MA30406B1 - Nouveaux composes - Google Patents

Nouveaux composes

Info

Publication number
MA30406B1
MA30406B1 MA31371A MA31371A MA30406B1 MA 30406 B1 MA30406 B1 MA 30406B1 MA 31371 A MA31371 A MA 31371A MA 31371 A MA31371 A MA 31371A MA 30406 B1 MA30406 B1 MA 30406B1
Authority
MA
Morocco
Prior art keywords
new compounds
compounds
inflammations
medicament
manufacture
Prior art date
Application number
MA31371A
Other languages
English (en)
Inventor
Keith Biggadike
Anthony William James Cooper
David House
Iain Mcfarlane Mclay
Grahame Robert Woollam
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB0607840A external-priority patent/GB0607840D0/en
Priority claimed from GB0620382A external-priority patent/GB0620382D0/en
Priority claimed from GB0706516A external-priority patent/GB0706516D0/en
Priority claimed from GB0706515A external-priority patent/GB0706515D0/en
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of MA30406B1 publication Critical patent/MA30406B1/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/10—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing aromatic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4409—Non condensed pyridines; Hydrogenated derivatives thereof only substituted in position 4, e.g. isoniazid, iproniazid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/02—Nasal agents, e.g. decongestants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/04—Antipruritics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/38—Drugs for disorders of the endocrine system of the suprarenal hormones
    • A61P5/44—Glucocorticosteroids; Drugs increasing or potentiating the activity of glucocorticosteroids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/54—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
    • C07D231/56—Benzopyrazoles; Hydrogenated benzopyrazoles

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pulmonology (AREA)
  • Dermatology (AREA)
  • Pain & Pain Management (AREA)
  • Immunology (AREA)
  • Diabetes (AREA)
  • Rheumatology (AREA)
  • Endocrinology (AREA)
  • Otolaryngology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicinal Preparation (AREA)

Abstract

La présente invention concerne des composés de formule (I) : des compositions pharmaceutiques comprenant les composés et l'emploi des composés dans la fabrication d'un médicament, en particulier pour le traitement des inflammations et/ou des états allergiques.
MA31371A 2006-04-20 2008-11-10 Nouveaux composes MA30406B1 (fr)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
GB0607840A GB0607840D0 (en) 2006-04-20 2006-04-20 Novel compounds
GB0620382A GB0620382D0 (en) 2006-10-13 2006-10-13 Novel compounds
GB0706516A GB0706516D0 (en) 2007-04-03 2007-04-03 Novel compounds
GB0706515A GB0706515D0 (en) 2007-04-03 2007-04-03 Novel compounds

Publications (1)

Publication Number Publication Date
MA30406B1 true MA30406B1 (fr) 2009-05-04

Family

ID=38093410

Family Applications (1)

Application Number Title Priority Date Filing Date
MA31371A MA30406B1 (fr) 2006-04-20 2008-11-10 Nouveaux composes

Country Status (17)

Country Link
US (2) US7943651B2 (fr)
EP (1) EP2013185B1 (fr)
JP (1) JP5298008B2 (fr)
KR (1) KR20090003349A (fr)
AR (1) AR060536A1 (fr)
AU (1) AU2007242851A1 (fr)
BR (1) BRPI0710240A2 (fr)
CA (1) CA2649509A1 (fr)
CR (1) CR10353A (fr)
EA (1) EA200801997A1 (fr)
ES (1) ES2388351T3 (fr)
MA (1) MA30406B1 (fr)
MX (1) MX2008013411A (fr)
NO (1) NO20084328L (fr)
PE (1) PE20071227A1 (fr)
TW (1) TW200811111A (fr)
WO (1) WO2007122165A1 (fr)

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GB0724254D0 (en) * 2007-12-12 2008-01-23 Glaxo Group Ltd Novel compounds
TWI445705B (zh) 2008-05-20 2014-07-21 Astrazeneca Ab 經苯基及苯并二基取代之吲唑衍生物
WO2009142568A1 (fr) * 2008-05-20 2009-11-26 Astrazeneca Ab Combinaison de (a) modulateurs des récepteurs des glucocorticoïdes et (b) d’un agoniste β2
BRPI0912267A2 (pt) 2008-05-23 2015-10-13 Amira Pharmaceuticals Inc sal farmaceuticamente aceitável, composição farmacêutica, artigo de fabricação, métodos para tratar asma, rinite alérgica, doença, lesões gástricas e dor, métodos para prevenir broncoconstrição e rinite alérgica, uso de um sal farmaceuticamente aceitável, e, processo para a preparação de um sal farmaceuticamente aceitável.
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PL2897589T3 (pl) * 2013-11-22 2018-06-29 Teva Branded Pharmaceutical Products R & D, Inc. Lek do inhalacji
TW201625247A (zh) 2014-05-12 2016-07-16 葛蘭素史密斯克藍智慧財產權有限公司 用於治療傳染性疾病之醫藥組合物
AU2018387793A1 (en) 2017-12-18 2020-07-30 Grünenthal GmbH Substituted pyrrolidine amides I
TW201927769A (zh) 2017-12-18 2019-07-16 德商歌林達有限公司 經取代之吡咯啶醯胺ｉｉ
TWI827785B (zh) 2019-01-11 2024-01-01 德商歌林達有限公司 經取代的吡咯啶醯胺iii
ES2946888T3 (es) 2019-06-19 2023-07-27 Gruenenthal Gmbh Pirrolidina-amidas sustituidas IV
WO2020254552A2 (fr) 2019-06-19 2020-12-24 Grünenthal GmbH Amides de pyrrolidine substitués v
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MX2008013411A (es) 2008-11-04
EP2013185B1 (fr) 2012-05-30
US8178573B2 (en) 2012-05-15
PE20071227A1 (es) 2008-02-18
CA2649509A1 (fr) 2007-11-01
AR060536A1 (es) 2008-06-25
US20090111866A1 (en) 2009-04-30
ES2388351T3 (es) 2012-10-11
BRPI0710240A2 (pt) 2011-08-09
WO2007122165A1 (fr) 2007-11-01
JP2009534353A (ja) 2009-09-24
AU2007242851A1 (en) 2007-11-01
KR20090003349A (ko) 2009-01-09
EA200801997A1 (ru) 2009-04-28
CR10353A (es) 2009-01-09
NO20084328L (no) 2008-11-18
US20070265326A1 (en) 2007-11-15
JP5298008B2 (ja) 2013-09-25
US7943651B2 (en) 2011-05-17
TW200811111A (en) 2008-03-01

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