JPS552623A - Spiro compound and its preparation - Google Patents
Spiro compound and its preparationInfo
- Publication number
- JPS552623A JPS552623A JP7470078A JP7470078A JPS552623A JP S552623 A JPS552623 A JP S552623A JP 7470078 A JP7470078 A JP 7470078A JP 7470078 A JP7470078 A JP 7470078A JP S552623 A JPS552623 A JP S552623A
- Authority
- JP
- Japan
- Prior art keywords
- furan
- substituted
- compound
- preparation
- spiro compound
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
- 150000003413 spiro compounds Chemical class 0.000 title abstract 2
- UHOVQNZJYSORNB-UHFFFAOYSA-N Benzene Chemical compound C1=CC=CC=C1 UHOVQNZJYSORNB-UHFFFAOYSA-N 0.000 abstract 3
- FAPWRFPIFSIZLT-UHFFFAOYSA-M Sodium chloride Chemical compound [Na+].[Cl-] FAPWRFPIFSIZLT-UHFFFAOYSA-M 0.000 abstract 2
- 125000005605 benzo group Chemical group 0.000 abstract 2
- HTSGKJQDMSTCGS-UHFFFAOYSA-N 1,4-bis(4-chlorophenyl)-2-(4-methylphenyl)sulfonylbutane-1,4-dione Chemical compound C1=CC(C)=CC=C1S(=O)(=O)C(C(=O)C=1C=CC(Cl)=CC=1)CC(=O)C1=CC=C(Cl)C=C1 HTSGKJQDMSTCGS-UHFFFAOYSA-N 0.000 abstract 1
- 229940035676 analgesics Drugs 0.000 abstract 1
- 239000000730 antalgic agent Substances 0.000 abstract 1
- 230000001741 anti-phlogistic effect Effects 0.000 abstract 1
- -1 antiphlogistics Substances 0.000 abstract 1
- 239000003699 antiulcer agent Substances 0.000 abstract 1
- 239000003054 catalyst Substances 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 229940079593 drug Drugs 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
- 239000000543 intermediate Substances 0.000 abstract 1
- 239000000463 material Substances 0.000 abstract 1
- 229910001507 metal halide Inorganic materials 0.000 abstract 1
- 150000005309 metal halides Chemical class 0.000 abstract 1
- 125000001624 naphthyl group Chemical group 0.000 abstract 1
- 125000002924 primary amino group Chemical group [H]N([H])* 0.000 abstract 1
- 239000011780 sodium chloride Substances 0.000 abstract 1
- YLQBMQCUIZJEEH-UHFFFAOYSA-N tetrahydrofuran Natural products C=1C=COC=1 YLQBMQCUIZJEEH-UHFFFAOYSA-N 0.000 abstract 1
Landscapes
- Furan Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
NEW MATERIAL:A spiro compound of formula I [ring A is benzene or naphthalene ring which is substituted with (substituted) OH, acyl sulfamoyl, or (substituted) amino]
EXAMPLE: 5-Benzyloxyspiro [benzo[b]furan-2(3H),1'-cyclopropan]-3-one.
USE: Anti-ulcer agent. Drugs such as antiphlogistics, analgesics, etc., or their intermediates.
PROCESS: The objective compound I is prepared by the decarbonation reaction of a compound II [e.g. 5-benzyloxy-4',5'-dihydrospiro[benzo[b]furan-2(3H),3'(2'H)- furan]-2',3-dione] pref. in the presence of a catalyst such as metal halide, etc., e.g. NaCl, etc.
COPYRIGHT: (C)1980,JPO&Japio
Priority Applications (19)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP7470078A JPS552623A (en) | 1978-06-19 | 1978-06-19 | Spiro compound and its preparation |
| GR57881A GR68525B (en) | 1978-06-19 | 1978-12-14 | |
| HU78TA1504A HU179601B (en) | 1977-12-27 | 1978-12-21 | Process for producing spirobenzofuranone derivatives |
| DK574078A DK149891C (en) | 1977-12-27 | 1978-12-21 | METHOD OF ANALOGUE FOR THE PREPARATION OF SPIROBENZOFURANON COMPOUNDS OR SALTS THEREOF WITH INORGANIC OR ORGANIC ACIDS OR ALKALIMETALS |
| CA318,527A CA1113467A (en) | 1977-12-27 | 1978-12-22 | Spirobenzofuranone compounds |
| AU42870/78A AU521851B2 (en) | 1977-12-07 | 1978-12-22 | Spirodenzofuranone compounds |
| NO78784367A NO151155C (en) | 1977-12-27 | 1978-12-22 | ANALOGY PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY EFFECTIVE SPIROBENZOFURANON COMPOUNDS |
| ES476330A ES476330A1 (en) | 1977-12-27 | 1978-12-26 | Spirobenzofuranone compounds, processes for their preparation and their use as medicines. |
| SU782700556A SU1044225A3 (en) | 1977-12-27 | 1978-12-26 | Process for preparing spirobenzofuran compounds |
| EP78300912A EP0003084B1 (en) | 1977-12-27 | 1978-12-27 | Spirobenzofuranone compounds, processes for their preparation and their use as medicines |
| AT0928478A AT372954B (en) | 1977-12-27 | 1978-12-27 | METHOD FOR PRODUCING NEW SPIROBENZOFURANONE COMPOUNDS |
| DE7878300912T DE2861651D1 (en) | 1977-12-27 | 1978-12-27 | Spirobenzofuranone compounds, processes for their preparation and their use as medicines |
| US06/115,548 US4284644A (en) | 1977-01-12 | 1980-01-25 | Spirobenzofuranone compounds |
| ES488332A ES8102114A1 (en) | 1977-12-27 | 1980-02-07 | Spirobenzofuranone compounds, processes for their preparation and their use as medicines. |
| AT110381A AT373594B (en) | 1978-06-19 | 1981-03-10 | METHOD FOR PRODUCING NEW SPIROBENZOFURANONE COMPOUNDS |
| US06/257,316 US4342779A (en) | 1977-12-27 | 1981-04-17 | 7-Acetylspirobenzofuranone compound |
| SG838/84A SG83884G (en) | 1977-12-27 | 1984-11-23 | Spirobenzofuranone compounds,processes for their preparation and their use as medicines |
| HK62/85A HK6285A (en) | 1977-12-27 | 1985-01-24 | Spirobenzofuranone compounds,processes for their preparation and their use as medicines |
| MY8500673A MY8500673A (en) | 1977-01-12 | 1985-12-31 | Spirobenzofuranone compounds, processes for their preparation and their use as medicine |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP7470078A JPS552623A (en) | 1978-06-19 | 1978-06-19 | Spiro compound and its preparation |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| JPS552623A true JPS552623A (en) | 1980-01-10 |
Family
ID=13554755
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP7470078A Pending JPS552623A (en) | 1977-01-12 | 1978-06-19 | Spiro compound and its preparation |
Country Status (1)
| Country | Link |
|---|---|
| JP (1) | JPS552623A (en) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS56154478A (en) * | 1980-04-23 | 1981-11-30 | Takeda Chem Ind Ltd | Spiro compound and its preparation |
-
1978
- 1978-06-19 JP JP7470078A patent/JPS552623A/en active Pending
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS56154478A (en) * | 1980-04-23 | 1981-11-30 | Takeda Chem Ind Ltd | Spiro compound and its preparation |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| JPS572298A (en) | Erythromycin derivative | |
| JPS5265267A (en) | Synthesis of spiro compounds | |
| JPS51122051A (en) | Process for preparation of acenaphthenes | |
| JPS5242868A (en) | Process for preparation of 3-(17beta-hydroxyandrosto-4-ene-3-one-17alpha-yl) propyolactone | |
| JPS5225792A (en) | Process for preparing 3-hydroxy-3-methyl cephalosporin derivatives | |
| JPS54106458A (en) | Sesquiterpene derivative | |
| JPS5242867A (en) | Process for preparation of 17alpha -(3-hydroxypropyl)- 17beta-hydroxy-androsto- 4 -ene-3-one | |
| JPS5564582A (en) | Spiro compound and its preparation | |
| JPS5653673A (en) | Alpha-methyl or ethyl-gamma-mono or dialkyl-substituted-gamma- butyro-lactone and its preparation | |
| JPS52153919A (en) | Preparation of resorcin | |
| JPS51122043A (en) | Process for preparation of 3-hydroxy-5- cycloxycyclopento-1-ene deriva tives | |
| JPS52144653A (en) | Preparation of beta-cyclododecene-1-yl-beta-alkoxycarbonylpropionic acid | |
| JPS5266530A (en) | Preparation of novel schiff base compounds | |
| JPS5236645A (en) | Novel process for preparation of vitamin a | |
| JPS5346962A (en) | Preparation of thiopheneacetic acids | |
| JPS57114575A (en) | Preparation of n-aroyl-bis-lactam | |
| JPS5721348A (en) | 2- 1-methyl-2-propenyl -3-hydroxyundecanoic derivative | |
| JPS57197279A (en) | Novel hexaminum compound and its preparation | |
| JPS5724368A (en) | 5-amino-1,4-dihydrocinnoline and its preparation | |
| JPS5394334A (en) | Preparation of high purity quinacridone | |
| JPS53121777A (en) | 2,3,4,5-tetrahydro-1h-2-benzazepin-3-ones and process for their preparation | |
| JPS5498752A (en) | Spiro compound and its preparation | |
| JPS5233997A (en) | Preparation of polyester | |
| JPS5528938A (en) | Alpha-substituted amino-epsilon-caprolactam | |
| JPS52105190A (en) | Preparation of cephalosporanic-acid-2-nitrobutylester |