JPS5724387A - Manufacture of heterocyclic alkylguanidine - Google Patents

Manufacture of heterocyclic alkylguanidine

Info

Publication number
JPS5724387A
JPS5724387A JP8369081A JP8369081A JPS5724387A JP S5724387 A JPS5724387 A JP S5724387A JP 8369081 A JP8369081 A JP 8369081A JP 8369081 A JP8369081 A JP 8369081A JP S5724387 A JPS5724387 A JP S5724387A
Authority
JP
Japan
Prior art keywords
formula
hydrogen
chem
group
compound
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP8369081A
Other languages
English (en)
Japanese (ja)
Inventor
Uiriamu Hiruzu Dereku
Reimondo Howaito Jiyooji
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Smith Kline and French Laboratories Ltd
Original Assignee
Smith Kline and French Laboratories Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Smith Kline and French Laboratories Ltd filed Critical Smith Kline and French Laboratories Ltd
Publication of JPS5724387A publication Critical patent/JPS5724387A/ja
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/64—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/68—Halogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Physical Or Chemical Processes And Apparatus (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
JP8369081A 1980-05-31 1981-05-30 Manufacture of heterocyclic alkylguanidine Pending JPS5724387A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB8017881 1980-05-31
AU71026/81A AU542270B2 (en) 1980-05-31 1981-05-26 Imidazolylalkylguanidine derivatives

Publications (1)

Publication Number Publication Date
JPS5724387A true JPS5724387A (en) 1982-02-08

Family

ID=36782531

Family Applications (1)

Application Number Title Priority Date Filing Date
JP8369081A Pending JPS5724387A (en) 1980-05-31 1981-05-30 Manufacture of heterocyclic alkylguanidine

Country Status (9)

Country Link
EP (1) EP0041359B1 (2)
JP (1) JPS5724387A (2)
AT (1) ATE10277T1 (2)
AU (1) AU542270B2 (2)
DE (1) DE3167163D1 (2)
DK (1) DK221081A (2)
GR (1) GR75661B (2)
IE (1) IE52019B1 (2)
ZA (1) ZA813659B (2)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1983003250A1 (fr) * 1982-03-16 1983-09-29 Furukawa, Yoshiyasu Derives de l'acide 4-chloro-2-phenylimidazole-5-acetique
JPS6383072A (ja) * 1986-09-15 1988-04-13 ホイマン・ファーマ・ジー・エム・ビー・エイチ・アンド・カンパニー 新規イミダゾリルグアニジン誘導体、その製造法及びその化合物を含有する医薬

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0199845B1 (de) * 1985-04-02 1990-08-01 HEUMANN PHARMA GMBH & CO Imidazolylalkylguanidinderivate, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende Arzneimittel
DE3621104A1 (de) * 1986-06-24 1988-01-07 Heumann Pharma Gmbh & Co 1,4-dihydropyridinderivate, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel
JPH06505265A (ja) * 1991-02-27 1994-06-16 シード・キャピタル・インベストメント・（エス・シー・アイ）・ベスローテン・フェンノートシャップ ヒスタミンｈ↓３受容体に対する作動的または拮抗的活性を有するイミダゾール誘導体
NL9100365A (nl) * 1991-02-27 1992-09-16 Seed Capital Investments Imidazoolderivaten met agonistische of antagonistische activiteit op de histamine h3-receptor.
FR2686084B1 (fr) * 1992-01-10 1995-12-22 Bioprojet Soc Civ Nouveaux derives de l'imidazole, leur preparation et leurs applications therapeutiques.
USRE37303E1 (en) * 1992-01-10 2001-07-31 Institut National Del La Sante Et De La Recherche Medicale Imidazole compounds and their therapeutic applications

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3763179A (en) * 1972-05-05 1973-10-02 Upjohn Co 2-imidazol-1-yl benzophenones
FR2254311A1 (en) * 1973-12-13 1975-07-11 Smith Kline French Lab 4-Alkyl-5-(2-aminoethyl)imidazole compsns - for diagnosing secretory activity of the stomach, prepd eg from 4-methylhistamine or hex-3-yne-1-ol

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1983003250A1 (fr) * 1982-03-16 1983-09-29 Furukawa, Yoshiyasu Derives de l'acide 4-chloro-2-phenylimidazole-5-acetique
JPS6383072A (ja) * 1986-09-15 1988-04-13 ホイマン・ファーマ・ジー・エム・ビー・エイチ・アンド・カンパニー 新規イミダゾリルグアニジン誘導体、その製造法及びその化合物を含有する医薬

Also Published As

Publication number Publication date
GR75661B (2) 1984-08-02
AU542270B2 (en) 1985-02-14
IE811202L (en) 1981-11-30
DK221081A (da) 1981-12-01
AU7102681A (en) 1981-12-10
EP0041359B1 (en) 1984-11-14
IE52019B1 (en) 1987-05-27
EP0041359A1 (en) 1981-12-09
DE3167163D1 (en) 1984-12-20
ZA813659B (en) 1982-08-25
ATE10277T1 (de) 1984-11-15

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