MA23130A1 - Procede de preparation d'un derive de benzylimidazopyridine servant d'antagoniste des recepteurs de l'angiotensine ii. - Google Patents

Procede de preparation d'un derive de benzylimidazopyridine servant d'antagoniste des recepteurs de l'angiotensine ii.

Info

Publication number
MA23130A1
MA23130A1 MA23437A MA23437A MA23130A1 MA 23130 A1 MA23130 A1 MA 23130A1 MA 23437 A MA23437 A MA 23437A MA 23437 A MA23437 A MA 23437A MA 23130 A1 MA23130 A1 MA 23130A1
Authority
MA
Morocco
Prior art keywords
benzylimidazopyridine
angiotensin
antagonist
receptors
derivative
Prior art date
Application number
MA23437A
Other languages
English (en)
Inventor
A Dasilva Jardine Paul
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of MA23130A1 publication Critical patent/MA23130A1/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C69/00—Esters of carboxylic acids; Esters of carbonic or haloformic acids
    • C07C69/74—Esters of carboxylic acids having an esterified carboxyl group bound to a carbon atom of a ring other than a six-membered aromatic ring
    • C07C69/757—Esters of carboxylic acids having an esterified carboxyl group bound to a carbon atom of a ring other than a six-membered aromatic ring having any of the groups OH, O—metal, —CHO, keto, ether, acyloxy, groups, groups, or in the acid moiety
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C69/00—Esters of carboxylic acids; Esters of carbonic or haloformic acids
    • C07C69/74—Esters of carboxylic acids having an esterified carboxyl group bound to a carbon atom of a ring other than a six-membered aromatic ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02—Silicon compounds
    • C07F7/08—Compounds having one or more C—Si linkages
    • C07F7/18—Compounds having one or more C—Si linkages as well as one or more C—O—Si linkages
    • C07F7/1804—Compounds having Si-O-C linkages

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
MA23437A 1993-03-10 1994-03-09 Procede de preparation d'un derive de benzylimidazopyridine servant d'antagoniste des recepteurs de l'angiotensine ii. MA23130A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US08/043,959 US5300668A (en) 1993-03-10 1993-03-10 Certain esters of 1-(4-X-methylphenyl)cyclopent-3-ene-1-carboxylic acid, wherein X is a trialkylsilyloxy, bromo or hydroxy group, as intermediates

Publications (1)

Publication Number Publication Date
MA23130A1 true MA23130A1 (fr) 1994-10-01

Family

ID=21929808

Family Applications (1)

Application Number Title Priority Date Filing Date
MA23437A MA23130A1 (fr) 1993-03-10 1994-03-09 Procede de preparation d'un derive de benzylimidazopyridine servant d'antagoniste des recepteurs de l'angiotensine ii.

Country Status (10)

Country Link
US (1) US5300668A (fr)
AP (1) AP9400618A0 (fr)
AU (1) AU6297394A (fr)
FI (1) FI941118L (fr)
HR (1) HRP940109A2 (fr)
HU (1) HUT67682A (fr)
IL (1) IL108843A0 (fr)
MA (1) MA23130A1 (fr)
SI (1) SI9400120A (fr)
WO (1) WO1994020498A1 (fr)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AP9400651A0 (en) * 1993-07-15 1995-12-30 Pfizer Azacyclic-heterocyclic compounds as angiotensin II receptor antagonists.
NZ290008A (en) * 1994-06-29 1998-08-26 Smithkline Beecham Corp Vitronectin receptor antagonists, comprising a fibrinogen antagonist analogue linked to a heterocycle
US5977101A (en) * 1995-06-29 1999-11-02 Smithkline Beecham Corporation Benzimidazoles/Imidazoles Linked to a Fibrinogen Receptor Antagonist Template Having Vitronectin Receptor Antagonist Activity
EP0914158B2 (fr) * 1996-04-05 2006-01-25 Takeda Chemical Industries, Ltd. Combinaison pharmaceutique comprenant un compose avec activite antagoniste de l'angiotensine ii et un compose qui augmente la sensibilite a l'insuline

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2573015A (en) * 1947-12-24 1951-10-30 Geigy Ag J R Basic esters of 1-aryl-cyclopentene-(3)-1-carboxylic acids
DE3927930A1 (de) * 1989-08-24 1991-02-28 Bayer Ag Cyclisch substituierte (chinolin-2-yl-methoxy)phenyl-essig-saeure-derivate
JPH05504969A (ja) * 1990-02-13 1993-07-29 メルク・エンド・カムパニー・インコーポレーテツド 置換ベンジル要素を含有するアンギオテンシン２アンタゴニスト類
WO1991011909A1 (fr) * 1990-02-13 1991-08-22 Merck & Co., Inc. Antagonistes de triazole angiotensine ii incorporant un element de benzyle substitue
DE4036645A1 (de) * 1990-11-16 1992-05-21 Hoechst Ag Substituierte azole, verfahren zu deren herstellung, deren enthaltende mittel und deren verwendung
DE4200954A1 (de) * 1991-04-26 1992-10-29 Bayer Ag Heterocyclisch substituierte phenylessigsaeurederivate

Also Published As

Publication number Publication date
FI941118A7 (fi) 1994-09-11
WO1994020498A1 (fr) 1994-09-15
SI9400120A (en) 1995-06-30
AP9400618A0 (en) 1995-08-10
HU9400706D0 (en) 1994-06-28
IL108843A0 (en) 1994-06-24
FI941118L (fi) 1994-09-11
AU6297394A (en) 1994-09-26
HRP940109A2 (en) 1997-06-30
FI941118A0 (fi) 1994-03-09
US5300668A (en) 1994-04-05
HUT67682A (en) 1995-04-28

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