MA28688B1 - Procede d'une nouvelle amidation tres selective - Google Patents
Procede d'une nouvelle amidation tres selectiveInfo
- Publication number
- MA28688B1 MA28688B1 MA29572A MA29572A MA28688B1 MA 28688 B1 MA28688 B1 MA 28688B1 MA 29572 A MA29572 A MA 29572A MA 29572 A MA29572 A MA 29572A MA 28688 B1 MA28688 B1 MA 28688B1
- Authority
- MA
- Morocco
- Prior art keywords
- carboxylic acid
- carboxyl group
- new
- aliphatic cyclic
- reacting
- Prior art date
Links
- 230000009435 amidation Effects 0.000 title 1
- 238000007112 amidation reaction Methods 0.000 title 1
- 238000000034 method Methods 0.000 title 1
- -1 aliphatic cyclic carboxamide Chemical class 0.000 abstract 3
- 125000003178 carboxy group Chemical group [H]OC(*)=O 0.000 abstract 3
- 150000001244 carboxylic acid anhydrides Chemical class 0.000 abstract 1
- 150000001732 carboxylic acid derivatives Chemical class 0.000 abstract 1
- 238000006243 chemical reaction Methods 0.000 abstract 1
- 239000003795 chemical substances by application Substances 0.000 abstract 1
- 230000032050 esterification Effects 0.000 abstract 1
- 238000005886 esterification reaction Methods 0.000 abstract 1
- 125000000524 functional group Chemical group 0.000 abstract 1
- 238000004519 manufacturing process Methods 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D267/00—Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one oxygen atom as the only ring hetero atoms
- C07D267/02—Seven-membered rings
- C07D267/08—Seven-membered rings having the hetero atoms in positions 1 and 4
- C07D267/12—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
- C07D267/14—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems condensed with one six-membered ring
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Engineering & Computer Science (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Physical Education & Sports Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Plural Heterocyclic Compounds (AREA)
- Peptides Or Proteins (AREA)
- Hydrogenated Pyridines (AREA)
Abstract
La présente invention divulgue un procédé industriel court de production, à rendement élevé, d'un carboxamide cyclique aliphatique ayant un groupe carboxyle, qui consiste à faire réagir sélectivement un groupe fonctionnel en utilisant un agent de condensation non coûteux sans protéger le groupe carboxyle par estérification, c'est-à-dire en faisant réagir un anhydride d'acide carboxylique, obtenu par la réaction d'un acide carboxylique et d'un halogénure d'acide carboxylique tertiaire, avec une amine secondaire cyclique aliphatique ayant un groupe carboxyle.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2004174417 | 2004-06-11 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MA28688B1 true MA28688B1 (fr) | 2007-06-01 |
Family
ID=34970324
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MA29572A MA28688B1 (fr) | 2004-06-11 | 2006-12-28 | Procede d'une nouvelle amidation tres selective |
Country Status (16)
| Country | Link |
|---|---|
| US (1) | US20070238721A1 (fr) |
| EP (1) | EP1753752A1 (fr) |
| JP (1) | JP2008501629A (fr) |
| CN (1) | CN101001854A (fr) |
| AU (1) | AU2005252111A1 (fr) |
| BR (1) | BRPI0511877A (fr) |
| CA (1) | CA2569686A1 (fr) |
| CR (1) | CR8803A (fr) |
| IL (1) | IL179308A0 (fr) |
| MA (1) | MA28688B1 (fr) |
| MX (1) | MXPA06014152A (fr) |
| NO (1) | NO20070123L (fr) |
| RU (1) | RU2006147285A (fr) |
| TW (1) | TW200604187A (fr) |
| WO (1) | WO2005121133A1 (fr) |
| ZA (1) | ZA200609972B (fr) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2009108700A1 (fr) | 2008-02-25 | 2009-09-03 | Sixpoint Materials, Inc. | Procédé de production de tranches de nitrure du groupe iii et tranches de nitrure du groupe iii |
| DE102008054612A1 (de) * | 2008-12-15 | 2010-06-17 | Evonik Röhm Gmbh | Verfahren zur Herstellung von N-Isopropyl(meth)acrylamid |
| TWI774767B (zh) * | 2017-05-12 | 2022-08-21 | 瑞士商多蒂孔股份有限公司 | 茚烷衍生物及其在有機電子產品的用途 |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB2140003A (en) * | 1983-04-13 | 1984-11-21 | Shell Int Research | Azetidine derivatives suitable for inducing male sterility in plants |
| JP3479796B2 (ja) * | 1995-09-13 | 2003-12-15 | 武田薬品工業株式会社 | ベンゾオキサゼピン化合物 |
| PT862562E (pt) * | 1995-09-13 | 2001-11-30 | Takeda Chemical Industries Ltd | Compostos de benzoxazepina sua producao e utilizacao como agentes para reducao dos niveis de lipidos |
| WO2002038180A1 (fr) * | 2000-11-09 | 2002-05-16 | Takeda Chemical Industries, Ltd. | Agent haute densite faisant monter le taux de lipoproteine-cholesterol |
| JP4138299B2 (ja) * | 2000-11-09 | 2008-08-27 | 武田薬品工業株式会社 | 高密度リポタンパク−コレステロール上昇剤 |
| DE60106497D1 (de) * | 2001-04-30 | 2004-11-18 | Lupin Lab Ltd | Ein verfahren zur herstellung von natrium fosinopril |
-
2005
- 2005-06-10 BR BRPI0511877-8A patent/BRPI0511877A/pt not_active IP Right Cessation
- 2005-06-10 US US11/628,906 patent/US20070238721A1/en not_active Abandoned
- 2005-06-10 CA CA002569686A patent/CA2569686A1/fr not_active Abandoned
- 2005-06-10 EP EP05751255A patent/EP1753752A1/fr not_active Withdrawn
- 2005-06-10 TW TW094119234A patent/TW200604187A/zh unknown
- 2005-06-10 CN CNA2005800268866A patent/CN101001854A/zh active Pending
- 2005-06-10 WO PCT/JP2005/011091 patent/WO2005121133A1/fr not_active Ceased
- 2005-06-10 ZA ZA200609972A patent/ZA200609972B/en unknown
- 2005-06-10 AU AU2005252111A patent/AU2005252111A1/en not_active Abandoned
- 2005-06-10 MX MXPA06014152A patent/MXPA06014152A/es not_active Application Discontinuation
- 2005-06-10 RU RU2006147285/04A patent/RU2006147285A/ru not_active Application Discontinuation
- 2005-06-10 JP JP2006549745A patent/JP2008501629A/ja active Pending
-
2006
- 2006-11-15 IL IL179308A patent/IL179308A0/en unknown
- 2006-12-11 CR CR8803A patent/CR8803A/es not_active Application Discontinuation
- 2006-12-28 MA MA29572A patent/MA28688B1/fr unknown
-
2007
- 2007-01-08 NO NO20070123A patent/NO20070123L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| MXPA06014152A (es) | 2007-01-29 |
| CR8803A (es) | 2007-04-20 |
| BRPI0511877A (pt) | 2008-01-15 |
| JP2008501629A (ja) | 2008-01-24 |
| ZA200609972B (en) | 2008-08-27 |
| WO2005121133A1 (fr) | 2005-12-22 |
| US20070238721A1 (en) | 2007-10-11 |
| CN101001854A (zh) | 2007-07-18 |
| IL179308A0 (en) | 2007-03-08 |
| TW200604187A (en) | 2006-02-01 |
| AU2005252111A1 (en) | 2005-12-22 |
| CA2569686A1 (fr) | 2005-12-22 |
| RU2006147285A (ru) | 2008-07-20 |
| NO20070123L (no) | 2007-03-07 |
| EP1753752A1 (fr) | 2007-02-21 |
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