MA25089A1 - Formulations intranasales de mesylate de sildenafil et procede pour leur preparation - Google Patents

Formulations intranasales de mesylate de sildenafil et procede pour leur preparation

Info

Publication number
MA25089A1
MA25089A1 MA25639A MA25639A MA25089A1 MA 25089 A1 MA25089 A1 MA 25089A1 MA 25639 A MA25639 A MA 25639A MA 25639 A MA25639 A MA 25639A MA 25089 A1 MA25089 A1 MA 25089A1
Authority
MA
Morocco
Prior art keywords
preparation
intranasal formulations
sildenafil mesylate
sildenafil
mesylate
Prior art date
Application number
MA25639A
Other languages
English (en)
Inventor
James Dunn Peter
Jayne Woods Joanna
Thomas Henry Brian
Billotte Anne
Vallance Marshall Peter
Original Assignee
Pfizer Res & Dev
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GBGB9813452.1A external-priority patent/GB9813452D0/en
Priority claimed from GBGB9820837.4A external-priority patent/GB9820837D0/en
Priority claimed from GBGB9903177.5A external-priority patent/GB9903177D0/en
Application filed by Pfizer Res & Dev filed Critical Pfizer Res & Dev
Publication of MA25089A1 publication Critical patent/MA25089A1/fr

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0043Nose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/08Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/10Drugs for genital or sexual disorders; Contraceptives for impotence

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Reproductive Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Endocrinology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Gynecology & Obstetrics (AREA)
  • Otolaryngology (AREA)
  • Pregnancy & Childbirth (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
MA25639A 1998-06-22 1999-06-21 Formulations intranasales de mesylate de sildenafil et procede pour leur preparation MA25089A1 (fr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB9813452.1A GB9813452D0 (en) 1998-06-22 1998-06-22 Pharmaceutical formulations
GBGB9820837.4A GB9820837D0 (en) 1998-09-24 1998-09-24 Pharmaceutical formulations
GBGB9903177.5A GB9903177D0 (en) 1999-02-13 1999-02-13 Pharmaceutical formulations

Publications (1)

Publication Number Publication Date
MA25089A1 true MA25089A1 (fr) 2000-12-31

Family

ID=27269368

Family Applications (1)

Application Number Title Priority Date Filing Date
MA25639A MA25089A1 (fr) 1998-06-22 1999-06-21 Formulations intranasales de mesylate de sildenafil et procede pour leur preparation

Country Status (40)

Country Link
US (2) US20020040139A1 (fr)
EP (1) EP0967214B1 (fr)
JP (1) JP3263379B2 (fr)
KR (1) KR100345824B1 (fr)
AP (1) AP1178A (fr)
AR (1) AR016993A1 (fr)
AT (1) ATE269866T1 (fr)
AU (1) AU746865B2 (fr)
BG (1) BG64372B1 (fr)
BR (1) BR9903273A (fr)
CA (1) CA2275554C (fr)
CZ (1) CZ294856B6 (fr)
DE (1) DE69918222T2 (fr)
DK (1) DK0967214T3 (fr)
DZ (1) DZ2826A1 (fr)
EA (1) EA001903B1 (fr)
ES (1) ES2221733T3 (fr)
GT (1) GT199900095A (fr)
HN (1) HN1999000096A (fr)
HR (1) HRP990195B1 (fr)
HU (1) HUP9902076A3 (fr)
ID (1) ID23554A (fr)
IL (1) IL130539A0 (fr)
IS (1) IS5085A (fr)
MA (1) MA25089A1 (fr)
MY (1) MY117967A (fr)
NO (1) NO317365B1 (fr)
NZ (1) NZ336382A (fr)
OA (1) OA11069A (fr)
PA (1) PA8476301A1 (fr)
PE (1) PE20000702A1 (fr)
PT (1) PT967214E (fr)
SG (1) SG77246A1 (fr)
SI (1) SI0967214T1 (fr)
SK (1) SK284574B6 (fr)
TN (1) TNSN99129A1 (fr)
TR (1) TR199901444A2 (fr)
TW (1) TWI223598B (fr)
UA (1) UA59385C2 (fr)
YU (1) YU29699A (fr)

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Also Published As

Publication number Publication date
BG64372B1 (bg) 2004-12-30
IL130539A0 (en) 2000-06-01
CZ9902257A3 (cs) 2000-11-15
ID23554A (id) 2000-05-04
IS5085A (is) 1999-12-23
CZ294856B6 (cs) 2005-03-16
CA2275554A1 (fr) 1999-12-22
AU746865B2 (en) 2002-05-02
HRP990195A2 (en) 2000-02-29
DK0967214T3 (da) 2004-09-27
EA001903B1 (ru) 2001-10-22
BG103510A (en) 2000-01-31
PA8476301A1 (es) 2000-09-29
SG77246A1 (en) 2000-12-19
SI0967214T1 (en) 2004-10-31
EP0967214A1 (fr) 1999-12-29
EA199900487A3 (ru) 2000-04-24
JP3263379B2 (ja) 2002-03-04
ATE269866T1 (de) 2004-07-15
SK81999A3 (en) 2001-01-18
UA59385C2 (uk) 2003-09-15
HU9902076D0 (en) 1999-08-30
US20030158206A1 (en) 2003-08-21
AR016993A1 (es) 2001-08-01
EA199900487A2 (ru) 1999-12-29
PT967214E (pt) 2004-08-31
HUP9902076A2 (hu) 2000-05-28
KR20000006310A (ko) 2000-01-25
DZ2826A1 (fr) 2003-12-01
BR9903273A (pt) 2000-05-09
NZ336382A (en) 1999-11-29
KR100345824B1 (ko) 2002-07-24
EP0967214B1 (fr) 2004-06-23
CA2275554C (fr) 2003-06-03
HN1999000096A (es) 2000-12-03
SK284574B6 (sk) 2005-06-02
AP9901585A0 (en) 1999-06-30
HUP9902076A3 (en) 2002-03-28
TR199901444A2 (xx) 2000-01-21
YU29699A (sh) 2003-02-28
NO993051D0 (no) 1999-06-21
DE69918222D1 (de) 2004-07-29
US20020040139A1 (en) 2002-04-04
JP2000034232A (ja) 2000-02-02
AU3579499A (en) 2000-01-06
TNSN99129A1 (fr) 2005-11-10
NO993051L (no) 1999-12-23
TWI223598B (en) 2004-11-11
DE69918222T2 (de) 2005-07-28
ES2221733T3 (es) 2005-01-01
HRP990195B1 (en) 2003-04-30
MY117967A (en) 2004-08-30
PE20000702A1 (es) 2000-08-16
AP1178A (en) 2003-06-30
GT199900095A (es) 2000-12-13
NO317365B1 (no) 2004-10-18
OA11069A (en) 2002-03-13

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