MA24485A1 - Atropisomeres de 3-heteroaryl-4(3h)-quinazo linones . - Google Patents

Atropisomeres de 3-heteroaryl-4(3h)-quinazo linones .

Info

Publication number: MA24485A1
Authority: MA; Morocco
Prior art keywords: linones; quinazo; atropisomers; heteroaryl; quinazo linones
Prior art date: 1997-02-28

Application number

MA24979A

Other languages

English (en)

Inventor

Mc Kowan Welch Willard Jr

Michael Devries Keith

Leo Chennard Bertrand

Original Assignee

Pfizer Prod Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1997-02-28

Filing date

1998-02-25

Publication date

1998-10-01

1998-02-25 Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc

1998-10-01 Publication of MA24485A1 publication Critical patent/MA24485A1/fr

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
- A61P21/02—Muscle relaxants, e.g. for tetanus or cramps
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/10—Spiro-condensed systems

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Bioinformatics & Cheminformatics (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Engineering & Computer Science (AREA)
Public Health (AREA)
Chemical Kinetics & Catalysis (AREA)
Neurology (AREA)
Cardiology (AREA)
Heart & Thoracic Surgery (AREA)
Biomedical Technology (AREA)
Neurosurgery (AREA)
Pain & Pain Management (AREA)
Orthopedic Medicine & Surgery (AREA)
Physical Education & Sports Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)

MA24979A 1997-02-28 1998-02-25 Atropisomeres de 3-heteroaryl-4(3h)-quinazo linones . MA24485A1 (fr)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US3854097P	1997-02-28	1997-02-28

Publications (1)

Publication Number	Publication Date
MA24485A1 true MA24485A1 (fr)	1998-10-01

Family

ID=21900535

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
MA24979A MA24485A1 (fr)	1997-02-28	1998-02-25	Atropisomeres de 3-heteroaryl-4(3h)-quinazo linones .

Country Status (40)

Country	Link
US (1)	US6380204B1 (fr)
EP (1)	EP0964860B1 (fr)
JP (1)	JP3299990B2 (fr)
KR (1)	KR20000075812A (fr)
CN (1)	CN1248254A (fr)
AP (1)	AP9801202A0 (fr)
AR (1)	AR011886A1 (fr)
AT (1)	ATE264854T1 (fr)
AU (1)	AU732448B2 (fr)
BG (1)	BG103687A (fr)
BR (1)	BR9807807A (fr)
CA (1)	CA2282279C (fr)
CO (1)	CO4950615A1 (fr)
DE (1)	DE69823339T2 (fr)
DK (1)	DK0964860T3 (fr)
DZ (1)	DZ2438A1 (fr)
EA (1)	EA001961B1 (fr)
ES (1)	ES2218801T3 (fr)
GT (1)	GT199800039A (fr)
HN (1)	HN1998000028A (fr)
HR (1)	HRP980108B1 (fr)
HU (1)	HUP0000935A3 (fr)
ID (1)	ID23435A (fr)
IL (1)	IL130897A0 (fr)
IS (1)	IS5141A (fr)
MA (1)	MA24485A1 (fr)
NO (1)	NO994178D0 (fr)
NZ (1)	NZ336627A (fr)
OA (1)	OA11088A (fr)
PA (1)	PA8446901A1 (fr)
PE (1)	PE57999A1 (fr)
PL (1)	PL335307A1 (fr)
PT (1)	PT964860E (fr)
SK (1)	SK113199A3 (fr)
TN (1)	TNSN98034A1 (fr)
TR (1)	TR199902094T2 (fr)
TW (1)	TW530055B (fr)
UA (1)	UA58536C2 (fr)
WO (1)	WO1998038187A1 (fr)
ZA (1)	ZA981665B (fr)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US6323208B1 (en)	1997-09-05	2001-11-27	Pfizer Inc	Atropisomers of 2,3-disubstituted-(5.6)-heteroaryl fused-pyrimidin-4-ones
JPH11279158A (ja) *	1998-02-09	1999-10-12	Pfizer Prod Inc	キナゾリン―４―オン誘導体の製造方法
US6890930B1 (en) *	1999-09-28	2005-05-10	3-Dimensional Pharmaceuticals, Inc.	Quinazolinones
US20080146562A1 (en) *	2003-08-08	2008-06-19	Ulysses Pharmaceutical Products Inc.,	Halogenated quinazolinyl nitrofurans as antibacterial agents
EP1660486A4 (fr) *	2003-08-08	2006-12-13	Ulysses Pharmaceutical Product	Quinazolinyl nitrofuranes halogenes utilises comme agents antibacteriens
GB0416730D0 (en)	2004-07-27	2004-09-01	Novartis Ag	Organic compounds
GB0507298D0 (en)	2005-04-11	2005-05-18	Novartis Ag	Organic compounds
US20100152209A1 (en) *	2005-11-04	2010-06-17	Hydra Biosciences Inc.	Compounds for Modulating TRPV3 Function
CA2663436A1 (fr) *	2006-10-04	2008-04-10	Pfizer Products Inc.	Derives de pyrido[4,3-d]pyrimidin-4(3h)-one utilises en tant qu'antagonistes du recepteur calcique
WO2008140750A1 (fr) *	2007-05-10	2008-11-20	Hydra Biosciences Inc.	Composés modulant la fonction du trp v3
AU2010229968A1 (en) *	2009-03-24	2011-10-13	Gilead Calistoga Llc	Atropisomers of2-purinyl-3-tolyl-quinazolinone derivatives and methods of use
ES2739973T3 (es)	2009-05-29	2020-02-05	Merck Sharp & Dohme	Inhibidores de PDE10 radiomarcados
WO2013105985A1 (fr)	2011-02-28	2013-07-18	Philadelphia Health & Education Corporation	Inhibiteurs à petites molécules de la recombinase rad51 et procédés associés
EP4574822A3 (fr)	2020-01-29	2025-08-27	Kamari Pharma Ltd.	Composés et compositions pour leur utilisation dans le traitement de troubles cutanés

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3748325A (en) *	1970-04-06	1973-07-24	Karamchand Premchand Private	Process for the preparation of quinazolinone derivatives
US4183931A (en) *	1977-09-08	1980-01-15	Research Corporation	2-Ketoalkyl-4(3H)-quinazolinones
WO1992013535A1 (fr) *	1991-02-06	1992-08-20	Research Corporation Technologies, Inc.	Quinazolones substituees a activite anticonvulsivante
BR9709085A (pt) *	1996-05-15	1999-08-03	Pfizer	Novas 2,3-dissubstituído-4(3H)-quinazolinonas
ES2184960T3 (es) *	1996-05-15	2003-04-16	Pfizer	Nuevas pirimidin-4-onas-(5,6)-heteroaril condensadas 2,3 disustituidas.

1998
- 1998-02-06 US US09/380,114 patent/US6380204B1/en not_active Expired - Fee Related
- 1998-02-06 AU AU57759/98A patent/AU732448B2/en not_active Ceased
- 1998-02-06 IL IL13089798A patent/IL130897A0/xx unknown
- 1998-02-06 KR KR1019997007885A patent/KR20000075812A/ko not_active Abandoned
- 1998-02-06 DK DK98901424T patent/DK0964860T3/da active
- 1998-02-06 CA CA002282279A patent/CA2282279C/fr not_active Expired - Fee Related
- 1998-02-06 BR BR9807807-0A patent/BR9807807A/pt not_active Application Discontinuation
- 1998-02-06 PT PT98901424T patent/PT964860E/pt unknown
- 1998-02-06 TR TR1999/02094T patent/TR199902094T2/xx unknown
- 1998-02-06 ID IDW990935D patent/ID23435A/id unknown
- 1998-02-06 CN CN98802796A patent/CN1248254A/zh active Pending
- 1998-02-06 HU HU0000935A patent/HUP0000935A3/hu unknown
- 1998-02-06 ES ES98901424T patent/ES2218801T3/es not_active Expired - Lifetime
- 1998-02-06 EP EP98901424A patent/EP0964860B1/fr not_active Expired - Lifetime
- 1998-02-06 DE DE69823339T patent/DE69823339T2/de not_active Expired - Fee Related
- 1998-02-06 JP JP53744998A patent/JP3299990B2/ja not_active Expired - Fee Related
- 1998-02-06 SK SK1131-99A patent/SK113199A3/sk unknown
- 1998-02-06 EA EA199900689A patent/EA001961B1/ru not_active IP Right Cessation
- 1998-02-06 NZ NZ336627A patent/NZ336627A/xx unknown
- 1998-02-06 PL PL98335307A patent/PL335307A1/xx unknown
- 1998-02-06 AT AT98901424T patent/ATE264854T1/de not_active IP Right Cessation
- 1998-02-06 WO PCT/IB1998/000151 patent/WO1998038187A1/fr not_active Ceased
- 1998-02-09 HN HN1998000028A patent/HN1998000028A/es unknown
- 1998-02-17 PA PA19988446901A patent/PA8446901A1/es unknown
- 1998-02-19 GT GT199800039A patent/GT199800039A/es unknown
- 1998-02-23 PE PE1998000127A patent/PE57999A1/es not_active Application Discontinuation
- 1998-02-25 MA MA24979A patent/MA24485A1/fr unknown
- 1998-02-25 TW TW087102713A patent/TW530055B/zh not_active IP Right Cessation
- 1998-02-25 CO CO98010303A patent/CO4950615A1/es unknown
- 1998-02-25 TN TNTNSN98034A patent/TNSN98034A1/fr unknown
- 1998-02-25 DZ DZ980048A patent/DZ2438A1/fr active
- 1998-02-26 AP APAP/P/1998/001202A patent/AP9801202A0/en unknown
- 1998-02-26 AR ARP980100872A patent/AR011886A1/es unknown
- 1998-02-27 ZA ZA9801665A patent/ZA981665B/xx unknown
- 1998-02-27 HR HR980108A patent/HRP980108B1/xx not_active IP Right Cessation
- 1998-06-02 UA UA99084850A patent/UA58536C2/uk unknown
1999
- 1999-07-30 IS IS5141A patent/IS5141A/is unknown
- 1999-08-20 OA OA9900186A patent/OA11088A/fr unknown
- 1999-08-24 BG BG103687A patent/BG103687A/xx unknown
- 1999-08-27 NO NO994178A patent/NO994178D0/no unknown

Also Published As

Publication number	Publication date
NO994178L (no)	1999-08-27
AU5775998A (en)	1998-09-18
HRP980108B1 (en)	2004-10-31
JP2000509732A (ja)	2000-08-02
AP9801202A0 (en)	1999-08-26
IS5141A (is)	1999-07-30
NO994178D0 (no)	1999-08-27
NZ336627A (en)	2000-12-22
TW530055B (en)	2003-05-01
GT199800039A (es)	1999-08-13
DK0964860T3 (da)	2004-07-26
ATE264854T1 (de)	2004-05-15
PL335307A1 (en)	2000-04-10
DE69823339T2 (de)	2005-05-12
HUP0000935A3 (en)	2002-04-29
HRP980108A2 (en)	1998-12-31
PE57999A1 (es)	1999-06-21
DZ2438A1 (fr)	2003-01-11
BR9807807A (pt)	2000-02-22
US6380204B1 (en)	2002-04-30
AR011886A1 (es)	2000-09-13
AU732448B2 (en)	2001-04-26
PA8446901A1 (es)	2000-05-24
EA199900689A1 (ru)	2000-02-28
DE69823339D1 (de)	2004-05-27
CA2282279A1 (fr)	1998-09-03
OA11088A (en)	2002-03-15
BG103687A (en)	2000-06-30
EP0964860B1 (fr)	2004-04-21
CN1248254A (zh)	2000-03-22
WO1998038187A1 (fr)	1998-09-03
CA2282279C (fr)	2004-11-02
HN1998000028A (es)	1999-02-09
EA001961B1 (ru)	2001-10-22
PT964860E (pt)	2004-07-30
SK113199A3 (en)	2001-10-08
TNSN98034A1 (fr)	2005-03-15
HUP0000935A2 (hu)	2001-04-28
ES2218801T3 (es)	2004-11-16
KR20000075812A (ko)	2000-12-26
EP0964860A1 (fr)	1999-12-22
ID23435A (id)	2000-04-20
TR199902094T2 (xx)	1999-12-21
CO4950615A1 (es)	2000-09-01
UA58536C2 (uk)	2003-08-15
JP3299990B2 (ja)	2002-07-08
IL130897A0 (en)	2001-01-28
ZA981665B (en)	1999-08-17

Publication	Publication Date	Title
ZA981666B (en)	1999-08-27	Atropisomers of 3-aryl-4(3H)-quinazolinones.
FR2715460B1 (fr)	1999-03-26	Structure de brûleur.
BR9806033B1 (pt)	2011-04-19	relógio.
FR2770110B1 (fr)	1999-11-19	Boitier, du type boitier de maquillage
BR9907304B1 (pt)	2008-11-18	refratÁrio de alumina-magnÉsia-grafita.
MX224819B (es)	2004-12-23	Empleo cosmetico de derivados de bis(resorcinil)triacina.
DZ2438A1 (fr)	2003-01-11	Atropisomères de 3-hétéroaryl-4(3h)-quinazolinones.
MA24551A1 (fr)	1998-12-31	W.c.
ES1036909Y (es)	1998-05-01	Pupitre infantil.
DZ2695A1 (fr)	2003-03-29	Maitrise des acridiens.
ES1035340Y (es)	1997-10-01	Expositor-contenedor de publicaciones.
ID21262A (id)	1999-05-12	Progestagen kristalin
ES1036260Y (es)	1997-12-16	Conjunto de coccion.
ES1037395Y (es)	1998-07-01	Tendedero antilluvia.
IT1301728B1 (it)	2000-07-07	Preparazione di un complesso antianemico.
ES1033267Y (es)	1997-01-01	Pieza de joyeria.
ES1033965Y (es)	1997-04-16	Pieza de joyeria.
EP0873349A4 (fr)	2001-03-14	Polypeptide de type iii activateur des monocytes et des cellules endotheliales
ES1038481Y (es)	1999-05-16	Ducha.
ES1029940Y (es)	1996-01-01	Pieza de construccion.
ES1039835Y (es)	1999-07-01	Jamba de puertas basculantes.
ES1029922Y (es)	1996-01-01	Baston-recogedor de excrementos.
ES1035807Y (es)	1997-12-16	Conjunto de sellos componibles.
ES1039318Y (es)	1999-05-16	Conjunto de sartenes.
ES1034145Y (es)	1997-05-01	Talonario autocopiativo de nuevas caracteristicas.