MA26756A1 - Derives de thiazole - Google Patents

Derives de thiazole

Info

Publication number: MA26756A1
Authority: MA; Morocco
Prior art keywords: thiazole derivatives; thiazole; derivatives
Prior art date: 1998-10-22

Application number

MA26171A

Other languages

English (en)

Inventor

Kurt Hilpert

Leo Alig

Thomas Weller

Original Assignee

Hoffmann La Roche

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1998-10-22

Filing date

2001-04-20

Publication date

2004-12-20

2001-04-20 Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche

2004-12-20 Publication of MA26756A1 publication Critical patent/MA26756A1/fr

Links

150000007979 thiazole derivatives Chemical class 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/38—Nitrogen atoms
- C07D277/44—Acylated amino or imino radicals
- C07D277/48—Acylated amino or imino radicals by radicals derived from carbonic acid, or sulfur or nitrogen analogues thereof, e.g. carbonylguanidines
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/06—Antipsoriatics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/10—Antimycotics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/04—Antineoplastic agents specific for metastasis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Physical Education & Sports Medicine (AREA)
Oncology (AREA)
Communicable Diseases (AREA)
Orthopedic Medicine & Surgery (AREA)
Rheumatology (AREA)
Urology & Nephrology (AREA)
Heart & Thoracic Surgery (AREA)
Cardiology (AREA)
Virology (AREA)
Gastroenterology & Hepatology (AREA)
Dermatology (AREA)
Ophthalmology & Optometry (AREA)
Immunology (AREA)
Vascular Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Thiazole And Isothizaole Compounds (AREA)
Medicinal Preparation (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Plural Heterocyclic Compounds (AREA)

MA26171A 1998-10-22 2001-04-20 Derives de thiazole MA26756A1 (fr)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
EP98119985		1998-10-22

Publications (1)

Publication Number	Publication Date
MA26756A1 true MA26756A1 (fr)	2004-12-20

Family

ID=8232838

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
MA26171A MA26756A1 (fr)	1998-10-22	2001-04-20	Derives de thiazole

Country Status (31)

Country	Link
US (1)	US6297266B1 (fr)
EP (1)	EP1123283B1 (fr)
JP (1)	JP3530137B2 (fr)
KR (1)	KR100469219B1 (fr)
CN (1)	CN1211375C (fr)
AR (1)	AR023058A1 (fr)
AT (1)	ATE266012T1 (fr)
AU (1)	AU760219B2 (fr)
BR (1)	BR9914666A (fr)
CA (1)	CA2347741C (fr)
CO (1)	CO5150186A1 (fr)
CZ (1)	CZ20011395A3 (fr)
DE (1)	DE69917058T2 (fr)
DK (1)	DK1123283T3 (fr)
ES (1)	ES2221482T3 (fr)
HK (1)	HK1047281A1 (fr)
HR (1)	HRP20010275A2 (fr)
HU (1)	HUP0104202A3 (fr)
ID (1)	ID28356A (fr)
IL (1)	IL142090A0 (fr)
MA (1)	MA26756A1 (fr)
NO (1)	NO20011908L (fr)
NZ (1)	NZ510676A (fr)
PE (1)	PE20001116A1 (fr)
PL (1)	PL347427A1 (fr)
PT (1)	PT1123283E (fr)
RU (1)	RU2214404C2 (fr)
TR (1)	TR200101115T2 (fr)
WO (1)	WO2000024724A1 (fr)
YU (1)	YU29201A (fr)
ZA (1)	ZA200102653B (fr)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US7125875B2 (en)	1999-04-15	2006-10-24	Bristol-Myers Squibb Company	Cyclic protein tyrosine kinase inhibitors
CA2366932C (fr)	1999-04-15	2009-08-25	Bristol-Myers Squibb Company	Inhibiteurs cycliques de proteine tyrosine kinase
WO2001052847A1 (fr) *	2000-01-19	2001-07-26	Alteon, Inc.	Composes thiazole, imidazole et oxazole et traitements de troubles associes au vieillissement des proteines
EP1313729B1 (fr)	2000-08-17	2007-03-21	Lumera Corporation	Conception et synthese de materiaux optiques non lineaires de pointe destines a des applications electro-optiques
ES2257461T3 (es)	2000-12-21	2006-08-01	Bristol-Myers Squibb Company	Inhibidores de tiazolilo de tirosina quinasas de la familia tec.
CA2580725A1 (fr) *	2004-09-20	2006-03-30	4Sc Ag	Nouveaux inhibiteurs heterocycliques du nf-?b
UA103319C2 (en)	2008-05-06	2013-10-10	Глаксосмитклайн Ллк	Thiazole- and oxazole-benzene sulfonamide compounds
WO2010012793A1 (fr) *	2008-08-01	2010-02-04	Bayer Cropscience Sa	Dérivés d'aminothiazole fongicides

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
IL95548A0 (en) *	1989-09-15	1991-06-30	Fujisawa Pharmaceutical Co	Thiazole derivatives,processes for the preparation thereof and pharmaceutical composition containing the same
US5273982A (en)	1990-03-09	1993-12-28	Hoffmann-La Roche Inc.	Acetic acid derivatives
CA2037153A1 (fr) *	1990-03-09	1991-09-10	Leo Alig	Derives de l'acide acetique
US6306840B1 (en) *	1995-01-23	2001-10-23	Biogen, Inc.	Cell adhesion inhibitors
JPH0987237A (ja) *	1995-09-21	1997-03-31	Kyowa Hakko Kogyo Co Ltd	芳香族誘導体
ES2185009T3 (es)	1996-04-10	2003-04-16	Merck & Co Inc	Antagonistas de alfa y beta 3'.
EP0907637A1 (fr)	1996-06-28	1999-04-14	MERCK PATENT GmbH	Derives de phenylalanine utilises comme inhibiteurs de l'integrine
EP0928790B1 (fr) *	1998-01-02	2003-03-05	F. Hoffmann-La Roche Ag	Dérivés du thiazole
SI0928793T1 (en) *	1998-01-02	2002-10-31	F. Hoffmann-La Roche Ag	Thiazole derivatives
US6100282A (en)	1998-01-02	2000-08-08	Hoffman-La Roche Inc.	Thiazole derivatives
US6001855A (en)	1998-01-02	1999-12-14	Hoffman-La Roche Inc.	Thiazole derivatives

1999
- 1999-10-15 IL IL14209099A patent/IL142090A0/xx unknown
- 1999-10-15 HK HK02108922.4A patent/HK1047281A1/zh unknown
- 1999-10-15 RU RU2001113285/04A patent/RU2214404C2/ru not_active IP Right Cessation
- 1999-10-15 BR BR9914666-5A patent/BR9914666A/pt not_active IP Right Cessation
- 1999-10-15 DK DK99970988T patent/DK1123283T3/da active
- 1999-10-15 NZ NZ510676A patent/NZ510676A/xx unknown
- 1999-10-15 EP EP99970988A patent/EP1123283B1/fr not_active Expired - Lifetime
- 1999-10-15 WO PCT/EP1999/007824 patent/WO2000024724A1/fr not_active Ceased
- 1999-10-15 AT AT99970988T patent/ATE266012T1/de not_active IP Right Cessation
- 1999-10-15 HU HU0104202A patent/HUP0104202A3/hu unknown
- 1999-10-15 ID IDW20010863A patent/ID28356A/id unknown
- 1999-10-15 TR TR2001/01115T patent/TR200101115T2/xx unknown
- 1999-10-15 HR HR20010275A patent/HRP20010275A2/hr not_active Application Discontinuation
- 1999-10-15 DE DE69917058T patent/DE69917058T2/de not_active Expired - Fee Related
- 1999-10-15 YU YU29201A patent/YU29201A/sh unknown
- 1999-10-15 CZ CZ20011395A patent/CZ20011395A3/cs unknown
- 1999-10-15 KR KR10-2001-7004899A patent/KR100469219B1/ko not_active Expired - Fee Related
- 1999-10-15 PL PL99347427A patent/PL347427A1/xx not_active Application Discontinuation
- 1999-10-15 CN CNB998124265A patent/CN1211375C/zh not_active Expired - Fee Related
- 1999-10-15 PT PT99970988T patent/PT1123283E/pt unknown
- 1999-10-15 JP JP2000578294A patent/JP3530137B2/ja not_active Expired - Fee Related
- 1999-10-15 ES ES99970988T patent/ES2221482T3/es not_active Expired - Lifetime
- 1999-10-15 CA CA002347741A patent/CA2347741C/fr not_active Expired - Fee Related
- 1999-10-15 AU AU11519/00A patent/AU760219B2/en not_active Ceased
- 1999-10-18 PE PE1999001048A patent/PE20001116A1/es not_active Application Discontinuation
- 1999-10-19 US US09/420,387 patent/US6297266B1/en not_active Expired - Fee Related
- 1999-10-20 CO CO99066263A patent/CO5150186A1/es unknown
- 1999-10-20 AR ARP990105306A patent/AR023058A1/es not_active Application Discontinuation
2001
- 2001-03-30 ZA ZA200102653A patent/ZA200102653B/en unknown
- 2001-04-18 NO NO20011908A patent/NO20011908L/no not_active Application Discontinuation
- 2001-04-20 MA MA26171A patent/MA26756A1/fr unknown

Also Published As

Publication number	Publication date
BR9914666A (pt)	2001-07-17
NZ510676A (en)	2003-06-30
DE69917058D1 (de)	2004-06-09
CN1211375C (zh)	2005-07-20
JP3530137B2 (ja)	2004-05-24
ZA200102653B (en)	2002-07-01
CA2347741C (fr)	2006-12-12
PE20001116A1 (es)	2000-10-27
CZ20011395A3 (cs)	2001-08-15
YU29201A (sh)	2005-06-10
NO20011908D0 (no)	2001-04-18
WO2000024724A1 (fr)	2000-05-04
EP1123283B1 (fr)	2004-05-06
HRP20010275A2 (en)	2002-06-30
ATE266012T1 (de)	2004-05-15
KR20010080243A (ko)	2001-08-22
HK1047281A1 (zh)	2003-02-14
CO5150186A1 (es)	2002-04-29
ES2221482T3 (es)	2004-12-16
KR100469219B1 (ko)	2005-02-07
ID28356A (id)	2001-05-17
EP1123283A1 (fr)	2001-08-16
NO20011908L (no)	2001-04-18
AU760219B2 (en)	2003-05-08
PL347427A1 (en)	2002-04-08
AR023058A1 (es)	2002-09-04
HUP0104202A2 (hu)	2002-03-28
AU1151900A (en)	2000-05-15
CA2347741A1 (fr)	2000-05-04
TR200101115T2 (tr)	2002-01-21
IL142090A0 (en)	2002-03-10
US6297266B1 (en)	2001-10-02
PT1123283E (pt)	2004-09-30
RU2214404C2 (ru)	2003-10-20
DE69917058T2 (de)	2005-04-07
DK1123283T3 (da)	2004-09-13
JP2002528442A (ja)	2002-09-03
HUP0104202A3 (en)	2003-12-29
CN1359381A (zh)	2002-07-17

Publication	Publication Date	Title
PT930302E (pt)	2003-07-31	Derivados de benzo-sulfona
NO20010193D0 (no)	2001-01-12	Tiobenzimidazol-derivater
MA26766A1 (fr)	2004-12-20	Derives de phenylglycine
ATE426598T1 (de)	2009-04-15	Epothilonderivate
PT1104422E (pt)	2004-06-30	Derivados de fenilxantina
NO20010514D0 (no)	2001-01-30	Aminometylkarboksylsyre-derivater
MA26591A1 (fr)	2004-12-20	Nouveaux derives de thiazole
PT1140924E (pt)	2006-08-31	Derivados de piperazina
PT1056716E (pt)	2003-04-30	Derivados de ciclo-hexanodiolo
DK1115716T3 (da)	2003-02-24	2-phenylpyran-4-on-derivater
DK1134219T3 (da)	2005-10-17	Cucloalkylsubstituerede aminomethylpyrrolidinderivater
ATE233253T1 (de)	2003-03-15	Chromanderivate
DK1060183T3 (da)	2003-08-11	5-deoxycytidinderivater
MA26480A1 (fr)	2004-12-20	Derives de phenoxymethylpiperidine
PT1123283E (pt)	2004-09-30	Derivados de tiazole
ATE217621T1 (de)	2002-06-15	Thiazol-derivate
DE59907635D1 (de)	2003-12-11	Pyrazolyldioxothiochromanoyl-derivate