JPS643178A - Production of amine derivative - Google Patents
Production of amine derivativeInfo
- Publication number
- JPS643178A JPS643178A JP15750387A JP15750387A JPS643178A JP S643178 A JPS643178 A JP S643178A JP 15750387 A JP15750387 A JP 15750387A JP 15750387 A JP15750387 A JP 15750387A JP S643178 A JPS643178 A JP S643178A
- Authority
- JP
- Japan
- Prior art keywords
- formula
- ethyleneimine
- expressed
- alkyl
- hydrogen sulfide
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
- 150000001412 amines Chemical class 0.000 title 1
- NOWKCMXCCJGMRR-UHFFFAOYSA-N Aziridine Chemical compound C1CN1 NOWKCMXCCJGMRR-UHFFFAOYSA-N 0.000 abstract 4
- 150000001875 compounds Chemical class 0.000 abstract 4
- RWSOTUBLDIXVET-UHFFFAOYSA-N Dihydrogen sulfide Chemical compound S RWSOTUBLDIXVET-UHFFFAOYSA-N 0.000 abstract 3
- 125000000217 alkyl group Chemical group 0.000 abstract 3
- 229910000037 hydrogen sulfide Inorganic materials 0.000 abstract 3
- 239000002994 raw material Substances 0.000 abstract 3
- XPFVYQJUAUNWIW-UHFFFAOYSA-N furfuryl alcohol Chemical class OCC1=CC=CO1 XPFVYQJUAUNWIW-UHFFFAOYSA-N 0.000 abstract 2
- 150000002576 ketones Chemical class 0.000 abstract 2
- 125000002252 acyl group Chemical group 0.000 abstract 1
- 229940079593 drug Drugs 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
Landscapes
- Furan Compounds (AREA)
Abstract
PURPOSE: To readily obtain the titled compound which is an intermediate for medicines from inexpensive raw materials in high yield, by reacting ethyleneimine as a starting raw material with a lower dialkyl ketone then with hydrogen sulfide and further reacting the resultant product with a furfuryl alcohol derivative.
CONSTITUTION: Ethyleneimine which is a starting raw material is reacted with a lower dialkyl ketone expressed by formula I (R1 and R2 are 1W4C alkyl) in a molar amount within the range of 0.5W1.5 times, preferably 0.9W1.0 based on the compound expressed by formula I at 0W50°C. The resultant product is subsequently reacted with hydrogen sulfide and then a furfuryl alcohol derivative expressed by formula II (R3 and R4 are 1W4C alkyl; R5 is H or acyl; ALK is 1W4C alkyl) at ambient temperature W 80°C to afford a compound expressed by formula III. Furthermore, the hydrogen sulfide is used in a amount within the range of 1W2 times based on the ethyleneimine and the compound expressed by formula II is used in a molar amount within the range of 0.5W2 times based on the ethyleneimine.
COPYRIGHT: (C)1989,JPO&Japio
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP62-157503A JPH013178A (en) | 1987-06-26 | Method for producing amine derivatives |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP62-157503A JPH013178A (en) | 1987-06-26 | Method for producing amine derivatives |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JPS643178A true JPS643178A (en) | 1989-01-06 |
| JPH013178A JPH013178A (en) | 1989-01-06 |
Family
ID=
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