JPS5673073A - Preparation of n-substituted imidazole - Google Patents
Preparation of n-substituted imidazoleInfo
- Publication number
- JPS5673073A JPS5673073A JP15021579A JP15021579A JPS5673073A JP S5673073 A JPS5673073 A JP S5673073A JP 15021579 A JP15021579 A JP 15021579A JP 15021579 A JP15021579 A JP 15021579A JP S5673073 A JPS5673073 A JP S5673073A
- Authority
- JP
- Japan
- Prior art keywords
- imidazolyl
- carbinol
- phosphine
- tri
- formula
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Landscapes
- Plural Heterocyclic Compounds (AREA)
Abstract
PURPOSE: To obtain the titled compound, useful as an agent, and having an antifungal activity readily in high yield, by reacting a carbinol as a starting material with a tri-(1-imidazolyl)phosphine.
CONSTITUTION: A carbinol of formula I (Y is O, S, direct bond, CH2-CH2 or CH= CH; A is phenyl or pyridyl) is reacted with a tri(1-imidazolyl)phosphine in the presence of a solvent, preferably acetonitrile or chloroform, at room temperature or under heating to give the aimed compound of formula II (Imd is 1-imidazolyl group). The tri-(1-imidazolyl)-phosphine is used in a molar amount of 1/3 or more, perferably 2/3-2 times, that of the carbinol of formula I.
COPYRIGHT: (C)1981,JPO&Japio
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP15021579A JPS5673073A (en) | 1979-11-19 | 1979-11-19 | Preparation of n-substituted imidazole |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP15021579A JPS5673073A (en) | 1979-11-19 | 1979-11-19 | Preparation of n-substituted imidazole |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| JPS5673073A true JPS5673073A (en) | 1981-06-17 |
Family
ID=15492043
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP15021579A Pending JPS5673073A (en) | 1979-11-19 | 1979-11-19 | Preparation of n-substituted imidazole |
Country Status (1)
| Country | Link |
|---|---|
| JP (1) | JPS5673073A (en) |
Cited By (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5173489A (en) * | 1986-04-10 | 1992-12-22 | The Dupont Merck Pharmaceutical Co. | α,α-disubstituted aromatics and heteroaromatics as cognition enhancers |
| US5300642A (en) * | 1986-04-10 | 1994-04-05 | The Du Pont Merck Pharmaceutical Company | α, α-disubstituted aromatics and heteroaromatics as cognition enhancers |
| US5434264A (en) * | 1988-08-23 | 1995-07-18 | The Du Pont Merck Pharmaceutical Company | α,α-disubstituted aromatics and heteroaromatics as cognition enhancers |
-
1979
- 1979-11-19 JP JP15021579A patent/JPS5673073A/en active Pending
Cited By (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5173489A (en) * | 1986-04-10 | 1992-12-22 | The Dupont Merck Pharmaceutical Co. | α,α-disubstituted aromatics and heteroaromatics as cognition enhancers |
| US5300642A (en) * | 1986-04-10 | 1994-04-05 | The Du Pont Merck Pharmaceutical Company | α, α-disubstituted aromatics and heteroaromatics as cognition enhancers |
| US5434264A (en) * | 1988-08-23 | 1995-07-18 | The Du Pont Merck Pharmaceutical Company | α,α-disubstituted aromatics and heteroaromatics as cognition enhancers |
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