53127491A
Authority
JP
Japan
Prior art keywords
carboxylate
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP4045678A
Other languages
English (en)
Japanese (ja)
Inventor
Daburiyu Ratokurifu Ronarudo
Jiee Rasubuinkuru Rinda
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Merck and Co Inc
Original Assignee
Merck and Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck and Co Inc filed Critical Merck and Co Inc
Publication of JPS53127491A publication Critical patent/JPS53127491A/ja
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D477/00—Heterocyclic compounds containing 1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbapenicillins, thienamycins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulphur-containing hetero ring
    • C07D477/10—Heterocyclic compounds containing 1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbapenicillins, thienamycins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulphur-containing hetero ring with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 4, and with a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • C07D477/12—Heterocyclic compounds containing 1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbapenicillins, thienamycins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulphur-containing hetero ring with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 4, and with a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2 with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, attached in position 6
    • C07D477/16—Heterocyclic compounds containing 1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbapenicillins, thienamycins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulphur-containing hetero ring with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 4, and with a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2 with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, attached in position 6 with hetero atoms or carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 3
    • C07D477/20—Sulfur atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
JP4045678A 1977-04-08 1978-04-07 33*22aminoethylthio**66ethyll77oxoo 11azabicyclo*3*2*0*heptaa22enee22 carboxylate Pending JPS53127491A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US78581177A 1977-04-08 1977-04-08
US86123077A 1977-12-16 1977-12-16

Publications (1)

Publication Number Publication Date
JPS53127491A true JPS53127491A (en) 1978-11-07

Family

ID=27120448

Family Applications (1)

Application Number Title Priority Date Filing Date
JP4045678A Pending JPS53127491A (en) 1977-04-08 1978-04-07 33*22aminoethylthio**66ethyll77oxoo 11azabicyclo*3*2*0*heptaa22enee22 carboxylate

Country Status (11)

Country Link
JP (1) JPS53127491A (fr)
CH (1) CH640236A5 (fr)
DE (1) DE2815157A1 (fr)
DK (1) DK123578A (fr)
FR (1) FR2386545A1 (fr)
GB (1) GB1595267A (fr)
IE (1) IE47043B1 (fr)
IT (1) IT1102456B (fr)
LU (1) LU79403A1 (fr)
NL (1) NL7802826A (fr)
SE (1) SE7803173L (fr)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5473788A (en) * 1977-11-17 1979-06-13 Sanraku Inc Antibiotic n-desacetyl ps-5
JPS5572191A (en) * 1978-11-22 1980-05-30 Sanraku Inc Antibiotic n-desacetyl ps-5

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GR62185B (en) * 1977-03-31 1979-03-02 Panlabs Inc Preparation process of an antibiotic ps-5 and its derivatives with inhibitory activity of b-lactamase
EP0005349A1 (fr) * 1978-05-06 1979-11-14 Beecham Group Plc Alkylcarbapénèmes, leur préparation, compositions pharmaceutiques les contenant et les intermédiaires
JPS55136282A (en) * 1979-04-06 1980-10-23 Shionogi & Co Ltd Novel antibiotic pa-31088-4
US4235922A (en) * 1979-06-15 1980-11-25 Merck & Co., Inc. 3-(2-Aminoethylthio)-6-ethyl-7-oxo-1-azabicyclo [3.2.0]hept-2-ene-2-carboxylic acid
DE3070269D1 (en) * 1979-08-10 1985-04-18 Beecham Group Plc Beta-lactam antibiotics, their preparation, pharmaceutical compositions containing them and their preparation
JPS5683489A (en) * 1979-12-12 1981-07-08 Shionogi & Co Ltd New antibiotic pa-39504-x1 and it preparation
JPS5764693A (en) * 1980-10-07 1982-04-19 Kowa Co Novel carbapenem compound and its preparation

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3950357A (en) * 1974-11-25 1976-04-13 Merck & Co., Inc. Antibiotics

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5473788A (en) * 1977-11-17 1979-06-13 Sanraku Inc Antibiotic n-desacetyl ps-5
JPS5572191A (en) * 1978-11-22 1980-05-30 Sanraku Inc Antibiotic n-desacetyl ps-5

Also Published As

Publication number Publication date
DE2815157A1 (de) 1978-10-19
IT1102456B (it) 1985-10-07
DK123578A (da) 1978-10-09
NL7802826A (nl) 1978-10-10
GB1595267A (en) 1981-08-12
IE780631L (en) 1978-10-08
CH640236A5 (en) 1983-12-30
SE7803173L (sv) 1978-10-09
IE47043B1 (en) 1983-12-14
IT7848747A0 (it) 1978-04-05
FR2386545B1 (fr) 1980-08-01
FR2386545A1 (fr) 1978-11-03
LU79403A1 (fr) 1978-11-27

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